中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共547条,第1-10条 帮助

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Application of ensemble learning for predicting GABAA receptor agonists 期刊论文  OAI收割
COMPUTERS IN BIOLOGY AND MEDICINE, 2024, 卷号: 169, 页码: 13
作者:  
Xiao, Fu;  Ding, Xiaoyu;  Shi, Yan;  Wang, Dingyan;  Wang, Yitian
  |  收藏  |  浏览/下载:8/0  |  提交时间:2024/03/25
Discovery, Optimization, and Evaluation of Novel Pyridin-2(1H)-one Analogues as Potent TRK Inhibitors for Cancer Treatment 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 2, 页码: 1168-1183
作者:  
Xu, Zichao;  Peng, Xia;  Zhang, Renjie;  Ji, Yinchun;  You, Mengke
  |  收藏  |  浏览/下载:6/0  |  提交时间:2024/02/27
Structure-based development of potent and selective type-II kinase inhibitors of RIPK1 期刊论文  OAI收割
ACTA PHARMACEUTICA SINICA B, 2024, 卷号: 14, 期号: 1, 页码: 319-334
作者:  
Qin, Ying;  Li, Dekang;  Qi, Chunting;  Xiang, Huaijiang;  Meng, Huyan
  |  收藏  |  浏览/下载:1/0  |  提交时间:2024/03/06
Discovery of a novel GPR35 agonist with high and equipotent species potency for oral treatment of IBD 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2023, 卷号: 96, 页码: 12
作者:  
Song, Zhaoxiang;  Lu, Dan;  Sun, Jun;  Ye, Yangliang;  Fang, Jiahui
  |  收藏  |  浏览/下载:19/0  |  提交时间:2024/01/16
GPR35  IBD  Lodoxamide  
Circuit-specific gene therapy reverses core symptoms in a primate Parkinson's disease model 期刊论文  OAI收割
CELL, 2023, 卷号: 186, 期号: 24, 页码: 5394-+
作者:  
Chen, Yefei;  Hong, Zexuan;  Wang, Jingyi;  Liu, Kunlin;  Liu, Jing
  |  收藏  |  浏览/下载:5/0  |  提交时间:2024/01/26
TI17, a novel compound, exerts anti-MM activity by impairing Trip13 function of DSBs repair and enhancing DNA damage 期刊论文  OAI收割
CANCER MEDICINE, 2023, 页码: 14
作者:  
Chang, Shuaikang;  Xiao, Wenqin;  Xie, Yongsheng;  Xu, Zhijian;  Li, Bo
  |  收藏  |  浏览/下载:4/0  |  提交时间:2023/12/11
The anticancer potential of chemical constituents of Moringa oleifera targeting CDK-2 inhibition in estrogen receptor positive breast cancer using in-silico and in vitro approches 期刊论文  OAI收割
BMC COMPLEMENTARY MEDICINE AND THERAPIES, 2023, 卷号: 23, 期号: 1, 页码: 17
作者:  
Sultan, Rida;  Ahmed, Abrar;  Wei, Li;  Saeed, Hamid;  Islam, Muhammad
  |  收藏  |  浏览/下载:6/0  |  提交时间:2023/12/19
Tetrandrine synergizes with MAPK inhibitors in treating KRAS-mutant pancreatic ductal adenocarcinoma via collaboratively modulating the TRAIL-death receptor axis 期刊论文  OAI收割
PHARMACOLOGICAL RESEARCH, 2023, 卷号: 197, 页码: 12
作者:  
Tang, Shuai;  Duan, Yichen;  Yuan, Tao;  Hu, Yutinh;  Yuan, Liang
  |  收藏  |  浏览/下载:5/0  |  提交时间:2023/12/11
Hyodeoxycholic acid alleviates non-alcoholic fatty liver disease through modulating the gut-liver axis 期刊论文  OAI收割
CELL METABOLISM, 2023, 卷号: 35, 期号: 10, 页码: 1752-+
作者:  
Kuang, Junliang;  Wang, Jieyi;  Li, Yitao;  Li, Mengci;  Zhao, Mingliang
  |  收藏  |  浏览/下载:4/0  |  提交时间:2023/12/08
AhR-STAT3-HO-1/COX-2 signalling pathway may restrict ferroptosis and improve hMSC accumulation and efficacy in mouse liver 期刊论文  OAI收割
BRITISH JOURNAL OF PHARMACOLOGY, 2023, 页码: 17
作者:  
Han, Li;  Ma, Chenhui;  Wu, Zhitao;  Xu, Huiming;  Li, Hai
  |  收藏  |  浏览/下载:4/0  |  提交时间:2023/12/08