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AT 2023lli: A Tidal Disruption Event with Prominent Optical Early Bump and Delayed Episodic X-Ray Emission
期刊论文
OAI收割
ASTROPHYSICAL JOURNAL LETTERS, 2024, 卷号: 964, 期号: 2
作者:
Huang, Shifeng
;
Jiang, Ning
;
Zhu, Jiazheng
;
Wang, Yibo
;
Wang, Tinggui
  |  
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2024/04/08
Discovery of a 1,6-naphthyridin-4-one-based AXL inhibitor with improved pharmacokinetics and enhanced in vivo antitumor efficacy
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 265, 页码: 17
作者:
Lan, Yaohan
;
Peng, Xia
;
Ji, Yinchun
;
Su, Yi
;
Duan, Wenhu
  |  
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2024/02/27
AXL inhibitor
In vivo antitumor efficacy
6-Naphthyridin-4-one derivatives
Scaffold hopping
Structure-based drug design
Discovery of a CB2 and 5-HT1A receptor dual agonist for the treatment of depression and anxiety
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 265, 页码: 20
作者:
Yang, Wenjiao
;
Gong, Xudong
;
Sun, Haiguo
;
Wu, Chunhui
;
Suo, Jin
  |  
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2024/03/06
CB2R agonist
5-HT1AR agonist
CB1R antagonist
Antidepressant
Anxiolytic
Diachronous slab-driven Early Cretaceous crustal extension and pulsed magmatic response in southeastern China: Insight from A-type granite and related rocks
期刊论文
OAI收割
GONDWANA RESEARCH, 2024, 卷号: 126, 页码: 22-39
作者:
Chen, Jing-Yuan
;
Yang, Jin-Hui
  |  
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2023/12/27
Southeastern China
Subduction
A-type granites
Diachronous extension
Early Cretaceous
Discovery, Optimization, and Evaluation of Novel Pyridin-2(1
H
)-one Analogues as Potent TRK Inhibitors for Cancer Treatment
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 2, 页码: 1168-1183
作者:
Xu, Zichao
;
Peng, Xia
;
Zhang, Renjie
;
Ji, Yinchun
;
You, Mengke
  |  
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2024/02/27
Proteogenomic characterization of small cell lung cancer identifies biological insights and subtype-specific therapeutic strategies
期刊论文
OAI收割
CELL, 2024, 卷号: 187, 期号: 1, 页码: 49
作者:
Liu, Qian
;
Zhang, Jing
;
Guo, Chenchen
;
Wang, Mengcheng
;
Wang, Chenfei
  |  
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2024/02/27
NICER, NuSTAR, and Insight-HXMT Views to the Newly Discovered Black Hole X-Ray Binary Swift J1727.8-1613
期刊论文
OAI收割
ASTROPHYSICAL JOURNAL LETTERS, 2024, 卷号: 960, 期号: 2
作者:
Peng, Jing-Qiang
;
Zhang, Shu
;
Shui, Qing-Cang
;
Zhang, Shuang-Nan
;
Kong, Ling-Da
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收藏
  |  
浏览/下载:1/0
  |  
提交时间:2024/03/29
Active degradation-nitrification microbial assemblages in the hypoxic zone in a subtropical estuary
期刊论文
OAI收割
SCIENCE OF THE TOTAL ENVIRONMENT, 2023, 卷号: 904, 页码: 14
作者:
Lu, Yanhong
;
Cheung, Shunyan
;
Koh, Xiu Pei
;
Xia, Xiaomin
;
Jing, Hongmei
  |  
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2024/03/11
Estuary
Hypoxia
AOA
Bacteria
Cooccurrence
Microbial interactions
Structure-based drug discovery of novel fused- pyrazolone carboxamide derivatives as potent and selective AXL inhibitors
期刊论文
OAI收割
ACTA PHARMACEUTICA SINICA B, 2023, 卷号: 13, 期号: 12, 页码: 4918-4933
作者:
Fang, Feifei
;
Dai, Yang
;
Wang, Hao
;
Ji, Yinchun
;
Liang, Xuewu
  |  
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2024/01/26
derivatives
Antitumor drug development
Potential AXL inhibitor
Antitumor activity
Structure-based drug design
Fused-pyrazolone carboxamide
An ultra-compact promoter drives widespread neuronal expression in mouse and monkey brains
期刊论文
OAI收割
CELL REPORTS, 2023, 卷号: 42, 期号: 11, 页码: 21
作者:
Wang, Jingyi
;
Lin, Jianbang
;
Chen, Yefei
;
Liu, Jing
;
Zheng, Qiongping
  |  
收藏
  |  
浏览/下载:31/0
  |  
提交时间:2024/01/16