中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共2179条,第1-10条 帮助

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Design and Synthesis of Novel Macrocyclic Derivatives as Potent and Selective Cyclin-Dependent Kinase 7 Inhibitors 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 页码: 20
作者:  
Niu, Pengpeng;  Tao, Yanxin;  Lin, Guohao;  Xu, Huiqi;  Meng, Qingyuan
  |  收藏  |  浏览/下载:0/0  |  提交时间:2024/05/22
Identification of a Novel Selective CDK9 Inhibitor for the Treatment of CRC: Design, Synthesis, and Biological Activity Evaluation 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 6, 页码: 4739-4756
作者:  
Zhong, Ye;  Xu, Jing;  Zhou, Ruochen;  Tang, Li;  Ding, Shaoyue
  |  收藏  |  浏览/下载:7/0  |  提交时间:2024/05/07
Synthesis of 1,4-epoxy-2-aryltetrahydro-1-benzazepines via rhodium(iii)-catalyzed C-H allylation/intramolecular 1,3-dipolar cycloaddition 期刊论文  OAI收割
CHEMICAL COMMUNICATIONS, 2024, 卷号: 60, 期号: 17, 页码: 2401-2404
作者:  
Wang, Xuan;  Li, Jianlong;  Du, Haifang;  Liang, Weihong;  Luo, Cheng
  |  收藏  |  浏览/下载:15/0  |  提交时间:2024/03/13
Gold-catalyzed endo-selective Ring-opening of Epoxides and its Application in Construction of Poly-ethers 期刊论文  OAI收割
CHEMISTRY-A EUROPEAN JOURNAL, 2024, 页码: 10
作者:  
Wu, Kehuan;  Kang, Kaiwen;  Liu, Dan;  Zhang, Chiyue;  Wang, Xinyu
  |  收藏  |  浏览/下载:10/0  |  提交时间:2024/03/25
Discovery of a potent and selective covalent threonine tyrosine kinase (TTK) inhibitor 期刊论文  OAI收割
BIOORGANIC CHEMISTRY, 2024, 卷号: 143, 页码: 16
作者:  
Sun, Yaoliang;  Chen, Zhiwen;  Liu, Guobin;  Chen, Xiaoai;  Shi, Zihan
  |  收藏  |  浏览/下载:12/0  |  提交时间:2024/03/25
Enzymatic Synthesis of Noncanonical α-Amino Acids Containing γ-Tertiary Alcohols 期刊论文  OAI收割
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2024, 页码: 9
作者:  
Zhang, Rui;  Zhang, Chenghua;  Tan, Jiamu;  He, Yifan;  Zhuo, Dan
  |  收藏  |  浏览/下载:24/0  |  提交时间:2024/02/27
Design, Synthesis, and Biological Evaluation of Potent and Selective PROTAC Degraders of Oncogenic KRASG12D 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 2, 页码: 1147-1167
作者:  
Zhou, Chuan;  Fan, Zisheng;  Gu, Yuejiao;  Ge, Zhiming;  Tao, Zhaofan
  |  收藏  |  浏览/下载:10/0  |  提交时间:2024/02/27
Discovery and bioinspired total syntheses of unprecedented sesquiterpenoid dimers unveiled bifurcating [4+2] cycloaddition and target differentiation of enantiomers 期刊论文  OAI收割
CHEMICAL SCIENCE, 2024, 卷号: 15, 期号: 4
作者:  
He, Tao-Bin;  Yan, Bing-Chao;  Zhou, Yuan-Fei;  Sang, Yue-Qian;  Li, Xiao-Nian
  |  收藏  |  浏览/下载:1/0  |  提交时间:2024/05/09
Design, Synthesis, and Structure-Activity Relationship of Novel Potent and Highly Selective Cysteinyl Leukotriene Receptor 1 (CysLT1R) Antagonists 期刊论文  OAI收割
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2024, 卷号: 44, 期号: 1, 页码: 259-276
作者:  
Wang Jingyi;  Liu Jinyu;  Chen Dongsheng;  Chen Huayan;  Xie Xin
  |  收藏  |  浏览/下载:0/0  |  提交时间:2024/05/07
Assessing the greenification potential of cyclodextrin-based molecularly imprinted polymers for pesticides detection 期刊论文  OAI收割
FOOD CHEMISTRY, 2023, 卷号: 429, 页码: 16
作者:  
Farooq, Saqib;  Xu, Lizhou;  Ostovan, Abbas;  Qin, Chunlian;  Liu, Yingjia
  |  收藏  |  浏览/下载:7/0  |  提交时间:2024/01/26