中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共55条,第1-10条 帮助

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Discovery, Optimization, and Evaluation of Novel Pyridin-2(1H)-one Analogues as Potent TRK Inhibitors for Cancer Treatment 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 2, 页码: 1168-1183
作者:  
Xu, Zichao;  Peng, Xia;  Zhang, Renjie;  Ji, Yinchun;  You, Mengke
  |  收藏  |  浏览/下载:10/0  |  提交时间:2024/02/27
Structure-based drug discovery of novel fused- pyrazolone carboxamide derivatives as potent and selective AXL inhibitors 期刊论文  OAI收割
ACTA PHARMACEUTICA SINICA B, 2023, 卷号: 13, 期号: 12, 页码: 4918-4933
作者:  
Fang, Feifei;  Dai, Yang;  Wang, Hao;  Ji, Yinchun;  Liang, Xuewu
  |  收藏  |  浏览/下载:7/0  |  提交时间:2024/01/26
Constructing N-Acyl/N-Sulfonyl Aza-Sulfur Derivatives from Amides/Sulfonamides and Thiophthalimides via Oxidant Regulation 期刊论文  OAI收割
ORGANIC LETTERS, 2023, 卷号: 25, 期号: 32, 页码: 6018-6023
作者:  
Li, Yazhou;  Wang, Yongkun;  Fang, Feifei;  Zhang, Yu;  Li, Chunpu
  |  收藏  |  浏览/下载:26/0  |  提交时间:2023/10/17
Late-Stage Functionalization for the Divergent Synthesis of Podophyllotoxin Derivatives by Rhodium Catalysis 期刊论文  OAI收割
CHEMISTRY-A EUROPEAN JOURNAL, 2023, 页码: 10
作者:  
Zhao, Yue;  Shen, Yangpeng;  He, Jian;  Li, Jing;  Zhou, Shengbin
  |  收藏  |  浏览/下载:138/0  |  提交时间:2023/10/17
Rapid Access to Polysubstituted Tetrahydrocarbazol-4-ones via Sequential Selective C-H Functionalization from N-Nitrosoanilines 期刊论文  OAI收割
CHINESE JOURNAL OF CHEMISTRY, 2023, 页码: 1957-1962
作者:  
Li, Chan;  Yang, Yanchen;  Fang, Feifei;  Liu, Chaoyi;  Li, Chunpu
  |  收藏  |  浏览/下载:10/0  |  提交时间:2023/10/17
Rh(III)-Catalyzed Synthesis of Substituted Isoindoles through a Direct C-H Activation/[4+1] Annulation and Acyl Migration Cascade of Oxadiazolones with Diazo Compounds 期刊论文  OAI收割
ORGANIC LETTERS, 2023, 页码: 5
作者:  
Yang, Xiaohao;  Ren, Hairu;  Zhou, Shengbin;  Li, Chunpu;  Liu, Chaoyi
  |  收藏  |  浏览/下载:8/0  |  提交时间:2023/10/17
Structural Optimization of Fibroblast Growth Factor Receptor Inhibitors for Treating Solid Tumors 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 66, 期号: 5, 页码: 3226-3249
作者:  
Li, Chunpu;  Dai, Yang;  Kong, Xiangtai;  Wang, Bao;  Peng, Xia
  |  收藏  |  浏览/下载:2/0  |  提交时间:2024/03/27
Synthesis of maleimide-braced peptide macrocycles and their potential anti-SARS-CoV-2 mechanisms 期刊论文  OAI收割
CHEMICAL COMMUNICATIONS, 2022, 页码: 4
作者:  
Li, Jian;  Sun, Jina;  Zhang, Xianglei;  Zhang, Ruxue;  Wang, Qian
  |  收藏  |  浏览/下载:25/0  |  提交时间:2023/04/10
Discovery of Novel Imidazo[4,5-c]quinoline Derivatives to Treat Inflammatory Bowel Disease (IBD) by Inhibiting Multiple Proinflammatory Signaling Pathways and Restoring Intestinal Homeostasis 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 页码: 21
作者:  
Liang, Xuewu;  Xie, Yongle;  Liu, Xuyi;  Xu, Hui;  Ren, Hairu
  |  收藏  |  浏览/下载:25/0  |  提交时间:2022/11/11
Structure-Activity Relationship Study of Indolin-5-yl-cyclopropanamine Derivatives as Selective Lysine Specific Demethylase 1 (LSD1) Inhibitors 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 65, 期号: 5, 页码: 4335-4349
作者:  
Li, Chunpu;  Su, Mingbo;  Zhu, Wei;  Kan, Weijuan;  Ge, Tianpeng
  |  收藏  |  浏览/下载:31/0  |  提交时间:2022/06/15