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Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
广州生物医药与健康研... [8]
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OAI收割 [8]
内容类型
期刊论文 [8]
发表日期
2016 [2]
2015 [4]
2013 [2]
学科主题
Pharmacolo... [8]
Chemistry [2]
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学科主题:Pharmacology & Pharmacy
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Structure-Based Design of Tetrahydroisoquinoline-7-carboxamides as Selective Discoidin Domain Receptor 1 (DDR1) Inhibitors
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 12, 页码: 5911-5916
Wang, Zhen
;
Bian, Huan
;
Bartual, Sergio G.
;
Du, Wenting
;
Luo, Jinfeng
;
Zhao, Hu
;
Zhang, Shasha
;
Mo, Cheng
;
Zhou, Yang
;
Xu, Yong
;
Tu, Zhengchao
;
Ren, Xiaomei
;
Lu, Xiaoyun
;
Brekken, Rolf A.
;
Yao, Libo
;
Bullock, Alex N.
;
Su, Jin
;
Ding, Ke
收藏
  |  
浏览/下载:50/0
  |  
提交时间:2016/12/16
Structure-Based Design of Tetrahydroisoquinoline-7-carboxamides as Selective Discoidin Domain Receptor 1 (DDR1) Inhibitors
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 12, 页码: 5911-5916
作者:
Yao, Libo
;
Ding, Ke
;
Su, Jin
;
Bullock, Alex N.
;
Brekken, Rolf A.
  |  
收藏
  |  
浏览/下载:32/0
  |  
提交时间:2018/12/13
Small-Molecule BET Inhibitors in Clinical and Preclinical Development and Their Therapeutic Potential
期刊论文
OAI收割
CURRENT TOPICS IN MEDICINAL CHEMISTRY, 2015, 卷号: 15, 期号: 8, 页码: 776-794
Yu, Lei
;
Wang, Zhen
;
Zhang, Zhang
;
Ren, Xiaomei
;
Lu, Xiaoyun
;
Ding, Ke
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2016/12/16
Hybrid pyrimidine alkynyls inhibit the clinically resistance related Bcr-Abl(T315I) mutant
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2015, 卷号: 25, 期号: 17, 页码: 3458-3463
作者:
Ding, Ke
;
Pan, Xiaofeng
;
Wang, Deping
;
Zhuang, Xiaoxi
;
Luo, Jingfeng
  |  
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2018/12/13
Small-Molecule BET Inhibitors in Clinical and Preclinical Development and Their Therapeutic Potential
期刊论文
OAI收割
CURRENT TOPICS IN MEDICINAL CHEMISTRY, 2015, 卷号: 15, 期号: 8, 页码: 776-794
作者:
Wang, Zhen
;
Zhang, Zhang
;
Ren, Xiaomei
;
Lu, Xiaoyun
;
Ding, Ke
  |  
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2018/12/13
Hybrid pyrimidine alkynyls inhibit the clinically resistance related Bcr-Abl(T315I) mutant
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2015, 卷号: 25, 期号: 17, 页码: 3458-3463
Lu, Xiaoyun
;
Zhang, Zhang
;
Ren, Xiaomei
;
Pan, Xiaofeng
;
Wang, Deping
;
Zhuang, Xiaoxi
;
Luo, Jingfeng
;
Yu, Rongmin
;
Ding, Ke
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2016/12/16
Identification of GZD824 as an Orally Bioavailable Inhibitor That Targets Phosphorylated and Nonphosphorylated Breakpoint Cluster Region-Abelson (Bcr-Abl) Kinase and Overcomes Clinically Acquired Mutation-Induced Resistance against Imatinib
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2013, 卷号: 56, 期号: 3
作者:
Wang, Deping
;
Feng, Yubing
;
Zhuang, Xiaoxi
;
Zhang, Fengxiang
;
Liu, Jianqi
  |  
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2018/12/13
Identification of GZD824 as an Orally Bioavailable Inhibitor That Targets Phosphorylated and Nonphosphorylated Breakpoint Cluster Region-Abelson (Bcr-Abl) Kinase and Overcomes Clinically Acquired Mutation-Induced Resistance against Imatinib
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2013, 卷号: 56, 期号: 3
Ren, Xiaomei
;
Pan, Xiaofen
;
Zhang, Zhang
;
Wang, Deping
;
Lu, Xiaoyun
;
Li, Yupeng
;
Wen, Donghai
;
Long, Huoyou
;
Luo, Jinfeng
;
Feng, Yubing
;
Zhuang, Xiaoxi
;
Zhang, Fengxiang
;
Liu, Jianqi
;
Leng, Fang
;
Lang, Xingfen
;
Bai, Yang
;
She, Miaoqin
;
Tu, Zhengchao
;
Pan, Jingxuan
;
Ding, Ke
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2016/12/16