中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
机构
采集方式
内容类型
发表日期
学科主题
筛选

浏览/检索结果: 共22条,第1-10条 帮助

条数/页: 排序方式:
The p300 Inhibitor A-485 Exerts Antitumor Activity in Growth Hormone Pituitary Adenoma 期刊论文  OAI收割
JOURNAL OF CLINICAL ENDOCRINOLOGY & METABOLISM, 2022, 页码: 10
作者:  
Ji, Chenxing;  Xu, Wen;  Ding, Hong;  Chen, Zhengyuan;  Shi, Chengzhang
  |  收藏  |  浏览/下载:34/0  |  提交时间:2022/06/15
Repressing MYC by targeting BET synergizes with selective inhibition of PI3K alpha against B cell lymphoma 期刊论文  OAI收割
CANCER LETTERS, 2022, 卷号: 524, 页码: 206-218
作者:  
Chen, Zi-qi;  Cao, Zhe-rui;  Wang, Yi;  Zhang, Xi;  Xu, Lan
  |  收藏  |  浏览/下载:52/0  |  提交时间:2021/12/16
CYH33  MYC  P300  BET  B cell lymphoma  PI3K  
Design, synthesis and biological evaluation of a novel spiro oxazolidinedione as potent p300/CBP HAT inhibitor for the treatment of ovarian cancer 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2021, 卷号: 52, 页码: 12
作者:  
Ding, Hong;  Pei, Yuan;  Li, Yuanqing;  Xu, Wen;  Mei, Lianghe
  |  收藏  |  浏览/下载:37/0  |  提交时间:2022/06/15
Targeting p300/CBP Attenuates Hepatocellular Carcinoma Progression through Epigenetic Regulation of Metabolism 期刊论文  OAI收割
CANCER RESEARCH, 2021, 卷号: 81, 期号: 4, 页码: 860-872
作者:  
Cai, Ling-Yan;  Chen, Shi-Jie;  Xiao, Sen-Hao;  Sun, Qin-Juan;  Ding, Chen-Hong
  |  收藏  |  浏览/下载:16/0  |  提交时间:2024/03/21
SL010110, a lead compound, inhibits gluconeogenesis via SIRT2-p300-mediated PEPCK1 degradation and improves glucose homeostasis in diabetic mice 期刊论文  OAI收割
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 13
作者:  
Ren, Yu-ran;  Ye, Yang-liang;  Feng, Ying;  Xu, Ti-fei;  Shen, Yu
  |  收藏  |  浏览/下载:26/0  |  提交时间:2021/05/24
p300/CBP inhibitor A-485 alleviates acute liver injury by regulating macrophage activation and polarization 期刊论文  OAI收割
THERANOSTICS, 2019, 卷号: 9, 期号: 26, 页码: 8344-8361
作者:  
Peng, Jinjin;  Li, Jiacheng;  Huang, Jing;  Xu, Pan;  Huang, Heming
  |  收藏  |  浏览/下载:28/0  |  提交时间:2020/07/01
Discovery and biological evaluation of thiobarbituric derivatives as potent p300/CBP inhibitors 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2018, 卷号: 26, 期号: 20, 页码: 5397-5407
作者:  
Lu, Wenchao;  Xiong, Huan;  Chen, Yu;  Wang, Chen;  Zhang, Hao
  |  收藏  |  浏览/下载:137/0  |  提交时间:2019/01/08
Identification of novel inhibitors of histone acetyltransferase hMOF through high throughput screening 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 157, 页码: 867-876
作者:  
Zhang, Rukang;  Wang, Jiang;  Zhao, Liang;  Liu, Shien;  Du, Daohai
  |  收藏  |  浏览/下载:36/0  |  提交时间:2019/01/08
Discovery of 1,8-acridinedione derivatives as novel GCN5 inhibitors via high throughput screening 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 151, 页码: 740-751
作者:  
Xiong, Huan;  Han, Jie;  Wang, Jun;  Lu, Wenchao;  Wang, Chen
  |  收藏  |  浏览/下载:27/0  |  提交时间:2019/01/08
Comparative Proteomic Analysis of Lysine Acetylation in Fish CIK Cells Infected with Aquareovirus 期刊论文  OAI收割
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 2017, 卷号: 18, 期号: 11, 页码: 21
作者:  
Guo, Hong;  Zhang, Jie;  Wang, Yaping;  Bu, Chen;  Zhou, Yanyan
  |  收藏  |  浏览/下载:25/0  |  提交时间:2019/07/03