中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [11]
采集方式
OAI收割 [11]
内容类型
期刊论文 [11]
发表日期
2022 [1]
2021 [2]
2019 [2]
2018 [1]
2017 [1]
2008 [1]
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专题:上海药物研究所
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Design, Synthesis, and Structure-Activity Relationship Studies of Bisamide Derivatives of Amphotericin B with Potent Efficacy and Low Toxicity
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 页码: 17
作者:
Ma, Huijun
;
Qian, Anran
;
Zheng, Yazhou
;
Meng, Xin
;
Wang, Ting
  |  
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2023/04/10
Activation pathway of a G protein-coupled receptor uncovers conformational intermediates as targets for allosteric drug design
期刊论文
OAI收割
NATURE COMMUNICATIONS, 2021, 卷号: 12, 期号: 1, 页码: 15
作者:
Lu, Shaoyong
;
He, Xinheng
;
Yang, Zhao
;
Chai, Zongtao
;
Zhou, Shuhua
  |  
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2021/11/04
Design, Synthesis, and Biological Evaluation of Novel Pyrimido[4,5-b]indole Derivatives Against Gram-Negative Multidrug-Resistant Pathogens
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 12, 页码: 8644-8665
作者:
Kong, Qidi
;
Pan, Wei
;
Xu, Heng
;
Xue, Yaru
;
Guo, Bin
  |  
收藏
  |  
浏览/下载:32/0
  |  
提交时间:2021/08/17
YTHDF1 links hypoxia adaptation and non-small cell lung cancer progression
期刊论文
OAI收割
NATURE COMMUNICATIONS, 2019, 卷号: 10, 页码: 14
作者:
Shi, Yulin
;
Fan, Songqing
;
Wu, Mengge
;
Zuo, Zhixiang
;
Li, Xingyang
  |  
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2020/07/01
Design, Synthesis, and Biological Evaluation of Novel DNA Gyrase-Inhibiting Spiropyrimidinetriones as Potent Antibiotics for Treatment of Infections Caused by Multidrug-Resistant Gram-Positive Bacteria
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 6, 页码: 2950-2973
作者:
Shi, Chenghui
;
Zhang, Yinyong
;
Wang, Ting
;
Lu, Wenchao
;
Zhang, Shuhua
  |  
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2020/07/01
Design, synthesis and biological evaluation of C(4) substituted monobactams as antibacterial agents against multidrug-resistant Gram-negative bacteria
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 151, 页码: 98-109
作者:
Kou, Qunhuan
;
Wang, Ting
;
Zou, Feng
;
Zhang, Shuhua
;
Chen, Qian
  |  
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2019/01/08
Monobactam
C(4) substituents
Pyridone
MDR Gram-negative bacteria
Antibacterial activity
Discovery of Novel Pyridone-Conjugated Monosulfactams as Potent and Broad-Spectrum Antibiotics for Multidrug-Resistant Gram-Negative Infections
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 60, 期号: 7, 页码: 2669-2684
作者:
Tan, Liang
;
Tao, Yunliang
;
Wang, Ting
;
Zou, Feng
;
Zhang, Shuhua
  |  
收藏
  |  
浏览/下载:49/0
  |  
提交时间:2019/01/08
Synthesis and biological evaluation of new N-linked 5-triazolylmethyl oxazolidinones
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2008, 卷号: 43, 期号: 8, 页码: 1706-1714
作者:
Fan, Houxing
;
Chen, Yilang
;
Jiang, Zhiteng
;
Zhang, Shuhua
;
Zhong, Dafang
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2019/01/08
oxazolidinone
linezolid
antibacterial agents
gram-positive organisms
Synthesis and antibacterial activity of novel fluoroquinolones containing substituted piperidines
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2007, 卷号: 17, 期号: 16, 页码: 4523-4526
作者:
Dang, Zhao
;
Yang, Yushe
;
Ji, Ruyun
;
Zhang, Shuhua
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2019/01/08
fluoroquinolone
antibacterial activity
piperidine
Synthesis and antibacterial activity of oxazolidinones containing triazolyl group
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2007, 卷号: 42, 期号: 8, 页码: 1137-1143
作者:
Fan, Houxing
;
Xu, Gang
;
Chen, Yflang
;
Jiang, Zhiteng
;
Zhang, Shuhua
  |  
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2019/01/08
oxazolidinone
linezolid
antibacterial agents
gram-positive organisms