中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共48条,第1-10条 帮助

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The p300 Inhibitor A-485 Exerts Antitumor Activity in Growth Hormone Pituitary Adenoma 期刊论文  OAI收割
JOURNAL OF CLINICAL ENDOCRINOLOGY & METABOLISM, 2022, 页码: 10
作者:  
Ji, Chenxing;  Xu, Wen;  Ding, Hong;  Chen, Zhengyuan;  Shi, Chengzhang
  |  收藏  |  浏览/下载:52/0  |  提交时间:2022/06/15
Discovery of a subtype-selective, covalent inhibitor against palmitoylation pocket of TEAD3 期刊论文  OAI收割
ACTA PHARMACEUTICA SINICA B, 2021, 卷号: 11, 期号: 10, 页码: 3206-3219
作者:  
Lu, Tian;  Li, Yong;  Lu, Wenchao;  Spitters, Twgm;  Fang, Xueyu
  |  收藏  |  浏览/下载:52/0  |  提交时间:2021/12/01
Discovery of thalidomide-based PROTAC small molecules as the highly efficient SHP2 degraders 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 218, 页码: 14
作者:  
Yang, Xiangbo;  Wang, Zhijia;  Pei, Yuan;  Song, Ning;  Xu, Lei
  |  收藏  |  浏览/下载:37/0  |  提交时间:2021/08/17
Rhodium-Catalyzed Twofold Unsymmetrical C-H Alkenylation-Annulation/Thiolation Reaction To Access Thiobenzofurans 期刊论文  OAI收割
ORGANIC LETTERS, 2021, 卷号: 23, 期号: 4, 页码: 1194-1198
作者:  
Lin, Jian;  Hu, Liuyu;  Chen, Chao;  Feng, Huijin;  Yu, Yang
  |  收藏  |  浏览/下载:15/0  |  提交时间:2021/05/24
Discovery of Highly Potent, Selective, and Orally Efficacious p300/CBP Histone Acetyltransferases Inhibitors 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 63, 期号: 3, 页码: 1337-1360
作者:  
Yang, Yaxi;  Zhang, Rukang;  Li, Zhaojun;  Mei, Lianghe;  Wan, Shili
  |  收藏  |  浏览/下载:38/0  |  提交时间:2020/07/01
雷公藤甲素衍生物雷腾舒的体外代谢研究 期刊论文  OAI收割
药学学报, 2019, 卷号: 54, 期号: 8, 页码: 1484
作者:  
徐叶;  杜江波;  冯慧瑾;  左建平;  许红涛
  |  收藏  |  浏览/下载:16/0  |  提交时间:2020/07/01
Rhodium(iii)-catalyzed alkyllation of primary c(sp(3))-h bonds with alpha-diazocarbonyl compounds 期刊论文  iSwitch采集
Chemical communications, 2016, 卷号: 52, 期号: 62, 页码: 9672-9675
作者:  
Hou, Wei;  Yang, Yaxi;  Wu, Yunxiang;  Feng, Huijin;  Li, Yuanchao
收藏  |  浏览/下载:40/0  |  提交时间:2019/05/09
Rhodium(III)-catalyzed alkyllation of primary C(sp(3))-H bonds with alpha-diazocarbonyl compounds 期刊论文  OAI收割
CHEMICAL COMMUNICATIONS, 2016, 卷号: 52, 期号: 62, 页码: 9672-9675
作者:  
Hou, Wei;  Yang, Yaxi;  Wu, Yunxiang;  Feng, Huijin;  Li, Yuanchao
  |  收藏  |  浏览/下载:25/0  |  提交时间:2019/01/08
Synthesis and their inhibitory activities of neuroinflammation of dehydroepiandrosterone derivatives 期刊论文  OAI收割
Chinese Journal of Medicinal Chemistry, 2016, 卷号: 26, 期号: 5, 页码: 353-360
作者:  
Wang Youfu;  Wang Rong;  Wang Junliang;  Feng Huijin;  Yang Yaxi
  |  收藏  |  浏览/下载:19/0  |  提交时间:2019/01/08
去氢表雄酮衍生物的合成及其抑制神经炎症活性研究 期刊论文  OAI收割
中国药物化学杂志, 2016, 卷号: 26, 期号: 5, 页码: 353
作者:  
王友富;  王荣;  王均良;  冯慧瑾;  杨亚玺
  |  收藏  |  浏览/下载:21/0  |  提交时间:2020/07/01