中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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  • 上海药物研究所 [841]
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Energy preservation for skeletal muscles: Shenqi Fuzheng injection prevents tissue wasting and restores bioenergetic profiles in a mouse model of chemotherapy-induced cachexia 期刊论文  OAI收割
PHYTOMEDICINE, 2024, 卷号: 125, 页码: 13
作者:  
Li, Wei;  Zhang, Zijia;  Berik, Entezar;  Liu, Yawen;  Pei, Wenqiang
  |  收藏  |  浏览/下载:15/0  |  提交时间:2024/04/09
PROTAC Prodrug-Integrated Nanosensitizer for Potentiating Radiation Therapy of Cancer 期刊论文  OAI收割
ADVANCED MATERIALS, 2024, 页码: 12
作者:  
Zhang, Shunan;  Lai, Yi;  Pan, Jiaxing;  Saeed, Madiha;  Li, Shiqin
  |  收藏  |  浏览/下载:13/0  |  提交时间:2024/04/09
DRAK2 suppresses autophagy by phosphorylating ULK1 at Ser56 to diminish pancreatic β cell function upon overnutrition 期刊论文  OAI收割
SCIENCE TRANSLATIONAL MEDICINE, 2024, 卷号: 16, 期号: 733, 页码: 16
作者:  
Lu, Yuting;  Xu, Junyu;  Li, Yufeng;  Wang, Ruoran;  Dai, Chengqiu
  |  收藏  |  浏览/下载:17/0  |  提交时间:2024/03/13
Discovery of Novel PROTAC Degraders of p300/CBP as Potential Therapeutics for Hepatocellular Carcinoma 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 4, 页码: 2466-2486
作者:  
Chang, Qi;  Li, Jiayi;  Deng, Yue;  Zhou, Ruilin;  Wang, Bingwei
  |  收藏  |  浏览/下载:13/0  |  提交时间:2024/03/25
Xuanbai Chengqi Decoction alleviates acute lung injury by inhibiting NLRP3 inflammasome 期刊论文  OAI收割
JOURNAL OF ETHNOPHARMACOLOGY, 2024, 卷号: 319, 页码: 13
作者:  
Wang, Shun;  Lin, Feifei;  Zhang, Chengxi;  Gao, Dan;  Qi, Zhuocao
  |  收藏  |  浏览/下载:11/0  |  提交时间:2023/12/08
Benzothiozinone derivatives with anti-tubercular Activity-Further side chain investigation 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 264, 页码: 11
作者:  
Wu, Xiaomei;  Wang, Wenxin;  Stelitano, Giovanni;  Riabova, Olga;  Wang, Bin
  |  收藏  |  浏览/下载:8/0  |  提交时间:2024/01/26
Discovery and exploration of novel somatostatin receptor subtype 5 (SSTR5) antagonists for the treatment of cholesterol gallstones 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 264, 页码: 16
作者:  
Han, Fanghui;  Zhao, Tingting;  Zhang, Yanglong;  Yun, Ying;  Xu, Yuanyuan
  |  收藏  |  浏览/下载:3/0  |  提交时间:2024/02/19
Design, Synthesis, and Biological Evaluation of Potent and Selective PROTAC Degraders of Oncogenic KRASG12D 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 2, 页码: 1147-1167
作者:  
Zhou, Chuan;  Fan, Zisheng;  Gu, Yuejiao;  Ge, Zhiming;  Tao, Zhaofan
  |  收藏  |  浏览/下载:10/0  |  提交时间:2024/02/27
Discovery and optimization of thieno[3,2-d]pyrimidine derivatives as highly selective inhibitors of cyclin-dependent kinase 7 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 263, 页码: 21
作者:  
Zhang, Hongjin;  Lin, Guohao;  Jia, Suyun;  Zhang, Ying;  Wu, Jianbo
  |  收藏  |  浏览/下载:5/0  |  提交时间:2024/01/26
Metabolite characterisation of the peptide-drug conjugate LN005 in liver S9s by UHPLC-Orbitrap-HRMS 期刊论文  OAI收割
XENOBIOTICA, 2024, 页码: 9
作者:  
Yuan, Yali;  Wang, Weiqiang;  Luo, Jing;  Tang, Chongzhuang;  Zheng, Yuandong
  |  收藏  |  浏览/下载:7/0  |  提交时间:2024/02/19