中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共27条,第1-10条 帮助

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Nanobodies and chemical cross-links advance the structural and functional analysis of PI3K alpha 期刊论文  OAI收割
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2022, 卷号: 119, 期号: 38, 页码: 9
作者:  
Hart, Jonathan R.;  Liu, Xiao;  Pan, Chen;  Liang, Anyi;  Ueno, Lynn
  |  收藏  |  浏览/下载:9/0  |  提交时间:2023/10/17
Structural basis of tethered agonism of the adhesion GPCRs ADGRD1 and ADGRF1 期刊论文  OAI收割
NATURE, 2022, 页码: 24
作者:  
Qu, Xiangli;  Qiu, Na;  Wang, Mu;  Zhang, Bingjie;  Du, Juan
  |  收藏  |  浏览/下载:28/0  |  提交时间:2022/06/15
Discovery of Novel Allosteric Modulators Targeting an Extra-Helical Binding Site of GLP-1R Using Structure- and Ligand-Based Virtual Screening 期刊论文  OAI收割
BIOMOLECULES, 2021, 卷号: 11, 期号: 7, 页码: 14
作者:  
Zhou, Qingtong;  Guo, Wanjing;  Dai, Antao;  Cai, Xiaoqing;  Vass, Marton
  |  收藏  |  浏览/下载:31/0  |  提交时间:2021/08/17
Affinity Mass Spectrometry-Based Fragment Screening Identified a New Negative Allosteric Modulator of the Adenosine A(2A) Receptor Targeting the Sodium Ion Pocket 期刊论文  OAI收割
ACS CHEMICAL BIOLOGY, 2021, 卷号: 16, 期号: 6, 页码: 991-1002
作者:  
Lu, Yan;  Liu, Hongyue;  Yang, Dehua;  Zhong, Li;  Xin, Ye
  |  收藏  |  浏览/下载:51/0  |  提交时间:2021/08/17
G protein-coupled receptors: structure- and function-based drug discovery 期刊论文  OAI收割
SIGNAL TRANSDUCTION AND TARGETED THERAPY, 2021, 卷号: 6, 期号: 1, 页码: 27
作者:  
Yang, Dehua;  Zhou, Qingtong;  Labroska, Viktorija;  Qin, Shanshan;  Darbalaei, Sanaz
  |  收藏  |  浏览/下载:28/0  |  提交时间:2021/05/24
Targeted Proteomics Combined with Affinity Mass Spectrometry Analysis Reveals Antagonist E7 Acts As an Intracellular Covalent Ligand of Orphan Receptor GPR52 期刊论文  OAI收割
ACS CHEMICAL BIOLOGY, 2020, 卷号: 15, 期号: 12, 页码: 3275-3284
作者:  
Ma, Mengna;  Guo, Shimeng;  Lin, Xi;  Li, Shanshan;  Wu, Yiran
  |  收藏  |  浏览/下载:27/0  |  提交时间:2021/05/24
A Novel G Protein-Biased and Subtype-Selective Agonist for a G Protein-Coupled Receptor Discovered from Screening Herbal Extracts 期刊论文  OAI收割
ACS CENTRAL SCIENCE, 2020, 卷号: 6, 期号: 2, 页码: 213-225
作者:  
Zhang, Bingjie;  Zhao, Simeng;  Yang, Dehua;  Wu, Yiran;  Xin, Ye
  |  收藏  |  浏览/下载:33/0  |  提交时间:2020/07/01
Accelerating the Throughput of Affinity Mass Spectrometry-Based Ligand Screening toward a G Protein-Coupled Receptor 期刊论文  OAI收割
ANALYTICAL CHEMISTRY, 2019, 卷号: 91, 期号: 13, 页码: 8162-8169
作者:  
Lu, Yan;  Qin, Shanshan;  Zhang, Bingjie;  Dai, Antao;  Cai, Xiaoqing
  |  收藏  |  浏览/下载:23/0  |  提交时间:2020/07/01
Efficient ligand discovery from natural herbs by integrating virtual screening, affinity mass spectrometry and targeted metabolomics 期刊论文  OAI收割
ANALYST, 2019, 卷号: 144, 期号: 9, 页码: 2881-2890
作者:  
Wang, Zhihua;  Liang, Hao;  Cao, Haijie;  Zhang, Bingjie;  Li, Jun
  |  收藏  |  浏览/下载:28/0  |  提交时间:2020/07/01
Crystal structure of the Frizzled 4 receptor in a ligand-free state 期刊论文  OAI收割
NATURE, 2018, 卷号: 560, 期号: 7720, 页码: 666-+
作者:  
Yang, Shifan;  Wu, Yiran;  Xu, Ting-Hai;  de Waal, Parker W.;  He, Yuanzheng
  |  收藏  |  浏览/下载:80/0  |  提交时间:2019/01/08