中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [202]
采集方式
OAI收割 [202]
内容类型
期刊论文 [197]
会议论文 [5]
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2024 [2]
2023 [24]
2022 [25]
2021 [19]
2020 [19]
2019 [18]
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Chemistry [3]
Biochemist... [2]
Pharmacolo... [2]
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浏览/检索结果:
共202条,第1-10条
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专题:上海药物研究所
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Discovery of hematopoietic progenitor kinase 1 inhibitors using machine learning-based screening and free energy perturbation
期刊论文
OAI收割
JOURNAL OF BIOMOLECULAR STRUCTURE & DYNAMICS, 2024, 页码: 13
作者:
Feng, Dazhi
;
Liu, Bo
;
Chen, Zhiwei
;
Xu, Jinyi
;
Geng, Meiyu
  |  
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2024/02/27
HPK1 inhibitor
machine learning
virtual screening
free energy perturbation
structural modification
Stachyose with effect on anti-angiogenic activity from Salvia yunnanensis
期刊论文
OAI收割
JOURNAL OF FUNCTIONAL FOODS, 2024, 卷号: 112, 页码: 10
作者:
Xu, Yangyang
;
He, Fei
;
Jin, Can
;
Su, Juan
;
Ding, Kan
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2024/03/25
Salvia yunnanensis
Stachyose
Anti-angiogenic activity
Galectin-3
Qing-Zhi-Tiao-Gan-Tang (QZTGT) prevents nonalcoholic steatohepatitis (NASH) by expression pattern correction
期刊论文
OAI收割
JOURNAL OF ETHNOPHARMACOLOGY, 2023, 卷号: 317, 页码: 14
作者:
Chu, Hang
;
Zhang, Weitao
;
Tan, Yan
;
Diao, Zhipeng
;
Li, Peng
  |  
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2023/10/17
Fibrosis
Inflammation
Lipogenesis
NASH
QZTGT
TMNP
C-terminal modification and functionalization of proteins via a self-cleavage tag triggered by a small molecule
期刊论文
OAI收割
NATURE COMMUNICATIONS, 2023, 卷号: 14, 期号: 1, 页码: 13
作者:
Zeng, Yue
;
Shi, Wei
;
Liu, Zhi
;
Xu, Hao
;
Liu, Liya
  |  
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2024/02/19
Discovery of zolinium TSG1180 as a novel agonist of transgelin-2 for treating asthma
期刊论文
OAI收割
Biomedicine & pharmacotherapy = Biomedecine & pharmacotherapie, 2023, 卷号: 167, 页码: 115556
作者:
Yuan, Hong-Kai
  |  
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2024/03/26
Active learning
Consensus labelling
Eye irritation
Serious eye damage
Structural alerts
Multiple heart-cutting two-dimensional liquid chromatography/charged aerosol detector assay of ginsenosides for quality evaluation of ginseng from diverse Chinese patent medicines
期刊论文
OAI收割
JOURNAL OF CHROMATOGRAPHY A, 2023, 卷号: 1708, 页码: 10
作者:
Xu, Xiao-yan
;
Jiang, Mei-ting
;
Wang, Yu
;
Sun, He
;
Jing, Qi
  |  
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2023/12/08
Multiple heart -cutting two-dimensional liquid
chromatography
Charged aerosol detector
Quantitative assay
Ginseng
Chinese patent medicine
Two new compounds from the Hainan Soft Corals Sinularia tumulosa and Sinularia depressa with their anti-inflammatory or cytotoxic activities
期刊论文
OAI收割
JOURNAL OF ASIAN NATURAL PRODUCTS RESEARCH, 2023, 卷号: 25, 期号: 10, 页码: 949-956
作者:
Xu, Ting
;
Yu, Dan-Dan
;
Su, Ming-Zhi
;
Yao, Li-Gong
;
Li, Song-Wei
  |  
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2024/03/27
Sinularia
marine natural product
anti-inflammatory activity
cytotoxicity
Otilonium Bromide acts as a selective USP28 inhibitor and exhibits cytotoxic activity against multiple human cancer cell lines
期刊论文
OAI收割
BIOCHEMICAL PHARMACOLOGY, 2023, 卷号: 215, 页码: 14
作者:
Xu, Zhuo
;
Wang, Hui
;
Meng, Qian
;
Ding, Yiluan
;
Zhu, Mengying
  |  
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2023/10/17
Otilonium Bromide
Deubiquitinase
USP28
Selective inhibitor
An unusual four-step cascade reaction for accessing furo[3,4-c]pyridine-1,4-diones via rhodium catalysis
期刊论文
OAI收割
ORGANIC CHEMISTRY FRONTIERS, 2023, 页码: 7
作者:
Li, Yidi
;
Xu, Huiying
;
Zhou, Zhi
;
Huang, Lin
;
Tang, Zhenhao
  |  
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2023/10/17
Preclinical Evaluation of 9MW2821, a Site-Specific Monomethyl Auristatin E-based Antibody-Drug Conjugate for Treatment of Nectin-4-expressing Cancers
期刊论文
OAI收割
MOLECULAR CANCER THERAPEUTICS, 2023, 卷号: 22, 期号: 8, 页码: 913-925
作者:
Zhou, Wei
;
Fang, Peng
;
Yu, Dongan
;
Ren, Hongyuan
;
You, Meng
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2023/10/17