中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
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上海药物研究所 [237]
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期刊论文 [1114]
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Deep convolutional neural network based on self-distillation for tool wear recognition
期刊论文
OAI收割
ENGINEERING APPLICATIONS OF ARTIFICIAL INTELLIGENCE, 2024, 卷号: 132, 页码: 12
作者:
Pan, Yi
;
Hao, Ling
;
He, Jianliang
;
Ding, Kun
;
Yu, Qiang
  |  
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2024/03/27
Tool fault diagnosis
Mobile inspection robots
Self-distillation
Industry 4.0
Deep learning
Design of functional coating with superior liquid repellency, self-cleaning, photodegradation and thermal insulation properties for building protection
期刊论文
OAI收割
PROGRESS IN ORGANIC COATINGS, 2024, 卷号: 188, 页码: 14
作者:
Ding, Xiaoya
;
Xu, Xuelei
;
Wang, Yi
;
Bao, Jiuwen
;
Zhang, Peng
  |  
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2024/04/07
Building protection
Energy saving
Super-hydrophobic
Liquid repellency
Inulin-like polysaccharide ABWW may impede CCl
4
induced hepatic stellate cell activation through mediating the FAK/PI3K/AKT signaling pathway
in vitro
&
in vivo
期刊论文
OAI收割
CARBOHYDRATE POLYMERS, 2024, 卷号: 326, 页码: 15
作者:
Dai, Xiaolan
;
Du, Zhenyun
;
Jin, Can
;
Tang, Bixi
;
Chen, Xia
  |  
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2024/02/19
Fructan
Hepatic fibrosis
Hepatic stellate cells
FAK/PI3K/AKT
A novel strategy for treating oncogene-mutated tumors by targeting tumor microenvironment and synergistically enhancing anti-PD-1 immunotherapy
期刊论文
OAI收割
CANCER COMMUNICATIONS, 2024, 页码: 5
作者:
Liu, Yingqiang
;
Tong, Linjiang
;
Zhang, Mengge
;
Zhang, Qi
;
Liu, Qiupei
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2024/03/13
Entanglement Generation of Polar Molecules via Deep Reinforcement Learning
期刊论文
OAI收割
JOURNAL OF CHEMICAL THEORY AND COMPUTATION, 2024
作者:
Zhang, Zuo-Yuan
;
Sun, Zhaoxi
;
Duan, Tao
;
Ding, Yi-Kai
;
Huang, Xinning
  |  
收藏
  |  
浏览/下载:46/0
  |  
提交时间:2024/03/26
Policy Gradient Adaptive Dynamic Programming for Model-Free Multi-Objective Optimal Control
期刊论文
OAI收割
IEEE/CAA Journal of Automatica Sinica, 2024, 卷号: 11, 期号: 4, 页码: 1060-1062
作者:
Hao Zhang
;
Yan Li
;
Zhuping Wang
;
Yi Ding
;
Huaicheng Yan
  |  
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2024/03/18
From bench to bedside: current development and emerging trend of KRAS-targeted therapy
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2023, 页码: 18
作者:
Chen, Yi
;
Liu, Qiu-pei
;
Xie, Hua
;
Ding, Jian
  |  
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2024/01/16
KRAS mutation
KRAS(G12C) inhibitor
Pan-KRAS inhibitor
SHP2 allosteric inhibitor
SOS1 inhibitor
combination therapy
Preclinical and early clinical studies of a novel compound SYHA1813 that efficiently crosses the blood-brain barrier and exhibits potent activity against glioblastoma
期刊论文
OAI收割
ACTA PHARMACEUTICA SINICA B, 2023, 卷号: 13, 期号: 12, 页码: 4748-4764
作者:
Liu, Yingqiang
;
Zhan, Zhengsheng
;
Kang, Zhuang
;
Li, Mengyuan
;
Lv, Yongcong
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2024/01/26
Small molecule inhibitor
Tumor microenvironment
Immune-checkpoint
immune-deficient mouse models
including temozolomide (TMZ) insensitive tumors. Notably
HDAC3 and HDAC8 PROTAC dual degrader reveals roles of histone acetylation in gene regulation
期刊论文
OAI收割
CELL CHEMICAL BIOLOGY, 2023, 卷号: 30, 期号: 11, 页码: 1421-+
作者:
Xiao, Yufeng
;
Hale, Seth
;
Awasthee, Nikee
;
Meng, Chengcheng
;
Zhang, Xuan
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2024/01/16
Identification of [1,2,4]Triazolo[4,3-a]pyrazine PARP1 inhibitors with overcome acquired resistance activities
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 259, 页码: 19
作者:
Wang, Pingyuan
;
Zhu, Wen-Ting
;
Wang, Yajing
;
Song, Shan-Shan
;
Xi, Yong
  |  
收藏
  |  
浏览/下载:58/0
  |  
提交时间:2023/10/17
PARP1 inhibitor
Synthetic lethality
Drug resistance
Anticancer
Structure -activity relationship