中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共36条,第1-10条 帮助

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Structure-Based Ligand Discovery Targeting the Transmembrane Domain of Frizzled Receptor FZD7 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 页码: 14
作者:  
Li, Cuixia;  Wu, Yiran;  Wang, Wenli;  Xu, Lu;  Zhou, Yan
  |  收藏  |  浏览/下载:14/0  |  提交时间:2023/10/17
Orthogonally Engineered Albumin with Attenuated Macrophage Phagocytosis for the Targeted Visualization and Phototherapy of Liver Cancer 期刊论文  OAI收割
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2023, 卷号: 145, 期号: 31, 页码: 17377-17388
作者:  
Dou, Wei-Tao;  Qiu, Peng;  Shi, Yuanyuan;  Zhu, Ling;  Guo, Chen
  |  收藏  |  浏览/下载:124/0  |  提交时间:2023/10/17
Cryo-EM structures of orphan GPR21 signaling complexes 期刊论文  OAI收割
NATURE COMMUNICATIONS, 2023, 卷号: 14, 期号: 1, 页码: 1
作者:  
Xi Lin;  Bo Chen;  Yiran Wu;  Yingqi Han;  Ao Qi
  |  收藏  |  浏览/下载:15/0  |  提交时间:2023/05/22
Structures of the human cholecystokinin receptors bound to agonists and antagonists 期刊论文  OAI收割
NATURE CHEMICAL BIOLOGY, 2021, 卷号: 17, 期号: 12, 页码: 1230-1237
作者:  
Zhang, Xuefeng;  He, Chenglin;  Wang, Mu;  Zhou, Qingtong;  Yang, Dehua
  |  收藏  |  浏览/下载:9/0  |  提交时间:2024/03/21
Structure-Based Design of Dual-Acting Compounds Targeting Adenosine A(2A) Receptor and Histone Deacetylase as Novel Tumor Immunotherapeutic Agents 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 22, 页码: 16573-16597
作者:  
Yan, Wenzhong;  Ling, Lijun;  Wu, Yiran;  Yang, Kexin;  Liu, Ruiquan
  |  收藏  |  浏览/下载:16/0  |  提交时间:2022/06/15
Discovery of Novel Allosteric Modulators Targeting an Extra-Helical Binding Site of GLP-1R Using Structure- and Ligand-Based Virtual Screening 期刊论文  OAI收割
BIOMOLECULES, 2021, 卷号: 11, 期号: 7, 页码: 14
作者:  
Zhou, Qingtong;  Guo, Wanjing;  Dai, Antao;  Cai, Xiaoqing;  Vass, Marton
  |  收藏  |  浏览/下载:31/0  |  提交时间:2021/08/17
Affinity Mass Spectrometry-Based Fragment Screening Identified a New Negative Allosteric Modulator of the Adenosine A(2A) Receptor Targeting the Sodium Ion Pocket 期刊论文  OAI收割
ACS CHEMICAL BIOLOGY, 2021, 卷号: 16, 期号: 6, 页码: 991-1002
作者:  
Lu, Yan;  Liu, Hongyue;  Yang, Dehua;  Zhong, Li;  Xin, Ye
  |  收藏  |  浏览/下载:52/0  |  提交时间:2021/08/17
G protein-coupled receptors: structure- and function-based drug discovery 期刊论文  OAI收割
SIGNAL TRANSDUCTION AND TARGETED THERAPY, 2021, 卷号: 6, 期号: 1, 页码: 27
作者:  
Yang, Dehua;  Zhou, Qingtong;  Labroska, Viktorija;  Qin, Shanshan;  Darbalaei, Sanaz
  |  收藏  |  浏览/下载:29/0  |  提交时间:2021/05/24
Targeted Proteomics Combined with Affinity Mass Spectrometry Analysis Reveals Antagonist E7 Acts As an Intracellular Covalent Ligand of Orphan Receptor GPR52 期刊论文  OAI收割
ACS CHEMICAL BIOLOGY, 2020, 卷号: 15, 期号: 12, 页码: 3275-3284
作者:  
Ma, Mengna;  Guo, Shimeng;  Lin, Xi;  Li, Shanshan;  Wu, Yiran
  |  收藏  |  浏览/下载:29/0  |  提交时间:2021/05/24
A unique hormonal recognition feature of the human glucagon-like peptide-2 receptor 期刊论文  OAI收割
CELL RESEARCH, 2020, 页码: 11
作者:  
Sun, Wen;  Chen, Li-Nan;  Zhou, Qingtong;  Zhao, Li-Hua;  Yang, Dehua
  |  收藏  |  浏览/下载:113/0  |  提交时间:2020/12/24