中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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期刊论文 [236]
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Discovery and optimization of thieno[3,2-d]pyrimidine derivatives as highly selective inhibitors of cyclin-dependent kinase 7
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 263, 页码: 21
作者:
Zhang, Hongjin
;
Lin, Guohao
;
Jia, Suyun
;
Zhang, Ying
;
Wu, Jianbo
  |  
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2024/01/26
Thieno[3
d ]pyrimidine derivative
Cyclin-dependent kinase 7
Small molecule inhibitor
Kinome selectivity
Triple negative breast cancer
Novel thieno[2,3-b]quinoline-procaine hybrid molecules: A new class of allosteric SHP-1 activators evolved from PTP1B inhibitors
期刊论文
OAI收割
CHINESE CHEMICAL LETTERS, 2023, 卷号: 34, 期号: 8, 页码: 6
作者:
Xu, Lei
;
Xuyan, Xuyang
;
Minmi, Minmin
;
Wang, Zhiji
;
Shee, Chao
  |  
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2023/10/17
Activator
PTPs
Inhibitor
Thieno[2
b ]quinoline derivatives
Diffuse large B-cell lymphoma
Discovery of novel Thieno[2,3-d]imidazole derivatives as agonists of human STING for antitumor immunotherapy using systemic administration
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 238, 页码: 16
作者:
Niu, Jing
;
Bai, Hudagula
;
Li, Zizhou
;
Gao, Yuzhe
;
Zhang, Yan
  |  
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2022/08/16
STING
cGAS
Non-cyclic dinucleotides (non-CDNs)
Systemic administration
Antitumor immunotherapy
Discovery of Thieno[2,3-e]indazole Derivatives as Novel Oral Selective Estrogen Receptor Degraders with Highly Improved Antitumor Effect and Favorable Druggability br
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 65, 期号: 7, 页码: 5724-5750
作者:
Lu, Zhengyu
;
Cao, Yangzhi
;
Zhang, Dan
;
Meng, Xin
;
Guo, Bin
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2022/08/16
Chain Conformation and Liquid-Crystalline Structures of a Poly(thieno)thiophene
期刊论文
OAI收割
MACROMOLECULES, 2022, 卷号: 55, 期号: 7, 页码: 2892-2903
作者:
Liu, C
;
Yang, WH
;
Jiang, HQ
;
Zhang, BQ
;
Liu, GM
  |  
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2023/11/10
Investigation of charge transport of monolayer polymeric films with field effect tuning and molecular doping for chemiresistive sensing application
期刊论文
OAI收割
ORGANIC ELECTRONICS, 2021, 卷号: 96
作者:
Zhou, Zheng
;
Wang, Jiawei
;
Xiao, Shaozhu
;
Jiang, Wenfeng
;
Lu, Congyan
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2021/12/01
EFFECT TRANSISTORS
CONDUCTING POLYMERS
UNIVERSAL CROSSOVER
MOBILITY
PERFORMANCE
SEMICONDUCTORS
MECHANISM
DRIVEN
Investigation of charge transport of monolayer polymeric films with field effect tuning and molecular doping for chemiresistive sensing application
期刊论文
OAI收割
ORGANIC ELECTRONICS, 2021, 卷号: 96
作者:
Zhou, Zheng
;
Wang, Jiawei
;
Xiao, Shaozhu
;
Jiang, Wenfeng
;
Lu, Congyan
  |  
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2021/12/01
EFFECT TRANSISTORS
CONDUCTING POLYMERS
UNIVERSAL CROSSOVER
MOBILITY
PERFORMANCE
SEMICONDUCTORS
MECHANISM
DRIVEN
Straightforward synthesis, characterization, and cytotoxicity evaluation of hybrids of natural alkaloid evodiamine/rutaecarpine and thieno[2,3-d]pyrimidinones
期刊论文
OAI收割
JOURNAL OF ASIAN NATURAL PRODUCTS RESEARCH, 2020, 卷号: 22, 期号: 1, 页码: 69-82
作者:
Nie, LF (Nie, Li-Fei)[ 1,2 ]
;
Wang, SS (Wang, Si-Si)[ 3 ]
;
Cao, JG (Cao, Jian-Guo)[ 3 ]
;
Liu, FZ (Liu, Fei-Ze)[ 1,2 ]
;
Xiamuxi, HBM (Xiamuxi, Hainimu)[ 1,2 ]
  |  
收藏
  |  
浏览/下载:154/0
  |  
提交时间:2020/01/15
Thieno[2
3-d]pyrimidinone
evodiamine
rutaecarpine
hybrid
cytotoxicity
Optimized Molecular Packing and Nonradiative Energy Loss Based on Terpolymer Methodology Combining Two Asymmetric Segments for High-Performance Polymer Solar Cells
期刊论文
OAI收割
ACS APPLIED MATERIALS & INTERFACES, 2020, 卷号: 12, 期号: 18, 页码: 20393-20403
作者:
Wang, XC
;
Han, JH
;
Huang, D
;
Wang, JN
;
Xie, Y
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2021/09/06
HIGH-EFFICIENCY
CHARGE SEPARATION
FULLERENE
ACCEPTOR
COPOLYMERS
MORPHOLOGY
STRATEGY
EVOLUTION
DYNAMICS
ENABLES
Design, synthesis, and biological evaluation of thieno[3,2-d]pyrimidine derivatives as potential simplified phosphatidylinositol 3-kinase alpha inhibitors
期刊论文
OAI收割
CHEMICAL BIOLOGY & DRUG DESIGN, 2019, 卷号: 94, 期号: 6, 页码: 2013-2022
作者:
Yang, Xiuyan
;
Deng, Meng
;
Zhang, Xi
;
Wang, Yi
;
Song, Kun
  |  
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2020/07/01
PI3K alpha inhibitors
proliferation inhibition
thieno[3
2-d]pyrimidine derivatives