中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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Structure-Activity Relationships of 2-(Arylthio)benzoic Acid FTO Inhibitors
期刊论文
OAI收割
ISRAEL JOURNAL OF CHEMISTRY, 2024, 页码: 13
作者:
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2024/03/25
RNA modification
m(6)A
FTO
anticancer
Novel imidazo[1,2,4] triazole derivatives: Synthesis, fluorescence, bioactivity for SHP1
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 265, 页码: 15
作者:
Yan, Xue
;
Zhang, Chun
;
Gao, Li-Xin
;
Liu, Min -Min
;
Yang, Yu-Ting
  |  
收藏
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浏览/下载:1/0
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提交时间:2024/02/27
Imidazo[124] triazole derivatives
Fluorescence property
SHP1
Bioactivity
Cellular imaging
High trophic level organisms and the complexity of soil micro-food webs at aggregate scale regulate carbon accumulation in cropland soils
期刊论文
OAI收割
AGRICULTURE ECOSYSTEMS & ENVIRONMENT, 2024, 卷号: 360, 页码: 13
作者:
Yao, Zhiyuan
;
Huang, Chuanxiong
;
Hu, Huiling
;
Wang, Tao
;
Li, Yulong
  |  
收藏
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浏览/下载:3/0
  |  
提交时间:2024/03/04
Soil biota
Organic fertilizer
Carbon sequestration
Sustainable agriculture
Soil quality
New chromone derivatives bearing thiazolidine-2,4-dione moiety as potent PTP1B inhibitors: Synthesis and biological activity evaluation
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2024, 卷号: 143, 页码: 9
作者:
Zheng, Yingying
;
Lu, Li
;
Li, Mengyue
;
Xu, Dehua
;
Zhang, Laishun
  |  
收藏
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浏览/下载:4/0
  |  
提交时间:2024/01/26
Chromone
Thiazolidine-2
4-dione
Protein tyrosine phosphatase 1B
Inhibitors
pH-responsive nanogels with enhanced antioxidant and antitumor activities on drug delivery and smart drug release
期刊论文
OAI收割
INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES, 2024, 卷号: 257, 页码: 16
作者:
Ma, Bing
;
Li, Qing
;
Mi, Yingqi
;
Zhang, Jingjing
;
Tan, Wenqiang
  |  
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2024/01/26
Benzimidazole-chitosan quaternary ammonium
salt
Nanogels
pH-responsive
Antioxidant activity
Antitumor activity
Design, synthesis and biological evaluation of betulinic acid derivatives as potential inhibitors of 3CL-protease of SARS-CoV-2
期刊论文
OAI收割
STEROIDS, 2024, 卷号: 202, 页码: 8
作者:
Liu, Yaowen
;
Nie, Tianqing
;
Hou, Jinjun
;
Long, Huali
;
Zhang, Zijia
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2024/03/13
3CLpro
SARS-CoV-2
Betulinic acid
Natural product
Inhibitory activity
Koilodenoids A-G, immunosuppressive spiro dimers of diterpenoids from
Koilodepas hainanense
: structural elucidation and biomimetic transformation
期刊论文
OAI收割
ORGANIC CHEMISTRY FRONTIERS, 2024, 页码: 8
作者:
Ren, Yu
;
Zheng, Cheng-Yu
;
Yao, Jia-Ying
;
He, Shi-Jun
;
Fan, Yao-Yue
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收藏
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浏览/下载:5/0
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提交时间:2024/03/06
Synthesis and Biological Evaluation of β-Lactam Derivatives Targeting Speckle-Type POZ Protein (SPOP)
期刊论文
OAI收割
ACS MEDICINAL CHEMISTRY LETTERS, 2024, 卷号: 15, 期号: 2, 页码: 270-279
作者:
Zhou, Chenmao
;
Hao, Xinyue
;
Chen, Zhengyang
;
Zhang, Runze
;
Zhou, Qian
  |  
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2024/03/13
Speckle-type POZ protein (SPOP)
SPOP inhibitors
Clear cell renal cell carcinoma (ccRCC)
Structure-activityrelationship (SAR)
Design, Synthesis, and Biological Evaluation of Potent and Selective PROTAC Degraders of Oncogenic KRAS
G12D
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 2, 页码: 1147-1167
作者:
Zhou, Chuan
;
Fan, Zisheng
;
Gu, Yuejiao
;
Ge, Zhiming
;
Tao, Zhaofan
  |  
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2024/02/27
Using the quantitative ion character-activity relationships (QICAR) model to predict the solid-liquid release of metals in soil
期刊论文
OAI收割
JOURNAL OF HAZARDOUS MATERIALS, 2024, 卷号: 461, 页码: 8
作者:
Shi, Wanyang
;
Wang, Xuedong
;
Yang, Junxing
;
Wang, Ying
;
Li, Mengjia
  |  
收藏
  |  
浏览/下载:62/0
  |  
提交时间:2023/11/06
Metal solid-liquid release
Ion character-activity
Bioavailability