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Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [26]
采集方式
OAI收割 [26]
内容类型
期刊论文 [26]
发表日期
2024 [1]
2023 [8]
2022 [7]
2021 [2]
2019 [1]
2018 [1]
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共26条,第1-10条
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内容类型:期刊论文
专题:上海药物研究所
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Discovery of GPX4 inhibitors through FP-based high-throughput screening
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 265, 页码: 14
作者:
Cao, Yu
;
Wu, Bin
;
Xu, Ying
;
Wang, Mingchen
;
Wu, Xinyu
  |  
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Discovery of a novel OGT inhibitor through high-throughput screening based on Homogeneous Time-Resolved Fluorescence (HTRF)
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2023, 卷号: 139, 页码: 12
作者:
Wu, Xinyu
;
Wang, Mingchen
;
Cao, Yu
;
Xu, Ying
;
Yang, Ziqun
  |  
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  |  
Discovery of novel triazine derivatives as potent retinoic acid receptor-related orphan receptor gamma t (ROR gamma t) inverse agonists
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 256, 页码: 18
作者:
Lu, Lixue
;
Chen, Song
;
Yu, Mingcheng
;
Zhou, Ronghui
;
Guo, Siqi
  |  
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  |  
YTHDF2 inhibition potentiates radiotherapy antitumor efficacy
期刊论文
OAI收割
CANCER CELL, 2023, 卷号: 41, 期号: 7, 页码: 1294-+
作者:
Wang, Liangliang
;
Dou, Xiaoyang
;
Chen, Shijie
;
Yu, Xianbin
;
Huang, Xiaona
  |  
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RNAincoder: a deep learning-based encoder for RNA and RNA-associated interaction
期刊论文
OAI收割
NUCLEIC ACIDS RESEARCH, 2023, 页码: 11
作者:
Wang, Yunxia
;
Chen, Zhen
;
Pan, Ziqi
;
Huang, Shijie
;
Liu, Jin
  |  
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Optimization of carbazole carboxamide RORγt agonists: Challenges in improving the metabolic stability and maintaining the agonistic activity
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 251, 页码: 115213
作者:
Sun, Nannan
;
Yu, Mingcheng
;
Jiang, Zhengyuan
;
Yang, Feng
;
Lu, Lixue
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Discovery of new small molecule inhibitors of the BPTF bromodomain
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2023, 卷号: 134, 页码: 106453
作者:
Liang, Xiaochen
;
Cao, Yu
;
Duan, Zhe
;
Wang, Mingchen
;
Zhang, Naixia
  |  
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  |  
Selective PPAR gamma modulator diosmin improves insulin sensitivity and promotes browning of white fat
期刊论文
OAI收割
JOURNAL OF BIOLOGICAL CHEMISTRY, 2023, 卷号: 299, 期号: 4, 页码: 14
作者:
Yu, Jian
;
Hu, Yepeng
;
Sheng, Maozheng
;
Gao, Mingyuan
;
Guo, Wenxiu
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Cyclization strategy leads to highly potent Bromodomain and extra-terminal (BET) Bromodomain inhibitors for the treatment of acute liver injury
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 247, 页码: 13
作者:
Chen, Chao
;
Lu, Tian
;
Chen, Panyu
;
Li, Zizhou
;
Yang, Yaxi
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Design, synthesis, and biological evaluation of novel carbazole derivatives as potent DNMT1 inhibitors with reasonable PK properties
期刊论文
OAI收割
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, 2022, 卷号: 37, 期号: 1, 页码: 1537-1555
作者:
Li, Ennian
;
Wang, Kai
;
Zhang, Bei
;
Guo, Siqi
;
Xiao, Senhao
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