中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [16]
水生生物研究所 [1]
武汉病毒研究所 [1]
昆明植物研究所 [1]
中国科学院大学 [1]
上海生物化学与细胞生... [1]
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OAI收割 [20]
iSwitch采集 [2]
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期刊论文 [22]
发表日期
2022 [2]
2021 [3]
2019 [1]
2018 [3]
2017 [1]
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学科主题
Biochemist... [1]
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The p300 Inhibitor A-485 Exerts Antitumor Activity in Growth Hormone Pituitary Adenoma
期刊论文
OAI收割
JOURNAL OF CLINICAL ENDOCRINOLOGY & METABOLISM, 2022, 页码: 10
作者:
Ji, Chenxing
;
Xu, Wen
;
Ding, Hong
;
Chen, Zhengyuan
;
Shi, Chengzhang
  |  
收藏
  |  
浏览/下载:34/0
  |  
提交时间:2022/06/15
p300
A-485
growth hormone pituitary adenoma
Repressing MYC by targeting BET synergizes with selective inhibition of PI3K alpha against B cell lymphoma
期刊论文
OAI收割
CANCER LETTERS, 2022, 卷号: 524, 页码: 206-218
作者:
Chen, Zi-qi
;
Cao, Zhe-rui
;
Wang, Yi
;
Zhang, Xi
;
Xu, Lan
  |  
收藏
  |  
浏览/下载:52/0
  |  
提交时间:2021/12/16
CYH33
MYC
P300
BET
B cell lymphoma
PI3K
Design, synthesis and biological evaluation of a novel spiro oxazolidinedione as potent p300/CBP HAT inhibitor for the treatment of ovarian cancer
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2021, 卷号: 52, 页码: 12
作者:
Ding, Hong
;
Pei, Yuan
;
Li, Yuanqing
;
Xu, Wen
;
Mei, Lianghe
  |  
收藏
  |  
浏览/下载:37/0
  |  
提交时间:2022/06/15
Epigenetics
Histone acetyltransferase
P300/CBP
Ovarian cancer
Targeting p300/CBP Attenuates Hepatocellular Carcinoma Progression through Epigenetic Regulation of Metabolism
期刊论文
OAI收割
CANCER RESEARCH, 2021, 卷号: 81, 期号: 4, 页码: 860-872
作者:
Cai, Ling-Yan
;
Chen, Shi-Jie
;
Xiao, Sen-Hao
;
Sun, Qin-Juan
;
Ding, Chen-Hong
  |  
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2024/03/21
SL010110, a lead compound, inhibits gluconeogenesis via SIRT2-p300-mediated PEPCK1 degradation and improves glucose homeostasis in diabetic mice
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 13
作者:
Ren, Yu-ran
;
Ye, Yang-liang
;
Feng, Ying
;
Xu, Ti-fei
;
Shen, Yu
  |  
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2021/05/24
SL010110
gluconeogenesis
primary mouse hepatocytes
PEPCK1
acetylation
degradation
p300/CBP inhibitor A-485 alleviates acute liver injury by regulating macrophage activation and polarization
期刊论文
OAI收割
THERANOSTICS, 2019, 卷号: 9, 期号: 26, 页码: 8344-8361
作者:
Peng, Jinjin
;
Li, Jiacheng
;
Huang, Jing
;
Xu, Pan
;
Huang, Heming
  |  
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2020/07/01
liver injury
inflammation
macrophages
epigenetics
acetyltransferase inhibitor
Discovery and biological evaluation of thiobarbituric derivatives as potent p300/CBP inhibitors
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2018, 卷号: 26, 期号: 20, 页码: 5397-5407
作者:
Lu, Wenchao
;
Xiong, Huan
;
Chen, Yu
;
Wang, Chen
;
Zhang, Hao
  |  
收藏
  |  
浏览/下载:137/0
  |  
提交时间:2019/01/08
Drug discovery
Epigenetics
Histone acetyltransferase
P300/CBP
Identification of novel inhibitors of histone acetyltransferase hMOF through high throughput screening
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 157, 页码: 867-876
作者:
Zhang, Rukang
;
Wang, Jiang
;
Zhao, Liang
;
Liu, Shien
;
Du, Daohai
  |  
收藏
  |  
浏览/下载:36/0
  |  
提交时间:2019/01/08
High throughput screening
Epigenetics
Histone acetyltransferase
MOF
Inhibitor
Discovery of 1,8-acridinedione derivatives as novel GCN5 inhibitors via high throughput screening
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 151, 页码: 740-751
作者:
Xiong, Huan
;
Han, Jie
;
Wang, Jun
;
Lu, Wenchao
;
Wang, Chen
  |  
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2019/01/08
Epigenetics
Histone acetyltransferase
GCN5
High throughput screening
1,8-Acridinedione derivative
Comparative Proteomic Analysis of Lysine Acetylation in Fish CIK Cells Infected with Aquareovirus
期刊论文
OAI收割
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 2017, 卷号: 18, 期号: 11, 页码: 21
作者:
Guo, Hong
;
Zhang, Jie
;
Wang, Yaping
;
Bu, Chen
;
Zhou, Yanyan
  |  
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2019/07/03
comparative proteomics
Ctenopharyngodon idella kidney cells
aquareovirus infection
lysine acetylation