中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共170条,第1-10条 帮助

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Synthesis and biological evaluation of pyrazole-fused oleanolic acid derivatives as novel inhibitors of inflammatory and osteoclast differentiation 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2023, 卷号: 80, 页码: 117177
作者:  
Yu, Yuanyuan;  Yuan, Wenlong;  Yuan, Jiaqi;  Wei, Wenhui;  He, Qian
  |  收藏  |  浏览/下载:4/0  |  提交时间:2024/03/27
Structure-based rational design enables efficient discovery of a new selective and potent AKT PROTAC degrader 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 238, 页码: 15
作者:  
Zhu, Cheng-Liang;  Luo, Xiaomin;  Tian, Tian;  Rao, Zijian;  Wang, Hanlin
  |  收藏  |  浏览/下载:28/0  |  提交时间:2022/08/16
Tailoring Multiple Sites of Metal-Organic Frameworks for Highly Efficient and Reversible Ammonia Adsorption 期刊论文  OAI收割
ACS APPLIED MATERIALS & INTERFACES, 2021, 卷号: 13, 期号: 47, 页码: 56025-56034
作者:  
Wang, Zhenzhen;  Li, Zhiyong;  Zhang, Xia-Guang;  Xia, Qingchun;  Wang, Huiyong
  |  收藏  |  浏览/下载:17/0  |  提交时间:2022/06/15
Synthesis and Biological Evaluation of C-17-Amino-Substituted Pyrazole-Fused Betulinic Acid Derivatives as Novel Agents for Osteoarthritis Treatment 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 18, 页码: 13676-13692
作者:  
Wang, Jie;  Wei, Wenhui;  Zhang, Xiaofei;  Cao, Shiqi;  Hu, Bintao
  |  收藏  |  浏览/下载:12/0  |  提交时间:2024/03/21
Design, synthesis, and biological evaluation of 4-benzoylamino-1H-pyrazole-3-carboxamide derivatives as potent CDK2 inhibitors 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 215, 页码: 12
作者:  
Lin, Tingting;  Li, Jiacheng;  Liu, Liping;  Li, Yuanqing;  Jiang, Hualiang
  |  收藏  |  浏览/下载:30/0  |  提交时间:2021/05/24
Synthetic Studies toward DNA-Encoded Heterocycles Based on the On-DNA Formation of alpha,beta-Unsaturated Ketones 期刊论文  OAI收割
ORGANIC LETTERS, 2021, 卷号: 23, 期号: 3, 页码: 908-913
作者:  
Liu, Sixiu;  Qi, Jingjing;  Lu, Weiwei;  Wang, Xuan;  Lu, Xiaojie
  |  收藏  |  浏览/下载:15/0  |  提交时间:2021/05/24
Electrochemical oxidation of acid orange 74 using Ru, IrO2, PbO2, and boron doped diamond anodes: Direct and indirect oxidation 期刊论文  OAI收割
JOURNAL OF ELECTROANALYTICAL CHEMISTRY, 2021, 卷号: 898
作者:  
Li, Aiyuan;  Weng, Jiaqi;  Yan, Xinmei;  Li, Hao;  Shi, Haibo
  |  收藏  |  浏览/下载:19/0  |  提交时间:2021/12/01
fDiscovery of pyrazole-thiophene derivatives as highly Potent, orally active Akt inhibitors 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 180, 页码: 72-85
作者:  
Zhan, Wenhu;  Che, Jinxin;  Xu, Lei;  Wu, Yizhe;  Hu, Xiaobei
  |  收藏  |  浏览/下载:20/0  |  提交时间:2020/07/01
Pd-Catalyzed intramolecular C-H activation and C-S formation to synthesize pyrazolo[5,1-b]benzothiazoles without an additional oxidant 期刊论文  OAI收割
ORGANIC CHEMISTRY FRONTIERS, 2019, 卷号: 6, 期号: 18, 页码: 3234-3237
作者:  
Peng, Yingyuan;  He, Qian;  Zhang, Xiaofei;  Yang, Chunhao
  |  收藏  |  浏览/下载:10/0  |  提交时间:2020/07/01
Discovery of 1,3-diphenyl-1H-pyrazole derivatives containing rhodanine-3-alkanoic acid groups as potential PTP1B inhibitors 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2019, 卷号: 29, 期号: 10, 页码: 1187-1193
作者:  
Sun, Liangpeng;  Wang, Peipei;  Xu, Lili;  Gao, Lixin;  Li, Jia
  |  收藏  |  浏览/下载:17/0  |  提交时间:2020/07/01