中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
广州生物医药与健康... [20]
昆明植物研究所 [1]
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OAI收割 [21]
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期刊论文 [21]
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2016 [10]
2015 [4]
2014 [2]
2013 [2]
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2009 [2]
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学科主题
Pharmacol... [21]
Chemistry [10]
Biochemist... [6]
Integrativ... [1]
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学科主题:Pharmacology & Pharmacy
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The discovery of novel and selective fatty acid binding protein 4 inhibitors by virtual screening and biological evaluation
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2016, 卷号: 24, 期号: 18, 页码: 4310-4317
作者:
Song, Ming
;
Xu, Yong
;
Zhang, Yan
;
Nie, Tao
;
Zhou, Yang
  |  
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2018/12/13
Structure-Based Design of Tetrahydroisoquinoline-7-carboxamides as Selective Discoidin Domain Receptor 1 (DDR1) Inhibitors
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 12, 页码: 5911-5916
Wang, Zhen
;
Bian, Huan
;
Bartual, Sergio G.
;
Du, Wenting
;
Luo, Jinfeng
;
Zhao, Hu
;
Zhang, Shasha
;
Mo, Cheng
;
Zhou, Yang
;
Xu, Yong
;
Tu, Zhengchao
;
Ren, Xiaomei
;
Lu, Xiaoyun
;
Brekken, Rolf A.
;
Yao, Libo
;
Bullock, Alex N.
;
Su, Jin
;
Ding, Ke
收藏
  |  
浏览/下载:50/0
  |  
提交时间:2016/12/16
Design and synthesis of N-(4-aminopyridin-2-yl)amides as B-Raf(V600E) inhibitors
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2016, 卷号: 26, 期号: 12, 页码: 2760-2763
Li, Xiaokai
;
Shen, Jiayi
;
Tan, Li
;
Zhang, Zhang
;
Gao, Donglin
;
Luo, Jinfeng
;
Cheng, Huimin
;
Zhou, Xiaoping
;
Ma, Jie
;
Ding, Ke
;
Lu, Xiaoyun
收藏
  |  
浏览/下载:42/0
  |  
提交时间:2016/12/16
3-aminopyrazolopyrazine derivatives as spleen tyrosine kinase inhibitors
期刊论文
OAI收割
CHEMICAL BIOLOGY & DRUG DESIGN, 2016, 卷号: 88, 期号: 5, 页码: 690-698
作者:
Tu, Zhengchao
;
Zhou, Xiaoping
;
Ding, Ke
;
Long, Huoyou
;
Luo, Jingfeng
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2018/12/13
Structure-Based Design of Tetrahydroisoquinoline-7-carboxamides as Selective Discoidin Domain Receptor 1 (DDR1) Inhibitors
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 12, 页码: 5911-5916
作者:
Yao, Libo
;
Ding, Ke
;
Su, Jin
;
Bullock, Alex N.
  |  
收藏
  |  
浏览/下载:32/0
  |  
提交时间:2018/12/13
Discovery of Benzo[cd]indol-2(1H)-ones as Potent and Specific BET Bromodomain Inhibitors: Structure-Based Virtual Screening, Optimization, and Biological Evaluation
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 4, 页码: 1565-1579
作者:
Tu, Zhengchao
;
Zhou, Yulai
;
Ding, Ke
;
Xu, Yong
;
Xue, Xiaoqian
  |  
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2018/12/13
Design and synthesis of N-(4-aminopyridin-2-yl)amides as B-Raf(V600E) inhibitors
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2016, 卷号: 26, 期号: 12, 页码: 2760-2763
作者:
Lu, Xiaoyun
;
Luo, Jinfeng
;
Cheng, Huimin
;
Zhou, Xiaoping
;
Ma, Jie
  |  
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2018/12/13
Discovery of Benzo[cd]indol-2(1H)-ones as Potent and Specific BET Bromodomain Inhibitors: Structure-Based Virtual Screening, Optimization, and Biological Evaluation
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 4, 页码: 1565-1579
Xue, Xiaoqian
;
Zhang, Yan
;
Liu, Zhaoxuan
;
Song, Ming
;
Xing, Yanli
;
Xiang, Qiuping
;
Wang, Zhen
;
Tu, Zhengchao
;
Zhou, Yulai
;
Ding, Ke
;
Xu, Yong
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2016/12/16
3-aminopyrazolopyrazine derivatives as spleen tyrosine kinase inhibitors
期刊论文
OAI收割
CHEMICAL BIOLOGY & DRUG DESIGN, 2016, 卷号: 88, 期号: 5, 页码: 690-698
Shen, Jiayi
;
Li, Xiaokai
;
Zhang, Zhang
;
Luo, Jingfeng
;
Long, Huoyou
;
Tu, Zhengchao
;
Zhou, Xiaoping
;
Ding, Ke
;
Lu, Xiaoyun
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2016/12/16
The discovery of novel and selective fatty acid binding protein 4 inhibitors by virtual screening and biological evaluation
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2016, 卷号: 24, 期号: 18, 页码: 4310-4317
Zhou, Yang
;
Nie, Tao
;
Zhang, Yan
;
Song, Ming
;
Li, Kuai
;
Ding, Mengxiao
;
Ding, Ke
;
Wu, Donghai
;
Xu, Yong
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2016/12/16