中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共171条,第1-10条 帮助

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Development of novel epoxyketone macrocyclic peptidyl proteasome inhibitors through OPA-mediated one-step cyclization of unprotected peptides 期刊论文  OAI收割
BIOORGANIC CHEMISTRY, 2025, 卷号: 156, 页码: 16
作者:  
Zeng, Gongruixue;  Xu, Gaoya;  Gao, Lixin;  Zheng, Xiaoli;  Chi, Xinglong
  |  收藏  |  浏览/下载:9/0  |  提交时间:2025/04/01
Auto-RapTAC: A Versatile and Sustainable Platform for the Automated Rapid Synthesis and Evaluation of PROTAC 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 页码: 15
作者:  
Chen, Jiexuan;  Wu, Mingfei;  Mo, Jun;  Hong, Ju;  Wang, Wei
  |  收藏  |  浏览/下载:13/0  |  提交时间:2025/04/01
Discovery of N-Benzylpiperidinol derivatives as USP7 inhibitors against Hematology 期刊论文  OAI收割
BIOORGANIC CHEMISTRY, 2024, 卷号: 153, 页码: 13
作者:  
Pan, Youlu;  Chen, Haifeng;  Fu, Jingfeng;  Zhang, Jingyu;  Wang, Peipei
  |  收藏  |  浏览/下载:13/0  |  提交时间:2024/10/21
Exploration of novel 20S proteasome activators featuring anthraquinone structures and their application in hypoxic cardiomyocyte protection 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2024, 卷号: 115, 页码: 10
作者:  
Yu, Qian;  Gao, Lixin;  Xu, Linhao;  Han, Yubing;  Cao, Yu
  |  收藏  |  浏览/下载:11/0  |  提交时间:2024/12/11
Enhanced strength-ductility synergy in a gradient hetero-structured CrCoNi medium-entropy alloy 期刊论文  OAI收割
JOURNAL OF MATERIALS RESEARCH AND TECHNOLOGY-JMR&T, 2024, 卷号: 33, 页码: 7491-7502
作者:  
Feng HQ(冯航旗);  Zhang HZ(张杭州);  He ZH(何政鸿);  Zhou LL(周玲玲);  Zhang ZH(张子晗)
  |  收藏  |  浏览/下载:76/0  |  提交时间:2024/12/19
Single-cell sequencing reveals the heterogeneity of pancreatic neuroendocrine tumors under genomic instability and histological grading 期刊论文  OAI收割
ISCIENCE, 2024, 卷号: 27, 期号: 9, 页码: 18
作者:  
Ye, Zeng;  Zhou, Yan;  Hu, Yuheng;  Li, Qiang;  Xu, Zijin
  |  收藏  |  浏览/下载:11/0  |  提交时间:2024/11/05
Stretch-induced hepatic endothelial mechanocrine promotes hepatocyte proliferation 期刊论文  OAI收割
HEPATOLOGY, 2024
作者:  
Wu Y(武亿);  Li LD(李林达);  Li, Wang;  Li N(李宁);  Zhang XY(张晓宇)
  |  收藏  |  浏览/下载:2/0  |  提交时间:2024/12/02
Discovery of a Highly Potent and Selective BRD9 PROTAC Degrader Based on E3 Binder Investigation for the Treatment of Hematological Tumors 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 页码: 28
作者:  
Duan, Haiting;  Zhang, Jingyu;  Gui, Renzhao;  Lu, Yang;  Pang, Ao
  |  收藏  |  浏览/下载:7/0  |  提交时间:2024/08/20
Discovery of potent small molecule ubiquitin-specific protease 10 inhibitors with anti-hepatocellular carcinoma activity through regulating YAP expression 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 272, 页码: 21
作者:  
Lu, Yang;  Gao, Jian;  Wang, Peipei;  Chen, Haifeng;  He, Xinjun
  |  收藏  |  浏览/下载:6/0  |  提交时间:2024/07/12
Ultrahigh surface hardness and excellent hardness gradient induced by ultrafine dual-carbides in a novel stainless bearing steel 期刊论文  OAI收割
JOURNAL OF MATERIALS RESEARCH AND TECHNOLOGY-JMR&T, 2024, 卷号: 30, 页码: 7420-7428
作者:  
Wang W(王为);  Yang MX(杨沐鑫);  Wang, Jing;  Xie JJ(谢季佳);  Wang, Jian
  |  收藏  |  浏览/下载:6/0  |  提交时间:2024/09/18