中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
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上海药物研究所 [31]
化学研究所 [22]
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期刊论文 [142]
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生命有机化学 [5]
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Peroxymonosulfate Activation by Cu-OMS-2 Nanofibers for Efficient Degradation of N-Containing Heterocycles in Aquatic Solution
期刊论文
OAI收割
LANGMUIR, 2023, 卷号: 39, 期号: 47, 页码: 16954-16964
作者:
Chen, Yongxin
;
Yang, Zihan
;
Cui, Jun
;
Wu, Yingqin
;
Zhang, Xilong
  |  
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2024/01/02
Exploration of novel four-membered-heterocycle constructed peptidyl proteasome inhibitors with improved metabolic stability for cancer treatment
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2023, 卷号: 138, 页码: 22
作者:
Wang, Hanlin
;
Wu, Zhaoxiao
;
Cao, Yu
;
Gao, Lixin
;
Shao, Jiaan
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2023/10/17
Metabolic stability
Four-membered heterocycles
Proteasome inhibitors
Multiple myeloma
Privileged heterocycles for DNA-encoded library design and hit-to-lead optimization
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 248, 页码: 26
作者:
Wen, Xin
;
Wu, Xinyuan
;
Jin, Rui
;
Lu, Xiaojie
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2023/04/10
DNA Encoded library
Drug discovery
Heterocycles
Hit identification
Lead generation
Comparative Study on Pyrolysis Kinetics Behavior and High-Temperature Fast Pyrolysis Product Analysis of Coastal Zone and Land Biomasses
期刊论文
OAI收割
ACS OMEGA, 2022, 卷号: 7, 期号: 12, 页码: 10144-10155
作者:
Li, Jie
;
Shang, Yanchao
;
Wei, Wei
;
Liu, Zhengyi
;
Qiao, Yingyun
  |  
收藏
  |  
浏览/下载:31/0
  |  
提交时间:2022/08/10
Synthesis and Protein Tyrosine Phosphatase 1B (PTP1B) Inhibitory Activity Evaluation of Novel N-Acylhydrazone Derivatives Containing Carbazole and Aromatic Ring/Aromatic Fused Heterocycle
期刊论文
OAI收割
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2021, 卷号: 41, 期号: 9, 页码: 3593-3607
作者:
Li Yingjun
;
Lin Ledi
;
Liu Jihong
;
Gao Lixin
;
Sheng Li
  |  
收藏
  |  
浏览/下载:42/0
  |  
提交时间:2021/12/01
PTP1B inhibitor
carbazole
N-actylhydrazone
synthesis
molecular docking
Investigating the property and strength of intermolecular interaction in saturated and unsaturated cyclic cations constructed ionic liquids
期刊论文
OAI收割
Journal of Molecular Liquids, 2021, 卷号: 335
作者:
Zhang, Tao
;
Ding, Wei-Lu
;
Zhang, Yaqin
;
Bi, Kailun
;
Lu, Yumiao
  |  
收藏
  |  
浏览/下载:0/0
  |  
提交时间:2023/06/21
Density functional theory - Hydrogen bonds - Negative ions - Binding energy - Positive ions - Ionic strength - Molecular dynamics - Binding sites
DNA-encoded C-H functionality via photoredox-mediated hydrogen atom transformation catalysis
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2021, 卷号: 42, 页码: 4
作者:
Shan, Jinming
;
Ling, Xing
;
Liu, JiaXiang
;
Wang, Xuan
;
Lu, Xiaojie
  |  
收藏
  |  
浏览/下载:31/0
  |  
提交时间:2021/08/17
Photoredox
Hydrogen atom transfer
N-Boc saturated heterocycle
DNA Encoded Library (DEL)
Discovery of 5-(3-bromo-2-(2,3-dibromo-4,5-dimethoxybenzyl)-4,5-dimethoxybenzylidene)thiazolidine-2,4-dione as a novel potent protein tyrosine phosphatase 1B inhibitor with antidiabetic properties
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2021, 卷号: 108, 页码: 13
作者:
Jiang, Bo
;
Luo, Jiao
;
Guo, Shuju
;
Wang, Lijun
  |  
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2021/05/11
Type 2 diabetes mellitus
Protein tyrosine phosphatase 1B inhibitors
Thiazolidinedione
Insulin signaling
Anti-diabetic activities
Bisaspochalasins D and E: Two Heterocycle-Fused Cytochalasan Homodimers from an Endophytic Aspergillus flavipes
期刊论文
OAI收割
JOURNAL OF ORGANIC CHEMISTRY, 2021, 卷号: 86, 期号: 16, 页码: 11198-11205
作者:
Wang,Li
;
Yu,Zhiyin
;
Guo,Xiaowei
;
Huang,Jian-Ping
;
Yan,Yijun
  |  
收藏
  |  
浏览/下载:50/0
  |  
提交时间:2022/04/02
A-D
ALKALOIDS
MEROCYTOCHALASANS
BIOSYNTHESIS
SKELETON
DIMER
A deep insight into polybenzoxazole formation in the heterocycle-containing polybenzoxazine: An enlightening thought for smarter precursor design
期刊论文
OAI收割
POLYMER, 2021, 卷号: 226
作者:
Liu, Jingkai
;
Cao, Lijun
;
Dai, Jinyue
;
Peng, Yunyan
;
Liu, Xiaoqing
  |  
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2021/12/01
RING-OPENING POLYMERIZATION
BENZOXAZINE
CATALYST