中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
广州生物医药与健康... [18]
昆明植物研究所 [14]
新疆理化技术研究所 [2]
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OAI收割 [34]
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期刊论文 [34]
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2016 [10]
2015 [4]
2014 [5]
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Pharmacol... [34]
Chemistry [10]
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浏览/检索结果:
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学科主题:Pharmacology & Pharmacy
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The discovery of novel and selective fatty acid binding protein 4 inhibitors by virtual screening and biological evaluation
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2016, 卷号: 24, 期号: 18, 页码: 4310-4317
作者:
Song, Ming
;
Xu, Yong
;
Zhang, Yan
;
Nie, Tao
;
Zhou, Yang
  |  
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2018/12/13
Structure-Based Design of Tetrahydroisoquinoline-7-carboxamides as Selective Discoidin Domain Receptor 1 (DDR1) Inhibitors
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 12, 页码: 5911-5916
Wang, Zhen
;
Bian, Huan
;
Bartual, Sergio G.
;
Du, Wenting
;
Luo, Jinfeng
;
Zhao, Hu
;
Zhang, Shasha
;
Mo, Cheng
;
Zhou, Yang
;
Xu, Yong
;
Tu, Zhengchao
;
Ren, Xiaomei
;
Lu, Xiaoyun
;
Brekken, Rolf A.
;
Yao, Libo
;
Bullock, Alex N.
;
Su, Jin
;
Ding, Ke
收藏
  |  
浏览/下载:50/0
  |  
提交时间:2016/12/16
Structure-Based Design of Tetrahydroisoquinoline-7-carboxamides as Selective Discoidin Domain Receptor 1 (DDR1) Inhibitors
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 12, 页码: 5911-5916
作者:
Yao, Libo
;
Ding, Ke
;
Su, Jin
;
Bullock, Alex N.
;
Brekken, Rolf A.
  |  
收藏
  |  
浏览/下载:32/0
  |  
提交时间:2018/12/13
Discovery of Benzo[cd]indol-2(1H)-ones as Potent and Specific BET Bromodomain Inhibitors: Structure-Based Virtual Screening, Optimization, and Biological Evaluation
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 4, 页码: 1565-1579
作者:
Tu, Zhengchao
;
Zhou, Yulai
;
Ding, Ke
;
Xu, Yong
;
Xue, Xiaoqian
  |  
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2018/12/13
Skp1: Implications in cancer and SCF-oriented anti-cancer drug discovery
期刊论文
OAI收割
PHARMACOLOGICAL RESEARCH, 2016, 卷号: 111, 页码: 34-42
作者:
Lu, Yongzhi
;
Hussain, Muzammal
;
Liu, Yong-Qiang
;
Su, Kai
;
Zhang, Jiancun
  |  
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2018/12/13
Identification of N-phenyl-2-(N-phenylphenylsulfonamido) acetamides as new ROR gamma inverse agonists: Virtual screening, structure-based optimization, and biological evaluation
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 116, 页码: 13-26
作者:
Xue, Xiaoqian
;
Song, Yu
;
Qian, Chao-Nan
;
Yan, Weiqun
;
Xing, Yanli
  |  
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2018/12/13
Discovery of Benzo[cd]indol-2(1H)-ones as Potent and Specific BET Bromodomain Inhibitors: Structure-Based Virtual Screening, Optimization, and Biological Evaluation
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 4, 页码: 1565-1579
Xue, Xiaoqian
;
Zhang, Yan
;
Liu, Zhaoxuan
;
Song, Ming
;
Xing, Yanli
;
Xiang, Qiuping
;
Wang, Zhen
;
Tu, Zhengchao
;
Zhou, Yulai
;
Ding, Ke
;
Xu, Yong
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2016/12/16
The discovery of novel and selective fatty acid binding protein 4 inhibitors by virtual screening and biological evaluation
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2016, 卷号: 24, 期号: 18, 页码: 4310-4317
Zhou, Yang
;
Nie, Tao
;
Zhang, Yan
;
Song, Ming
;
Li, Kuai
;
Ding, Mengxiao
;
Ding, Ke
;
Wu, Donghai
;
Xu, Yong
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2016/12/16
Skp1: Implications in cancer and SCF-oriented anti-cancer drug discovery
期刊论文
OAI收割
PHARMACOLOGICAL RESEARCH, 2016, 卷号: 111, 页码: 34-42
Hussain, Muzammal
;
Lu, Yongzhi
;
Liu, Yong-Qiang
;
Su, Kai
;
Zhang, Jiancun
;
Liu, Jinsong
;
Zhou, Guang-Biao
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2016/12/16
Identification of N-phenyl-2-(N-phenylphenylsulfonamido) acetamides as new ROR gamma inverse agonists: Virtual screening, structure-based optimization, and biological evaluation
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 116, 页码: 13-26
Song, Yu
;
Xue, Xiaoqian
;
Wu, Xishan
;
Wang, Rui
;
Xing, Yanli
;
Yan, Weiqun
;
Zhou, Yulai
;
Qian, Chao-Nan
;
Zhang, Yan
;
Xu, Yong
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2016/12/16