中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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新疆理化技术研究... [260]
上海药物研究所 [24]
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期刊论文 [312]
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Discovery of a CB2 and 5-HT1A receptor dual agonist for the treatment of depression and anxiety
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 265, 页码: 20
作者:
Yang, Wenjiao
;
Gong, Xudong
;
Sun, Haiguo
;
Wu, Chunhui
;
Suo, Jin
  |  
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2024/03/06
CB2R agonist
5-HT1AR agonist
CB1R antagonist
Antidepressant
Anxiolytic
Repurposing of Rutan showed effective treatment for COVID-19 disease
期刊论文
OAI收割
FRONTIERS IN MEDICINE, 2023, 卷号: 10, 页码: 13
作者:
Salikhov, Shavkat I.
;
Abdurakhmonov, Ibrokhim Y.
;
Oshchepkova, Yuliya I.
;
Ziyavitdinov, Jamolitdin F.
;
Berdiev, Nodir Sh.
  |  
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2024/01/26
COVID-19
SARS-CoV-2
3CLpro
RdRp
Rhus coriaria
Rutan
clinical trial
Toad venom bufadienolides and bufotoxins: An updated review
期刊论文
OAI收割
DRUG DEVELOPMENT RESEARCH, 2023, 页码: 24
作者:
Asrorov, Akmal M.
;
Kayumov, Muzaffar
;
Mukhamedov, Nurkhodja
;
Yashinov, Ansor
;
Mirakhmetova, Ziyoda
  |  
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2023/10/17
arenobufagin
bufadienolides
bufalin
bufotalin
cinobufagin
cinobufotalin
gamabufotalin
Three new feruloyl glucuronopyranosyl glycerols from Eriocaulon buergerianum with their anti-fibrotic effects on hepatic stellate cells
期刊论文
OAI收割
NATURAL PRODUCT RESEARCH, 2023, 卷号: 37, 期号: 6, 页码: 956-966
作者:
Zhang, Yong
;
Li, Hao
;
Xu, Zhijian
;
Shi, Yulong
;
Li, Bo
  |  
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2024/03/27
Eriocaulon buergerianum
Eriocaulaceae
feruloyl glucuronopyranosyl glycerols
TGF-beta 1 receptor
hepatic fibrosis
Root-Extracted lignanamides from Limonium gmelinii (Willd.) Kuntze with a potential PTP1B inhibitory activity by regulating PI3K/AKT signaling pathway
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2023, 卷号: 132, 页码: 9
作者:
Tuohongerbieke, Amanguli
;
Liu, Liu
;
Li, Jun
;
Xin, Xuelei
;
Aisa, Haji Akber
  |  
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2023/10/17
Limonium gmelinii (Willd
) Kuntze
Plumbaginaceae
Lignanamides
Protein tyrosine phosphatase 1B inhibitors
PI3K
AKT Signaling Pathway
Traditional Use, Phytochemical Profiles and Pharmacological Properties of Artemisia Genus from Central Asia
期刊论文
OAI收割
MOLECULES, 2022, 卷号: 27, 期号: 16, 页码: 38
作者:
Nurlybekova, Aliya
;
Kudaibergen, Aidana
;
Kazymbetova, Aizhan
;
Amangeldi, Magzhan
;
Baiseitova, Aizhamal
  |  
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2022/09/30
Artemisia genus
TKM
Kazakhstan
sequiterpene lactone
essential oils
flavonoids
alpha-glucosidase
PTP1B
BNA
antioxidant
Safety, tolerability, and pharmacokinetics of VV116, an oral nucleoside analog against SARS-CoV-2, in Chinese healthy subjects
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2022, 页码: 9
作者:
Qian, Hong-jie
;
Wang, Yu
;
Zhang, Meng-qi
;
Xie, Yuan-chao
;
Wu, Qing-qing
  |  
收藏
  |  
浏览/下载:37/0
  |  
提交时间:2022/06/15
VV116
nucleoside analog
SARS-CoV-2
safety
pharmacokinetics
healthy subjects
Design, synthesis, in vitro evaluation of a new pyrrolo[1,2-a]thiazolo[5,4-d]pyrimidinone derivatives as cholinesterase inhibitors against Alzheimer's disease
期刊论文
OAI收割
JOURNAL OF HETEROCYCLIC CHEMISTRY, 2022, 页码: 16
作者:
Zeng, Yan
;
Nie, Lifei
;
Liu, Liu
;
Niu, Chao
;
Li, Yi
  |  
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2022/06/15
Phenolic Compounds and Bioactivities from Pomegranate (Punica granatum L.) Peels
期刊论文
OAI收割
JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY, 2022, 卷号: 70, 期号: 12, 页码: 3678-3686
作者:
Ruan, JH (Ruan, Jing-Hui) [1] , [2]
;
Li, J (Li, Jun) [1]
;
Adili, G (Adili, Guliqire) [2]
;
Sun, GY (Sun, Guang-Ying) [1]
;
Abuduaini, M (Abuduaini, Munire) [1] , [2]
  |  
收藏
  |  
浏览/下载:66/0
  |  
提交时间:2022/05/06
Punica granatum L.
pomegranate peel
sphenolic compounds
antioxidant
antimicrobial
antitumor
Synthesis and Biological Activities of Dihydrooxazolo[5,4-d]- pyrrolo[1,2-a]pyrimidinones
期刊论文
OAI收割
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2022, 卷号: 42, 期号: 2, 页码: 543-556
作者:
Zeng, Y (Zeng Yan) [1] , [2]
;
Nie, LF (Nie Lifei) [1]
;
Niu, C (Niu Chao) [1]
;
Mamatjan, A (Mamatjan Aytilla) [1] , [2]
;
Bozorov, K (Bozorov Khurshed) [1]
  |  
收藏
  |  
浏览/下载:59/0
  |  
提交时间:2022/05/17
oxazopyrimidinone
synthesis
bioisosterism
anticancer activity
antimicrobial activity
structure-activity relationships (SARs)