中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
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大连化学物理研究... [468]
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Design and Synthesis of Novel Macrocyclic Derivatives as Potent and Selective Cyclin-Dependent Kinase 7 Inhibitors
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 页码: 20
作者:
Niu, Pengpeng
;
Tao, Yanxin
;
Lin, Guohao
;
Xu, Huiqi
;
Meng, Qingyuan
  |  
收藏
  |  
浏览/下载:0/0
  |  
提交时间:2024/05/22
Identification of a Novel Selective CDK9 Inhibitor for the Treatment of CRC: Design, Synthesis, and Biological Activity Evaluation
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 6, 页码: 4739-4756
作者:
Zhong, Ye
;
Xu, Jing
;
Zhou, Ruochen
;
Tang, Li
;
Ding, Shaoyue
  |  
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2024/05/07
Synthesis of 1,4-epoxy-2-aryltetrahydro-1-benzazepines
via
rhodium(
iii
)-catalyzed C-H allylation/intramolecular 1,3-dipolar cycloaddition
期刊论文
OAI收割
CHEMICAL COMMUNICATIONS, 2024, 卷号: 60, 期号: 17, 页码: 2401-2404
作者:
Wang, Xuan
;
Li, Jianlong
;
Du, Haifang
;
Liang, Weihong
;
Luo, Cheng
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2024/03/13
Gold-catalyzed
endo
-selective Ring-opening of Epoxides and its Application in Construction of Poly-ethers
期刊论文
OAI收割
CHEMISTRY-A EUROPEAN JOURNAL, 2024, 页码: 10
作者:
Wu, Kehuan
;
Kang, Kaiwen
;
Liu, Dan
;
Zhang, Chiyue
;
Wang, Xinyu
  |  
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2024/03/25
6-endo ring-opening of epoxide
Baldwin's rules
gold-catalyzed reactions
marine ladder-like poly-ethers
Nakanishi hypothesis
Discovery of a potent and selective covalent threonine tyrosine kinase (TTK) inhibitor
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2024, 卷号: 143, 页码: 16
作者:
Sun, Yaoliang
;
Chen, Zhiwen
;
Liu, Guobin
;
Chen, Xiaoai
;
Shi, Zihan
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2024/03/25
Inhibitor
Cancer
Threonine tyrosine kinase (TTK)
Covalent
Enzymatic Synthesis of Noncanonical α-Amino Acids Containing γ-Tertiary Alcohols
期刊论文
OAI收割
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2024, 页码: 9
作者:
Zhang, Rui
;
Zhang, Chenghua
;
Tan, Jiamu
;
He, Yifan
;
Zhuo, Dan
  |  
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2024/02/27
Asymmetric Synthesis
Biocatalysis
Noncanonical Amino Acids
Quantum Chemical Calculations
Tertiary Alcohols
Design, Synthesis, and Biological Evaluation of Potent and Selective PROTAC Degraders of Oncogenic KRAS
G12D
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 2, 页码: 1147-1167
作者:
Zhou, Chuan
;
Fan, Zisheng
;
Gu, Yuejiao
;
Ge, Zhiming
;
Tao, Zhaofan
  |  
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2024/02/27
Discovery and bioinspired total syntheses of unprecedented sesquiterpenoid dimers unveiled bifurcating [4+2] cycloaddition and target differentiation of enantiomers
期刊论文
OAI收割
CHEMICAL SCIENCE, 2024, 卷号: 15, 期号: 4
作者:
He, Tao-Bin
;
Yan, Bing-Chao
;
Zhou, Yuan-Fei
;
Sang, Yue-Qian
;
Li, Xiao-Nian
  |  
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2024/05/09
DIELS-ALDER REACTION
BIOMIMETIC SYNTHESES
EFFICIENT ACCESS
DEHYDROGENATION
CYCLOHEXANONES
BIOSYNTHESIS
CONVERSION
OXIDATION
DYNAMICS
PHENOLS
Design, Synthesis, and Structure-Activity Relationship of Novel Potent and Highly Selective Cysteinyl Leukotriene Receptor 1 (CysLT1R) Antagonists
期刊论文
OAI收割
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2024, 卷号: 44, 期号: 1, 页码: 259-276
作者:
Wang Jingyi
;
Liu Jinyu
;
Chen Dongsheng
;
Chen Huayan
;
Xie Xin
  |  
收藏
  |  
浏览/下载:0/0
  |  
提交时间:2024/05/07
cysteinyl leukotriene
cysteinyl leukotriene receptor 1 (CysLT1R)
selective antagonists
Assessing the greenification potential of cyclodextrin-based molecularly imprinted polymers for pesticides detection
期刊论文
OAI收割
FOOD CHEMISTRY, 2023, 卷号: 429, 页码: 16
作者:
Farooq, Saqib
;
Xu, Lizhou
;
Ostovan, Abbas
;
Qin, Chunlian
;
Liu, Yingjia
  |  
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2024/01/26
Cyclodextrins
Molecularly Imprinted Polymers
Pesticide detection
Green chemistry
Environmental safety