中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共153条,第1-10条 帮助

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Design, synthesis and structure-activity relationship studies of novel macrocyclic 2,4-diaminopyrimidines as HPK1 inhibitors 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2025, 卷号: 128, 页码: 12
作者:  
Wu, Feifei;  Sun, Jiaqi;  Xu, Mingyang;  Li, Huiyu;  Wei, Jiarui
  |  收藏  |  浏览/下载:1/0  |  提交时间:2025/08/20
Solid-state screening and dry powder inhaler development of ziyuglycoside II sodium salt for enhanced bioavailability 期刊论文  OAI收割
INTERNATIONAL JOURNAL OF PHARMACEUTICS, 2025, 卷号: 681, 页码: 11
作者:  
Zhang, Hanwen;  Wang, Siwen;  Slimani, Sara;  Lv, Yuting;  Nie, Qin
  |  收藏  |  浏览/下载:6/0  |  提交时间:2025/08/20
Tracheal Targeted Nanogrid Delivery Systems of Dexamethasone Visualized by Single-Particle Tracing and Multiscale Pathological Mapping 期刊论文  OAI收割
ACS NANO, 2025, 卷号: 19, 期号: 25, 页码: 23414-23430
作者:  
Cao, Zeying;  Zhou, Shilin;  Zhao, Yanli;  Wu, Qian;  Huang, Chenxi
  |  收藏  |  浏览/下载:2/0  |  提交时间:2025/08/20
Design, Synthesis, and biological evaluation of 7H-Pyrrolo[2,3-d] pyrimidines as potent HPK1 kinase inhibitors 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2025, 卷号: 119, 页码: 13
作者:  
Wu, Feifei;  Li, Huiyu;  Li, Weiqiang;  Zhang, Laishun;  An, Qi
  |  收藏  |  浏览/下载:20/0  |  提交时间:2025/04/01
Targeting QPCTL: An Emerging Therapeutic Opportunity 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 68, 期号: 2, 页码: 929-943
作者:  
Yu, Lei;  Sun, Yaoliang;  Xie, Longyan;  Tan, Xiao;  Wang, Ping
  |  收藏  |  浏览/下载:22/0  |  提交时间:2025/04/01
Discovery of an Efficacious RET PROTAC Degrader with Enhanced Antiproliferative Activity against Resistant Cancer Cells Harboring RET Solvent-Front Mutations 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 68, 期号: 1, 页码: 753-775
作者:  
Zhang, Qian;  He, Yingqi;  Rao, Danni;  He, Rui;  Yu, Lei
  |  收藏  |  浏览/下载:18/0  |  提交时间:2025/02/28
Discovery of Pyrido[2,3-d]pyrimidin-7-one Derivatives as Highly Potent and Efficacious Ectonucleotide Pyrophosphatase/Phosphodiesterase 1 (ENPP1) Inhibitors for Cancer Treatment 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 5, 页码: 3986-4006
作者:  
Sun, Yaoliang;  Chen, Manman;  Han, Yuyan;  Li, Weiqiang;  Ma, Xiaoyu
  |  收藏  |  浏览/下载:37/0  |  提交时间:2024/05/07
Discovery of a potent and selective covalent threonine tyrosine kinase (TTK) inhibitor 期刊论文  OAI收割
BIOORGANIC CHEMISTRY, 2024, 卷号: 143, 页码: 16
作者:  
Sun, Yaoliang;  Chen, Zhiwen;  Liu, Guobin;  Chen, Xiaoai;  Shi, Zihan
  |  收藏  |  浏览/下载:52/0  |  提交时间:2024/03/25
Discovery and Structural Optimization of Covalent ZAP-70 Kinase Inhibitors against Psoriasis 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 页码: 15
作者:  
Rao, Danni;  Yang, Tao;  Feng, Huixu;  An, Qi;  Zhang, Shaofeng
  |  收藏  |  浏览/下载:42/0  |  提交时间:2023/10/17
Microplastics in canned, salt-dried, and instant sea cucumbers sold for human consumption 期刊论文  OAI收割
MARINE POLLUTION BULLETIN, 2023, 卷号: 192, 页码: 8
作者:  
Mohsen, Mohamed;  Lin, Chenggang;  Abdalla, Mohnad;  Liu, Shilin;  Yang, Hongsheng
  |  收藏  |  浏览/下载:42/0  |  提交时间:2023/12/07