中国科学院机构知识库网格
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Construction of a myoglobin scaffold-based biocatalyst for the biodegradation of sulfadiazine and sulfathiazole
期刊论文
OAI收割
JOURNAL OF HAZARDOUS MATERIALS, 2024, 卷号: 465, 页码: 10
作者:
Zhang, Weikang
;
Lin, Yingwu
;
Meng, Xiangmin
;
Wang, Qiaoning
;
Chen, Lingxin
  |  
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2024/01/26
Sulfonamides
Myoglobin
Biocatalysis
Biodegradation
Directed evolution
Discovery of a 1,6-naphthyridin-4-one-based AXL inhibitor with improved pharmacokinetics and enhanced in vivo antitumor efficacy
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 265, 页码: 17
作者:
Lan, Yaohan
;
Peng, Xia
;
Ji, Yinchun
;
Su, Yi
;
Duan, Wenhu
  |  
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2024/02/27
AXL inhibitor
In vivo antitumor efficacy
6-Naphthyridin-4-one derivatives
Scaffold hopping
Structure-based drug design
Synthesis of 2-amino-9
H
-chromeno[2,3-
d
]thiazol-9-ones with anti-inflammatory activity
via
cascade reactions of 2-amino-3 iodochromones with amines and carbon disulfide
期刊论文
OAI收割
RSC ADVANCES, 2024, 卷号: 14, 期号: 5, 页码: 3158-3162
作者:
Tan, Jiangtao
;
He, Yifan
;
Lin, Yu
;
Zhong, Yuanchen
;
He, Shijun
  |  
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2024/02/27
Discovery, Optimization, and Evaluation of Novel Pyridin-2(1
H
)-one Analogues as Potent TRK Inhibitors for Cancer Treatment
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 2, 页码: 1168-1183
作者:
Xu, Zichao
;
Peng, Xia
;
Zhang, Renjie
;
Ji, Yinchun
;
You, Mengke
  |  
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2024/02/27
Discovery of JN122, a Spiroindoline-Containing Molecule that Inhibits MDM2/p53 Protein-Protein Interaction and Exerts Robust In Vivo Antitumor Efficacy
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 66, 期号: 24, 页码: 16991-17025
作者:
Cheng, Jing
;
Yan, Ziqin
;
Jiang, Kailong
;
Liu, Chen
;
Xu, Dehua
  |  
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2024/02/19
Structure-based drug discovery of novel fused- pyrazolone carboxamide derivatives as potent and selective AXL inhibitors
期刊论文
OAI收割
ACTA PHARMACEUTICA SINICA B, 2023, 卷号: 13, 期号: 12, 页码: 4918-4933
作者:
Fang, Feifei
;
Dai, Yang
;
Wang, Hao
;
Ji, Yinchun
;
Liang, Xuewu
  |  
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2024/01/26
derivatives
Antitumor drug development
Potential AXL inhibitor
Antitumor activity
Structure-based drug design
Fused-pyrazolone carboxamide
Discovery of PVD-06 as a Subtype-Selective and Efficient PTPN2 Degrader
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 66, 期号: 22, 页码: 15269-15287
作者:
Hu, Linghao
;
Li, Huiyun
;
Qin, Junlin
;
Yang, Dan
;
Liu, Jieming
  |  
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2024/02/27
Discovery of a highly potent NPAS3 heterodimer inhibitor by covalently modifying ARNT
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2023, 卷号: 139, 页码: 10
作者:
Li, Peizhuo
;
Tian, Yucheng
;
Shang, Qinghong
;
Tang, Cailing
;
Hou, Zeng
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2023/10/17
NPAS3
Covalent inhibitor
Protein -protein interaction
5-nitrothiazole warhead
LINC00955 suppresses colorectal cancer growth by acting as a molecular scaffold of TRIM25 and Sp1 to Inhibit DNMT3B-mediated methylation of the PHIP promoter
期刊论文
OAI收割
BMC CANCER, 2023, 卷号: 23, 期号: 1, 页码: 20
作者:
Ren, Ganglin
;
Li, Hongyan
;
Hong, Dan
;
Hu, Fangyu
;
Jin, Rongjia
  |  
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2023/12/08
LINC00955
Colorectal cancer
Cell cycle
CDK2
PHIP
Sp1
A first genome survey sequencing of alvinocaridid shrimp Shinkaicaris leurokolos in deep-sea hydrothermal vent environment
期刊论文
OAI收割
JOURNAL OF THE MARINE BIOLOGICAL ASSOCIATION OF THE UNITED KINGDOM, 2023, 卷号: 103, 页码: 8
作者:
Wang, Aiyang
;
Cheng, Jiao
;
Xin, Qian
;
Sha, Zhongli
;
Hui, Min
  |  
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2023/12/13
genome survey
hydrothermal vent
microsatellite DNA
mitogenome
Shinkaicaris leurokolos