中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共4条,第1-4条 帮助

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Identification of methyl (5-(6-((4-(methylsulfonyl)piperazin-1-yl)methyl)-4-morpholinopyrrolo[2,1-f][1,2,4]triazin-2-yl)-4-(trifluoromethyl)pyridin-2-yl)carbamate (CYH33) as an orally bioavailable, highly potent, PI3K alpha inhibitor for the treatment of advanced solid tumors 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 209, 页码: 10
作者:  
Xiang, Hao-Yue;  Wang, Xiang;  Chen, Yan-Hong;  Zhang, Xi;  Tan, Cun
  |  收藏  |  浏览/下载:22/0  |  提交时间:2021/05/24
Design, synthesis and antiproliferative activity evaluation of a series of pyrrolo [2,1-f] [1,2,4] triazine derivatives 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2020, 卷号: 30, 期号: 12, 页码: 4
作者:  
Xiang, Hao-Yue;  Chen, Yan-Hong;  Wang, Yi;  Zhang, Xi;  Ding, Jian
  |  收藏  |  浏览/下载:27/0  |  提交时间:2020/07/01
Copper(II)-catalyzed cascade approach for the synthesis of pyrrolo[2,1-f][1,2,4]triazine-fused isoquinolines 期刊论文  OAI收割
RSC ADVANCES, 2014, 卷号: 4, 期号: 22, 页码: 11168-11175
作者:  
Chen, Jianyang;  Liu, Bo;  Chen, Yanhong;  He, Qian;  Yang, Chunhao
  |  收藏  |  浏览/下载:11/0  |  提交时间:2019/01/08
Studies of chirality effect of 4-(phenylamino)-pyrrolo[2,1-f][1,2,4]triazine on p38 alpha by molecular dynamics simulations and free energy calculations 期刊论文  iSwitch采集
Journal of computer-aided molecular design, 2009, 卷号: 23, 期号: 10, 页码: 737-745
作者:  
Chen, Quan;  Cui, Wei;  Ji, Mingjuan
收藏  |  浏览/下载:27/0  |  提交时间:2019/05/10