中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共45条,第1-10条 帮助

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Discovery of a New-Generation S-Adenosylmethionine-Noncompetitive Covalent Inhibitor Targeting the Lysine Methyltransferase Enhancer of Zeste Homologue 2 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 66, 期号: 11, 页码: 7629-7644
作者:  
Zhang, Yi;  Yang, Hong;  Li, Bingbing;  Li, Jiayi;  Li, Huaxuan
  |  收藏  |  浏览/下载:20/0  |  提交时间:2023/10/17
Downscaling mapping method for local climate zones from the perspective of deep learning 期刊论文  OAI收割
URBAN CLIMATE, 2023, 卷号: 49, 页码: 101500
作者:  
Yu, Wenbo;  Yang, Jun;  Wu, Feng;  He, Baojie;  Yu, Huisheng
  |  收藏  |  浏览/下载:13/0  |  提交时间:2023/05/06
Regional thermal environment changes: Integration of satellite data and land use/land cover 期刊论文  OAI收割
ISCIENCE, 2023, 卷号: 26, 期号: 2, 页码: 105820
作者:  
Ren, Jiayi;  Yang, Jun;  Wu, Feng;  Sun, Wei;  Xiao, Xiangming
  |  收藏  |  浏览/下载:8/0  |  提交时间:2023/07/14
Improved Surface Soil Organic Carbon Mapping of SoilGrids250m Using Sentinel-2 Spectral Images in the Qinghai-Tibetan Plateau 期刊论文  OAI收割
REMOTE SENSING, 2023, 卷号: 15, 期号: 1, 页码: 17
作者:  
Yang, Jiayi;  Fan, Junjian;  Lan, Zefan;  Mu, Xingmin;  Wu, Yiping
  |  收藏  |  浏览/下载:22/0  |  提交时间:2023/02/13
Structure-activity relationship study of a series of nucleoside derivatives bearing sulfonamide scaffold as potent and selective PRMT5 inhibitors 期刊论文  OAI收割
BIOORGANIC CHEMISTRY, 2023, 卷号: 130, 页码: 20
作者:  
Chen, Yuting;  Shi, Qiongyu;  Yang, Hong;  Li, Jiayi;  Zhou, Kaixin
  |  收藏  |  浏览/下载:20/0  |  提交时间:2023/04/10
Attribution of Urban Diurnal Thermal Environmental Change: Importance of Global-Local Effects 期刊论文  OAI收割
IEEE JOURNAL OF SELECTED TOPICS IN APPLIED EARTH OBSERVATIONS AND REMOTE SENSING, 2023, 卷号: 16, 页码: 8087-8101
作者:  
Yu, Wenbo;  Yang, Jun;  Cong, Nan;  Ren, Jiayi;  Yu, Huisheng
  |  收藏  |  浏览/下载:5/0  |  提交时间:2023/11/29
Glycosyltransferase-related long non-coding RNA signature predicts the prognosis of colon adenocarcinoma 期刊论文  OAI收割
FRONTIERS IN ONCOLOGY, 2022, 卷号: 12
作者:  
Zhang, Jiawei;  Wu, Yinan;  Mu, Jiayi;  Xin, Dijia;  Wang, Luyao
  |  收藏  |  浏览/下载:20/0  |  提交时间:2022/12/22
Discovery of a potent and selective proteolysis targeting chimera (PROTAC) degrader of NSD3 histone methyltransferase 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 239, 页码: 18
作者:  
Sun, Yaoliang;  Zhang, Ying;  Chen, Xiaoai;  Yu, Aisong;  Du, Wenhao
  |  收藏  |  浏览/下载:41/0  |  提交时间:2022/08/30
Discovery of novel benzimidazole derivatives as potent p300 bromodomain inhibitors with anti-proliferative activity in multiple cancer cells 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2022, 卷号: 66, 页码: 16
作者:  
Chen, Zonglong;  Li, Jiayi;  Yang, Hong;  He, Yulong;  Shi, Qiongyu
  |  收藏  |  浏览/下载:35/0  |  提交时间:2022/08/16
Design, synthesis and biological evaluation of (R)-5-methylpyrrolidin-2-ones as p300 bromodomain inhibitors with Anti-Tumor activities in multiple tumor lines 期刊论文  OAI收割
BIOORGANIC CHEMISTRY, 2022, 卷号: 124, 页码: 15
作者:  
Liu, Ruiqi;  Yang, Hong;  Chen, Zonglong;  Zhou, Kaixin;  Shi, Qiongyu
  |  收藏  |  浏览/下载:37/0  |  提交时间:2022/08/16