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Cu-mediated selective O-arylation on C-6 substituted pyridin-2-ones

文献类型：期刊论文

作者Chen, Taijie1; Huang, Qingqing3; Luo, Yu1; Hu, Youhong2; Lu, Wei3
刊名TETRAHEDRON LETTERS
出版日期2013-03-13
卷号54期号:11页码:1401-1404
关键词Chan Evans Lam cross-coupling Arylboronic acids Selectivity O-arylation Pyridin-2-ones
ISSN号0040-4039
DOI10.1016/j.tetlet.2012.12.126
文献子类Article
英文摘要A practical and mild strategy has been developed for the selective O-arylation on C-6 substituted pyridin-2-ones with a series of arylboronic acids, using Cu(OTf)(2) as the catalyst, DABCO as the ligand, Et3N as the base, and K2HPO4 as the additive. This method affords O-arylated pyridin-2-ones with good selectivity and yields (C) 2013 Elsevier Ltd. All rights reserved.
WOS关键词CATALYZED N-ARYLATION ; ARYLBORONIC ACIDS ; COUPLING REACTIONS ; CUPRIC ACETATE ; ARYL ; HETEROCYCLES ; INHIBITORS ; EFFICIENT
资助项目National Natural Science Foundation of China[81172936] ; National Natural Science Foundation of China[21102046] ; Fundamental Research Funds for the Central Universities[00000000] ; Laboratory of Organic Functional Molecules, the Sino-French Institute of ECNU[00000000]
WOS研究方向Chemistry
语种英语
WOS记录号WOS:000315306900016
出版者PERGAMON-ELSEVIER SCIENCE LTD
源URL[http://119.78.100.183/handle/2S10ELR8/277697]  
专题药物化学研究室
通讯作者Luo, Yu
作者单位1.E China Normal Univ, Dept Chem, Shanghai 200062, Peoples R China;
2.Chinese Acad Sci, Shanghai Inst Mat Med, Shanghai 201203, Peoples R China
3.E China Normal Univ, Inst Drug Discovery & Dev, Shanghai 200062, Peoples R China;
推荐引用方式
GB/T 7714		 Chen, Taijie,Huang, Qingqing,Luo, Yu,et al. Cu-mediated selective O-arylation on C-6 substituted pyridin-2-ones[J]. TETRAHEDRON LETTERS,2013,54(11):1401-1404.
APA Chen, Taijie,Huang, Qingqing,Luo, Yu,Hu, Youhong,&Lu, Wei.(2013).Cu-mediated selective O-arylation on C-6 substituted pyridin-2-ones.TETRAHEDRON LETTERS,54(11),1401-1404.
MLA Chen, Taijie,et al."Cu-mediated selective O-arylation on C-6 substituted pyridin-2-ones".TETRAHEDRON LETTERS 54.11(2013):1401-1404.

入库方式： OAI收割

来源：上海药物研究所

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