中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [20]
地理科学与资源研究所 [4]
西安光学精密机械研究... [3]
自动化研究所 [2]
生态环境研究中心 [2]
西北高原生物研究所 [1]
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OAI收割 [35]
内容类型
期刊论文 [35]
发表日期
2023 [9]
2022 [7]
2021 [7]
2020 [4]
2019 [2]
2018 [3]
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Engineerin... [1]
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Discovery of 5-trifluoromethyl-2-aminopyrimidine derivatives as potent dual inhibitors of FLT3 and CHK1
期刊论文
OAI收割
RSC MEDICINAL CHEMISTRY, 2023, 页码: 14
作者:
Deng, Minjie
;
Gao, Yue
;
Wang, Peipei
;
Du, Wenjing
;
Xu, Gaoya
  |  
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2024/02/19
Design, synthesis and biological evaluation of 2-aminopyrimidine derivatives as potent FLT3 inhibitors
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2023, 卷号: 96, 页码: 5
作者:
Lian, Xuanmin
;
Gao, Yue
;
Li, Xuemei
;
Wang, Peipei
;
Tong, Lexian
  |  
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2023/12/11
2-aminopyrimidine
FLT3 inhibitors
MV4-11
FLT3 mutations
Discovery of 2-Aminopyrimidine Derivatives as Potent Dual FLT3/CHK1 Inhibitors with Significantly Reduced hERG Inhibitory Activities
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 页码: 23
作者:
Li, Xuemei
;
Wang, Peipei
;
Wang, Chang
;
Jin, Tingting
;
Xu, Ran
  |  
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2023/10/17
Discovery of pyrido[4,3-d]pyrimidinone derivatives as novel Wee1 inhibitors
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2023, 卷号: 87, 页码: 12
作者:
Ye, Qingqing
;
Ma, Jingkun
;
Wang, Peipei
;
Wang, Chang
;
Sun, Mei
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2023/10/17
Wee1 inhibitor
Scaffold hopping
Riverine organic pollution source and yield from the whole Changjiang river network: Effects of urbanization under changing hydrology
期刊论文
OAI收割
JOURNAL OF HYDROLOGY, 2023, 卷号: 620, 页码: 129544
作者:
Wang, Fang
;
Zhang, Peipei
;
Yan, Weijin
;
Jia, Mingrui
;
Su, Xiaokang
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2023/07/14
Preventive and therapeutic benefits of nelfinavir in rhesus macaques and human beings infected with SARS-CoV-2
期刊论文
OAI收割
Signal Transduction and Targeted Therapy, 2023, 卷号: 8, 期号: 5, 页码: 2384-2391
作者:
Xu, Zhijian
;
Shi, Danrong
;
Han, Jianbao
;
Ling, Yun
;
Jiang, Xiangrui
  |  
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2024/03/27
Design, Synthesis, and Biological Evaluation of 2-Aminothiazole Derivatives as Novel Checkpoint Kinase 1 (CHK1) Inhibitors
期刊论文
OAI收割
CHEMMEDCHEM, 2023, 页码: 19
作者:
Deng, Minjie
;
Wang, Peipei
;
Long, Xiubing
;
Xu, Gaoya
;
Wang, Chang
  |  
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2023/04/10
2-aminothiazole
CHK1 inhibitors
antiproliferation
hematologic malignancies
biological activity
Design, synthesis, and evaluation of pyrido.[3,4-b]pyrazin-2(1H)-one derivatives as potent FLT3 inhibitors
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2023, 卷号: 79, 页码: 117155
作者:
Sun, Mei
;
Wang, Chang
;
Wang, Peipei
;
Ye, Qingqing
;
Zhou, Yubo
  |  
收藏
  |  
浏览/下载:0/0
  |  
提交时间:2024/04/09
FLT3
FLT3-D835Y
Acute myeloid leukemia
Structure -activity relationships
High-throughput screening of SARS-CoV-2 main and papain-like protease inhibitors
期刊论文
OAI收割
PROTEIN & CELL, 2023, 卷号: 14, 期号: 1, 页码: 17-27
作者:
Zang, Yi
;
Su, Mingbo
;
Wang, Qingxing
;
Cheng, Xi
;
Zhang, Wenru
  |  
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2024/03/27
high-throughput screening
SARS
CoV-2
main
papain-like
proteases
Dual inhibition of CHK1/FLT3 enhances cytotoxicity and overcomes adaptive and acquired resistance in FLT3-ITD acute myeloid leukemia
期刊论文
OAI收割
LEUKEMIA, 2022, 页码: 11
作者:
Jiang, Kailong
;
Li, Xuemei
;
Wang, Chang
;
Hu, Xiaobei
;
Wang, Peipei
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2023/04/10