中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [33]
上海生物化学与细胞生... [1]
上海营养与健康研究所 [1]
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OAI收割 [35]
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期刊论文 [35]
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2024 [1]
2023 [4]
2022 [8]
2021 [13]
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Cell Biolo... [1]
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Molecular features of the ligand-free GLP-1R, GCGR and GIPR in complex with G
s
proteins
期刊论文
OAI收割
CELL DISCOVERY, 2024, 卷号: 10, 期号: 1, 页码: 13
作者:
Cong, Zhaotong
;
Zhao, Fenghui
;
Li, Yang
;
Luo, Gan
;
Mai, Yiting
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2024/03/13
Structural and mechanistic insights provided by single particle cryo-EM analysis of phosphoinositide 3-kinase (PI3Ka)
期刊论文
OAI收割
BIOCHIMICA ET BIOPHYSICA ACTA-REVIEWS ON CANCER, 2023, 卷号: 1878, 期号: 5, 页码: 6
作者:
Vogt, Peter K.
;
Hart, Jonathan R.
;
Yang, Su
;
Zhou, Qingtong
;
Yang, Dehua
  |  
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2023/10/17
Phosphoinositide 3-kinase
BYL-719
Nanobody
CXMS
Mutants
Structural insights into the interaction of three Y- shaped ligands with PI3Kα
期刊论文
OAI收割
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2023, 卷号: 120, 期号: 34, 页码: 9
作者:
Zhou, Qingtong
;
Liu, Xiao
;
Neri, Dario
;
Li, Wenxin
;
Favalli, Nicholas
  |  
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2023/12/08
phosphoinositide 3-kinase
drug target
ligand
binding pocket
chemical scaffold
Structural insights into ligand recognition and subtype selectivity of the human melanocortin-3 and melanocortin-5 receptors
期刊论文
OAI收割
CELL DISCOVERY, 2023, 卷号: 9, 期号: 1, 页码: 15
作者:
Feng, Wenbo
;
Zhou, Qingtong
;
Chen, Xianyue
;
Dai, Antao
;
Cai, Xiaoqing
  |  
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2023/10/17
Ligand recognition mechanism of the human relaxin family peptide receptor 4 (RXFP4)
期刊论文
OAI收割
NATURE COMMUNICATIONS, 2023, 卷号: 14, 期号: 1, 页码: 492
作者:
Chen, Yan
;
Zhou, Qingtong
;
Wang, Jiang
;
Xu, Youwei
;
Wang, Yun
  |  
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2024/03/27
Cryo-EM structures of cancer-specific helical and kinase domain mutations of PI3K alpha
期刊论文
OAI收割
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2022, 卷号: 119, 期号: 46, 页码: 11
作者:
Liu, Xiao
;
Zhou, Qingtong
;
Hart, Jonathan R.
;
Xu, Yingna
;
Yang, Su
  |  
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2023/10/17
phosphoinositide 3-kinase (PI3K)
mass spectrometry
mutants
Molecular recognition of morphine and fentanyl by the human mu-opioid receptor
期刊论文
OAI收割
CELL, 2022, 卷号: 185, 期号: 23, 页码: 4361-+
作者:
Zhuang, Youwen
;
Wang, Yue
;
He, Bingqing
;
He, Xinheng
;
Zhou, X. Edward
  |  
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2023/04/10
Nanobodies and chemical cross-links advance the structural and functional analysis of PI3K alpha
期刊论文
OAI收割
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2022, 卷号: 119, 期号: 38, 页码: 9
作者:
Hart, Jonathan R.
;
Liu, Xiao
;
Pan, Chen
;
Liang, Anyi
;
Ueno, Lynn
  |  
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2023/10/17
phosphoinositide 3-kinase (PI3K)
nanobody
conformational changes
chemical cross-linking
mass spectrometry
Structural insights into ligand recognition and selectivity of somatostatin receptors
期刊论文
OAI收割
CELL RESEARCH, 2022, 页码: 12
作者:
Zhao, Wenli
;
Han, Shuo
;
Qiu, Na
;
Feng, Wenbo
;
Lu, Mengjie
  |  
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2022/08/16
Structural basis of peptidomimetic agonism revealed by small-molecule GLP-1R agonists Boc5 and WB4-24
期刊论文
OAI收割
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2022, 卷号: 119, 期号: 20, 页码: 10
作者:
Cong, Zhaotong
;
Zhou, Qingtong
;
Li, Yang
;
Chen, Li-Nan
;
Zhang, Zi-Chen
  |  
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2022/09/30
glucagon-like peptide-1 receptor
type 2 diabetes mellitus
cryoelectron microscopy
peptidomimetic agonism