中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共36条,第1-10条 帮助

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An LQT2-related mutation in the voltage-sensing domain is involved in switching the gating polarity of hERG 期刊论文  OAI收割
BMC BIOLOGY, 2024, 卷号: 22, 期号: 1, 页码: 14
作者:  
Liu, Zhipei;  Wang, Feng;  Yuan, Hui;  Tian, Fuyun;  Yang, Chuanyan
  |  收藏  |  浏览/下载:8/0  |  提交时间:2024/03/13
Discovery of 2-Aminopyrimidine Derivatives as Potent Dual FLT3/CHK1 Inhibitors with Significantly Reduced hERG Inhibitory Activities 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 页码: 23
作者:  
Li, Xuemei;  Wang, Peipei;  Wang, Chang;  Jin, Tingting;  Xu, Ran
  |  收藏  |  浏览/下载:13/0  |  提交时间:2023/10/17
Discovery of (S)-N-(2-Amino-4-fluorophenyl)-4-(1-(3-(4-((dimethylamino)methyl)phenyl)-6-oxopyridazin-1(6H)-yl)ethyl)benzamide as Potent Class I Selective HDAC Inhibitor for Oral Anticancer Drug Candidate 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 66, 期号: 10, 页码: 7016-7037
作者:  
Li, Daqiang;  Zhang, Zhuo;  Li, Yalei;  Wang, Xinyi;  Zhong, Hanyue
  |  收藏  |  浏览/下载:17/0  |  提交时间:2023/10/17
Molecular Determinants for the High-Affinity Blockade of Human Ether-a-go-go-Related Gene K+ Channel by Tolterodine 期刊论文  OAI收割
JOURNAL OF CARDIOVASCULAR PHARMACOLOGY, 2022, 卷号: 80, 期号: 5, 页码: 679-689
作者:  
Wang, Na;  Yang, Yang;  Wen, Jing;  Fan, Xin-Rong;  Li, Jian
  |  收藏  |  浏览/下载:24/0  |  提交时间:2022/12/13
Design, synthesis and biological evaluation of (R)-5-methylpyrrolidin-2-ones as p300 bromodomain inhibitors with Anti-Tumor activities in multiple tumor lines 期刊论文  OAI收割
BIOORGANIC CHEMISTRY, 2022, 卷号: 124, 页码: 15
作者:  
Liu, Ruiqi;  Yang, Hong;  Chen, Zonglong;  Zhou, Kaixin;  Shi, Qiongyu
  |  收藏  |  浏览/下载:36/0  |  提交时间:2022/08/16
The novel therapeutic strategy of vilazodone-donepezil chimeras as potent triple-target ligands for the potential treatment of Alzheimer's disease with comorbid depression 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 229, 页码: 22
作者:  
Li, Xiaokang;  Li, Jinwen;  Huang, Yunyuan;  Gong, Qi;  Fu, Yan
  |  收藏  |  浏览/下载:31/0  |  提交时间:2022/06/15
Characteristics of hERG and hNav1.5 channel blockade by sulcardine sulfate, a novel anti-arrhythmic compound 期刊论文  OAI收割
European journal of pharmacology, 2018, 卷号: 844, 页码: 130-138
作者:  
Chen, Weihai;  Gan, Lu;  Wang, Yiping
  |  收藏  |  浏览/下载:18/0  |  提交时间:2019/01/08
Synthesis and biological evaluation of a series of multi-target N-substituted cyclic imide derivatives with potential antipsychotic effect 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 145, 页码: 74-85
作者:  
Xu, Mingshuo;  Wang, Yu;  Yang, Feipu;  Wu, Chunhui;  Wang, Zhen
  |  收藏  |  浏览/下载:50/0  |  提交时间:2019/01/08
Machine Learning-Based Modeling of Drug Toxicity 期刊论文  OAI收割
Methods in molecular biology (Clifton, N.J.), 2018, 卷号: 1754, 页码: 247-264
作者:  
Lu, Jing;  Lu, Dong;  Fu, Zunyun;  Zheng, Mingyue;  Luo, Xiaomin
  |  收藏  |  浏览/下载:15/0  |  提交时间:2019/01/08
Identification of small-molecule ion channel modulators in C. elegans channelopathy models 期刊论文  OAI收割
NATURE COMMUNICATIONS, 2018, 卷号: 9, 期号: -, 页码: 3941
作者:  
Jiang, Qiang;  Li, Kai;  Chen, Xin;  Liu, Xi-Juan;  Yuan, Jie
  |  收藏  |  浏览/下载:10/0  |  提交时间:2020/12/09