中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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Structure-Based Design of Tetrahydroisoquinoline-7-carboxamides as Selective Discoidin Domain Receptor 1 (DDR1) Inhibitors 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 12, 页码: 5911-5916
Wang, Zhen; Bian, Huan; Bartual, Sergio G.; Du, Wenting; Luo, Jinfeng; Zhao, Hu; Zhang, Shasha; Mo, Cheng; Zhou, Yang; Xu, Yong; Tu, Zhengchao; Ren, Xiaomei; Lu, Xiaoyun; Brekken, Rolf A.; Yao, Libo; Bullock, Alex N.; Su, Jin; Ding, Ke
收藏  |  浏览/下载:50/0  |  提交时间:2016/12/16
Structure-Based Design of Tetrahydroisoquinoline-7-carboxamides as Selective Discoidin Domain Receptor 1 (DDR1) Inhibitors 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 12, 页码: 5911-5916
作者:  
Yao, Libo;  Ding, Ke;  Su, Jin;  Bullock, Alex N.;  Brekken, Rolf A.
  |  收藏  |  浏览/下载:32/0  |  提交时间:2018/12/13
Small-Molecule BET Inhibitors in Clinical and Preclinical Development and Their Therapeutic Potential 期刊论文  OAI收割
CURRENT TOPICS IN MEDICINAL CHEMISTRY, 2015, 卷号: 15, 期号: 8, 页码: 776-794
Yu, Lei; Wang, Zhen; Zhang, Zhang; Ren, Xiaomei; Lu, Xiaoyun; Ding, Ke
收藏  |  浏览/下载:25/0  |  提交时间:2016/12/16
Hybrid pyrimidine alkynyls inhibit the clinically resistance related Bcr-Abl(T315I) mutant 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2015, 卷号: 25, 期号: 17, 页码: 3458-3463
作者:  
Ding, Ke;  Pan, Xiaofeng;  Wang, Deping;  Zhuang, Xiaoxi;  Luo, Jingfeng
  |  收藏  |  浏览/下载:22/0  |  提交时间:2018/12/13
Small-Molecule BET Inhibitors in Clinical and Preclinical Development and Their Therapeutic Potential 期刊论文  OAI收割
CURRENT TOPICS IN MEDICINAL CHEMISTRY, 2015, 卷号: 15, 期号: 8, 页码: 776-794
作者:  
Wang, Zhen;  Zhang, Zhang;  Ren, Xiaomei;  Lu, Xiaoyun;  Ding, Ke
  |  收藏  |  浏览/下载:10/0  |  提交时间:2018/12/13
Hybrid pyrimidine alkynyls inhibit the clinically resistance related Bcr-Abl(T315I) mutant 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2015, 卷号: 25, 期号: 17, 页码: 3458-3463
Lu, Xiaoyun; Zhang, Zhang; Ren, Xiaomei; Pan, Xiaofeng; Wang, Deping; Zhuang, Xiaoxi; Luo, Jingfeng; Yu, Rongmin; Ding, Ke
收藏  |  浏览/下载:22/0  |  提交时间:2016/12/16
Identification of GZD824 as an Orally Bioavailable Inhibitor That Targets Phosphorylated and Nonphosphorylated Breakpoint Cluster Region-Abelson (Bcr-Abl) Kinase and Overcomes Clinically Acquired Mutation-Induced Resistance against Imatinib 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2013, 卷号: 56, 期号: 3
作者:  
Wang, Deping;  Feng, Yubing;  Zhuang, Xiaoxi;  Zhang, Fengxiang;  Liu, Jianqi
  |  收藏  |  浏览/下载:23/0  |  提交时间:2018/12/13
Identification of GZD824 as an Orally Bioavailable Inhibitor That Targets Phosphorylated and Nonphosphorylated Breakpoint Cluster Region-Abelson (Bcr-Abl) Kinase and Overcomes Clinically Acquired Mutation-Induced Resistance against Imatinib 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2013, 卷号: 56, 期号: 3
Ren, Xiaomei; Pan, Xiaofen; Zhang, Zhang; Wang, Deping; Lu, Xiaoyun; Li, Yupeng; Wen, Donghai; Long, Huoyou; Luo, Jinfeng; Feng, Yubing; Zhuang, Xiaoxi; Zhang, Fengxiang; Liu, Jianqi; Leng, Fang; Lang, Xingfen; Bai, Yang; She, Miaoqin; Tu, Zhengchao; Pan, Jingxuan; Ding, Ke
收藏  |  浏览/下载:23/0  |  提交时间:2016/12/16