Constructing N-Acyl/N-Sulfonyl Aza-Sulfur Derivatives from Amides/Sulfonamides and Thiophthalimides via Oxidant Regulation
文献类型：期刊论文
| 作者 | Li, Yazhou1,2; Wang, Yongkun1,2; Fang, Feifei2,3; Zhang, Yu2,3; Li, Chunpu2; Yu, Tao2; Chen, Qiangqiang1,2; Wang, Jiang2,3 ; Liu, Hong1,2
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| 刊名 | ORGANIC LETTERS
 |
| 出版日期 | 2023-08-04 |
| 卷号 | 25期号:32页码:6018-6023 |
| ISSN号 | 1523-7060 |
| DOI | 10.1021/acs.orglett.3c02166 |
| 通讯作者 | Wang, Jiang(jwang@lglab.ac.cn) ; Liu, Hong(hliu@simm.ac.cn) |
| 英文摘要 | Here, we have constructed five distinct types of N-acyl or N-sulfonyl aza-sulfur scaffoldsusing readilyavailable (sulfon)amides and thiophthalimides with precise regulationof oxidants. Our novel methods feature one-pot mild reaction conditionsand simple operation, thereby making them highly convenient for thelate-stage diversification of various amide drugs, bioactive molecules,and peptides. |
| WOS关键词 | IN-VITRO ; SULFONAMIDES ; INHIBITOR |
| 资助项目 | National Natural Science Foundation of China[82130105] ; National Natural Science Foundation of China[82121005] ; National Natural Science Foundation of China[92253305] ; National Natural Science Foundation of China[22177124] ; Lingang Laboratory[LG202103-03-02] ; Lingang Laboratory[LG-GG-202204-02] |
| WOS研究方向 | Chemistry |
| 语种 | 英语 |
| 出版者 | AMER CHEMICAL SOC |
| WOS记录号 | WOS:001043167600001 |
| 源URL | [http://119.78.100.183/handle/2S10ELR8/306857]  |
| 专题 | 新药研究国家重点实验室 |
| 通讯作者 | Wang, Jiang; Liu, Hong |
| 作者单位 | 1.Nanjing Univ Chinese Med, Sch Chinese Mat Med, Nanjing 210023, Jiangsu, Peoples R China 2.Chinese Acad Sci, Inst Mat Med, State Key Lab Drug Res, Shanghai 201203, Peoples R China 3.Lingang Lab, Shanghai 200031, Peoples R China |
| 推荐引用方式 GB/T 7714 | Li, Yazhou,Wang, Yongkun,Fang, Feifei,et al. Constructing N-Acyl/N-Sulfonyl Aza-Sulfur Derivatives from Amides/Sulfonamides and Thiophthalimides via Oxidant Regulation[J]. ORGANIC LETTERS,2023,25(32):6018-6023. |
| APA | Li, Yazhou.,Wang, Yongkun.,Fang, Feifei.,Zhang, Yu.,Li, Chunpu.,...&Liu, Hong.(2023).Constructing N-Acyl/N-Sulfonyl Aza-Sulfur Derivatives from Amides/Sulfonamides and Thiophthalimides via Oxidant Regulation.ORGANIC LETTERS,25(32),6018-6023. |
| MLA | Li, Yazhou,et al."Constructing N-Acyl/N-Sulfonyl Aza-Sulfur Derivatives from Amides/Sulfonamides and Thiophthalimides via Oxidant Regulation".ORGANIC LETTERS 25.32(2023):6018-6023. |
入库方式： OAI收割
来源：上海药物研究所
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