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Rh(III)-Catalyzed Hydroarylation of Alkyne MIDA Boronates via C-H Activation of Indole Derivatives

文献类型：期刊论文

作者Fei, Xiao1,2,3,4; Li, Chunpu3,4; Yu, Xinhong1,2; Liu, Hong3,4
刊名JOURNAL OF ORGANIC CHEMISTRY
出版日期2019-06-07
卷号84期号:11页码:6840-6850
ISSN号0022-3263
DOI10.1021/acs.joc.9b00638
通讯作者Yu, Xinhong(xhyu@ecust.edu.cn) ; Liu, Hong(hliu@simm.ac.cn)
英文摘要An efficient approach to trans-indolylvinylboronate derivatives has been developed using an Rh-catalyzed hydroarylation of alkyne N-methyliminodiacetic acid boronates via C-H activation. This protocol constitutes a straightforward route for the synthesis of B-containing aza-heterocycles in good yields with excellent functional group tolerance.
WOS关键词DIVERGENT SYNTHESIS ; PROPARGYL ALCOHOLS ; BOND ACTIVATION ; ANNULATION ; ACCESS ; EFFICIENT ; DIFUNCTIONALIZATION ; ISOINDOLINONES ; PLATFORM ; ANALOGS
资助项目National Natural Science Foundation of China[81620108027] ; National Natural Science Foundation of China[21632008] ; National Natural Science Foundation of China[91229204] ; National Natural Science Foundation of China[81220108025] ; National Natural Science Foundation of China[81602975] ; Major Project of Chinese National Programs for Fundamental Research and Development[2015CB910304] ; National S&T Major Projects[2014ZX09507002-001] ; National S&T Major Projects[2015ZX09103003]
WOS研究方向Chemistry
语种英语
WOS记录号WOS:000471212000029
出版者AMER CHEMICAL SOC
源URL[http://119.78.100.183/handle/2S10ELR8/289400]  
专题新药研究国家重点实验室
通讯作者Yu, Xinhong; Liu, Hong
作者单位1.East China Univ Sci & Technol, Sch Pharm, State Key Lab Bioengn Reactors, Shanghai 200237, Peoples R China
2.East China Univ Sci & Technol, Sch Pharm, Shanghai Key Lab New Drug Design, Shanghai 200237, Peoples R China
3.Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, 555 Zu Chong Zhi Rd, Shanghai 201203, Peoples R China
4.Chinese Acad Sci, Shanghai Inst Mat Med, Key Lab Receptor Res, 555 Zu Chong Zhi Rd, Shanghai 201203, Peoples R China
推荐引用方式
GB/T 7714		 Fei, Xiao,Li, Chunpu,Yu, Xinhong,et al. Rh(III)-Catalyzed Hydroarylation of Alkyne MIDA Boronates via C-H Activation of Indole Derivatives[J]. JOURNAL OF ORGANIC CHEMISTRY,2019,84(11):6840-6850.
APA Fei, Xiao,Li, Chunpu,Yu, Xinhong,&Liu, Hong.(2019).Rh(III)-Catalyzed Hydroarylation of Alkyne MIDA Boronates via C-H Activation of Indole Derivatives.JOURNAL OF ORGANIC CHEMISTRY,84(11),6840-6850.
MLA Fei, Xiao,et al."Rh(III)-Catalyzed Hydroarylation of Alkyne MIDA Boronates via C-H Activation of Indole Derivatives".JOURNAL OF ORGANIC CHEMISTRY 84.11(2019):6840-6850.

入库方式： OAI收割

来源：上海药物研究所

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