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A simple copper-catalyzed two-step one-pot synthesis of indolo[1,2-a]quinazoline

文献类型：期刊论文

作者Li, Chunpu1,2; Zhang, Lei1; Shu, Shuangjie1; Liu, Hong1,2
刊名BEILSTEIN JOURNAL OF ORGANIC CHEMISTRY
出版日期2014-10-21
卷号10页码:2441-2447
关键词copper one pot synthetic methods
ISSN号1860-5397
DOI10.3762/bjoc.10.254
文献子类Article
英文摘要A convenient CuI/L-proline-catalyzed, two-step one-pot method has been developed for the preparation of indolo[1,2-a]quinazoline derivatives using a sequential Ullmann-type C-C and C-N coupling. This protocol provides an operationally simple and rapid strategy for preparing indolo[1,2-a]quinazoline derivatives and displays good functional group tolerance. All the starting materials are commercial available or can be easily prepared.
WOS关键词COUPLING REACTIONS ; N-ARYLATION ; C-N ; METHYLENE-COMPOUNDS ; ROOM-TEMPERATURE ; ARYL IODIDES ; DERIVATIVES ; NUCLEOPHILES ; DISCOVERY ; HALIDES
资助项目National Natural Science Foundation of China[21021063] ; National Natural Science Foundation of China[91229204] ; National Natural Science Foundation of China[81025017] ; Program of Shanghai Subject Chief Scientist[XD1407100]
WOS研究方向Chemistry
语种英语
WOS记录号WOS:000344500900001
出版者BEILSTEIN-INSTITUT
源URL[http://119.78.100.183/handle/2S10ELR8/276867]  
专题药物化学研究室
通讯作者Liu, Hong
作者单位1.Chinese Acad Sci, Shanghai Inst Mat Med, Key Lab Receptor Res, Shanghai 201203, Peoples R China
2.China Pharmaceut Univ, Dept Med Chem, Nanjing 210009, Jiangsu, Peoples R China;
推荐引用方式
GB/T 7714		 Li, Chunpu,Zhang, Lei,Shu, Shuangjie,et al. A simple copper-catalyzed two-step one-pot synthesis of indolo[1,2-a]quinazoline[J]. BEILSTEIN JOURNAL OF ORGANIC CHEMISTRY,2014,10:2441-2447.
APA Li, Chunpu,Zhang, Lei,Shu, Shuangjie,&Liu, Hong.(2014).A simple copper-catalyzed two-step one-pot synthesis of indolo[1,2-a]quinazoline.BEILSTEIN JOURNAL OF ORGANIC CHEMISTRY,10,2441-2447.
MLA Li, Chunpu,et al."A simple copper-catalyzed two-step one-pot synthesis of indolo[1,2-a]quinazoline".BEILSTEIN JOURNAL OF ORGANIC CHEMISTRY 10(2014):2441-2447.

入库方式： OAI收割

来源：上海药物研究所

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