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上海药物研究所 [283]
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期刊论文 [292]
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Application of ensemble learning for predicting GABA
A
receptor agonists
期刊论文
OAI收割
COMPUTERS IN BIOLOGY AND MEDICINE, 2024, 卷号: 169, 页码: 13
作者:
Xiao, Fu
;
Ding, Xiaoyu
;
Shi, Yan
;
Wang, Dingyan
;
Wang, Yitian
  |  
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2024/03/25
GABA(A )receptor
Benzodiazepine
Agonist
Machine learning
Classification
Naringenin improves muscle endurance via activation of the Sp1-ERRg transcriptional axis
期刊论文
OAI收割
CELL REPORTS, 2023, 卷号: 42, 期号: 11, 页码: 25
作者:
Lv, Zhenyu
;
Meng, Jiao
;
Yao, Sheng
;
Xiao, Fu
;
Li, Shilong
  |  
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2023/12/11
Design, synthesis and biological evaluation of chalcone derivatives as potent and orally active hCYP3A4 inhibitors
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2023, 卷号: 95, 页码: 9
作者:
Lu, Shiwei
;
Zhang, Feng
;
Gong, Jiahao
;
Huang, Jian
;
Zhu, Guanghao
  |  
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2023/12/08
Cytochrome P450 3A4 (CYP3A4)
Inhibitors
Isoquinoline chalcones
Orally active
Loops Mediate Agonist-Induced Activation of the Stimulator of Interferon Genes Protein
期刊论文
OAI收割
JOURNAL OF CHEMICAL INFORMATION AND MODELING, 2023, 页码: 9
作者:
Li, Rui
;
Chen, Lin
;
He, Xinheng
;
Cao, Duanhua
;
Zhang, Zehong
  |  
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2023/12/11
αExtractor: a system for automatic extraction of chemical information from biomedical literature
期刊论文
OAI收割
SCIENCE CHINA-LIFE SCIENCES, 2023, 页码: 4
作者:
Xiong, Jiacheng
;
Liu, Xiaohong
;
Li, Zhaojun
;
Xiao, Hongzhong
;
Wang, Guangchao
  |  
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2023/12/08
LogD7.4 prediction enhanced by transferring knowledge from chromatographic retention time, microscopic pKa and logP
期刊论文
OAI收割
JOURNAL OF CHEMINFORMATICS, 2023, 卷号: 15, 期号: 1, 页码: 13
作者:
Wang, Yitian
;
Xiong, Jiacheng
;
Xiao, Fu
;
Zhang, Wei
;
Cheng, Kaiyang
  |  
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2023/10/17
logD7.4
Lipid solubility
Graph neural network
Molecular property prediction
OTTM: an automated classification tool for translational drug discovery from omics data
期刊论文
OAI收割
BRIEFINGS IN BIOINFORMATICS, 2023, 页码: 12
作者:
Yang, Xiaobo
;
Zhang, Bei
;
Wang, Siqi
;
Lu, Ye
;
Chen, Kaixian
  |  
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2023/10/17
OTTM
omics data
translational drug discovery
literature mining
hepatocellular carcinoma
Learning protein fitness landscapes with deep mutational scanning data from multiple sources
期刊论文
OAI收割
CELL SYSTEMS, 2023, 卷号: 14, 期号: 8, 页码: 22
作者:
Chen, Lin
;
Zhang, Zehong
;
Li, Zhenghao
  |  
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2023/10/17
Design, synthesis and biological evaluation of salicylanilides as novel allosteric inhibitors of human pancreatic lipase
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2023, 卷号: 91, 页码: 11
作者:
Zhao, Yitian
;
Zhang, Min
;
Hou, Xudong
;
Han, Jiaxin
;
Qin, Xiaoya
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2023/10/17
Salicylanilide
hPL inhibitor
Structure -activity relationship
Anti -obesity
Spermine is a natural suppressor of AR signaling in castration-resistant prostate cancer
期刊论文
OAI收割
CELL REPORTS, 2023, 卷号: 42, 期号: 7, 页码: 24
作者:
Li, Xiao
;
Li, Fei
;
Ye, Fei
;
Guo, Haotian
;
Chen, Wentao
  |  
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2023/10/17