中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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The discovery of novel and selective fatty acid binding protein 4 inhibitors by virtual screening and biological evaluation 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2016, 卷号: 24, 期号: 18, 页码: 4310-4317
作者:  
Song, Ming;  Xu, Yong;  Zhang, Yan;  Nie, Tao;  Zhou, Yang
  |  收藏  |  浏览/下载:21/0  |  提交时间:2018/12/13
Structure-Based Design of Tetrahydroisoquinoline-7-carboxamides as Selective Discoidin Domain Receptor 1 (DDR1) Inhibitors 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 12, 页码: 5911-5916
Wang, Zhen; Bian, Huan; Bartual, Sergio G.; Du, Wenting; Luo, Jinfeng; Zhao, Hu; Zhang, Shasha; Mo, Cheng; Zhou, Yang; Xu, Yong; Tu, Zhengchao; Ren, Xiaomei; Lu, Xiaoyun; Brekken, Rolf A.; Yao, Libo; Bullock, Alex N.; Su, Jin; Ding, Ke
收藏  |  浏览/下载:50/0  |  提交时间:2016/12/16
Structure-Based Design of Tetrahydroisoquinoline-7-carboxamides as Selective Discoidin Domain Receptor 1 (DDR1) Inhibitors 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 12, 页码: 5911-5916
作者:  
Yao, Libo;  Ding, Ke;  Su, Jin;  Bullock, Alex N.;  Brekken, Rolf A.
  |  收藏  |  浏览/下载:32/0  |  提交时间:2018/12/13
Discovery of Benzo[cd]indol-2(1H)-ones as Potent and Specific BET Bromodomain Inhibitors: Structure-Based Virtual Screening, Optimization, and Biological Evaluation 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 4, 页码: 1565-1579
作者:  
Tu, Zhengchao;  Zhou, Yulai;  Ding, Ke;  Xu, Yong;  Xue, Xiaoqian
  |  收藏  |  浏览/下载:24/0  |  提交时间:2018/12/13
Skp1: Implications in cancer and SCF-oriented anti-cancer drug discovery 期刊论文  OAI收割
PHARMACOLOGICAL RESEARCH, 2016, 卷号: 111, 页码: 34-42
作者:  
Lu, Yongzhi;  Hussain, Muzammal;  Liu, Yong-Qiang;  Su, Kai;  Zhang, Jiancun
  |  收藏  |  浏览/下载:24/0  |  提交时间:2018/12/13
Identification of N-phenyl-2-(N-phenylphenylsulfonamido) acetamides as new ROR gamma inverse agonists: Virtual screening, structure-based optimization, and biological evaluation 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 116, 页码: 13-26
作者:  
Xue, Xiaoqian;  Song, Yu;  Qian, Chao-Nan;  Yan, Weiqun;  Xing, Yanli
  |  收藏  |  浏览/下载:23/0  |  提交时间:2018/12/13
Discovery of Benzo[cd]indol-2(1H)-ones as Potent and Specific BET Bromodomain Inhibitors: Structure-Based Virtual Screening, Optimization, and Biological Evaluation 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 4, 页码: 1565-1579
Xue, Xiaoqian; Zhang, Yan; Liu, Zhaoxuan; Song, Ming; Xing, Yanli; Xiang, Qiuping; Wang, Zhen; Tu, Zhengchao; Zhou, Yulai; Ding, Ke; Xu, Yong
收藏  |  浏览/下载:20/0  |  提交时间:2016/12/16
The discovery of novel and selective fatty acid binding protein 4 inhibitors by virtual screening and biological evaluation 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2016, 卷号: 24, 期号: 18, 页码: 4310-4317
Zhou, Yang; Nie, Tao; Zhang, Yan; Song, Ming; Li, Kuai; Ding, Mengxiao; Ding, Ke; Wu, Donghai; Xu, Yong
收藏  |  浏览/下载:20/0  |  提交时间:2016/12/16
Skp1: Implications in cancer and SCF-oriented anti-cancer drug discovery 期刊论文  OAI收割
PHARMACOLOGICAL RESEARCH, 2016, 卷号: 111, 页码: 34-42
Hussain, Muzammal; Lu, Yongzhi; Liu, Yong-Qiang; Su, Kai; Zhang, Jiancun; Liu, Jinsong; Zhou, Guang-Biao
收藏  |  浏览/下载:24/0  |  提交时间:2016/12/16
Identification of N-phenyl-2-(N-phenylphenylsulfonamido) acetamides as new ROR gamma inverse agonists: Virtual screening, structure-based optimization, and biological evaluation 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 116, 页码: 13-26
Song, Yu; Xue, Xiaoqian; Wu, Xishan; Wang, Rui; Xing, Yanli; Yan, Weiqun; Zhou, Yulai; Qian, Chao-Nan; Zhang, Yan; Xu, Yong
收藏  |  浏览/下载:29/0  |  提交时间:2016/12/16