中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
紫金山天文台 [25]
上海药物研究所 [16]
武汉植物园 [5]
高能物理研究所 [4]
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期刊论文 [89]
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Residue-Selective Inhibitors Discovery via Covalent DNA-Encoded Chemical Libraries with Diverse Warheads
期刊论文
OAI收割
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2025, 卷号: 147, 期号: 18, 页码: 15469-15481
作者:
Wu, Xinyuan
;
Pan, Jiayi
;
Fan, Rufeng
;
Zhang, Yiwei
  |  
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2025/06/23
Pharmacokinetics and Safety of TPN171 (a PDE5 Inhibitor) in Patients With Mild or Moderate Hepatic Impairment Versus Participants With Normal Hepatic Function: A Phase I Study
期刊论文
OAI收割
CLINICAL PHARMACOLOGY IN DRUG DEVELOPMENT, 2025, 页码: 7
作者:
Zhou, Jing
;
Zhang, Hong
;
Ding, Yanhua
;
Wang, Zhen
;
Wang, Yu
  |  
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2025/06/23
hepatic impairment
pharmacokinetics
phosphodiesterase-5 inhibitor
TPN171
Proteome-Wide Data Guides the Discovery of Lysine-Targeting Covalent Inhibitors Using DNA-Encoded Chemical Libraries
期刊论文
OAI收割
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2025, 页码: 14
作者:
Wu, Xinyuan
;
Li, Shunyao
;
Liang, Ting
;
Yu, Qing
;
Zhang, Yiwei
  |  
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2025/06/23
Activity-based protein profiling data
Covalent DNA-encoded chemical library
Covalent ligand selection
Lysine-targeting covalent inhibitors
Facile synthesis of pyridazinone-focused DNA-encoded libraries
期刊论文
OAI收割
TETRAHEDRON LETTERS, 2024, 卷号: 142, 页码: 4
作者:
Lv, Yuhan
;
Mu, Baiyang
;
Qin, Shaozhao
;
Wu, Xinyuan
;
Lu, Weiwei
  |  
收藏
  |  
浏览/下载:37/0
  |  
提交时间:2024/06/27
A New Blind Selection Approach for Lunar Landing Zones Based on Engineering Constraints Using Sliding Window
期刊论文
OAI收割
Remote Sensing, 2023, 卷号: 15, 期号: 12
作者:
Hengxi Liu
;
Yongzhi Wang
;
Shibo Wen
;
Jianzhong Liu
;
Jiaxiang Wang
  |  
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2024/05/13
DNA-encoded focused indazole library synthesis by a palladium- mediated C-N(sp(2)) cross-coupling reaction between DNA-linked (hetero)aryl halides and aromatic nitrogen heterocycles
期刊论文
OAI收割
TETRAHEDRON LETTERS, 2022, 卷号: 96, 页码: 6
作者:
Yang, Juan
;
Xia, Shengdi
;
Liu, Jiaxiang
;
Yu, Zikun
;
Mei, Lianghe
  |  
收藏
  |  
浏览/下载:45/0
  |  
提交时间:2022/08/16
Human-Climate Coupled Changes in Vegetation Community Complexity of China Since 1980s
期刊论文
OAI收割
EARTHS FUTURE, 2022, 卷号: 10, 期号: 7
作者:
Su, Yanjun
;
Guo, Qinghua
;
Guan, Hongcan
;
Hu, Tianyu
;
Jin, Shichao
  |  
收藏
  |  
浏览/下载:32/0
  |  
提交时间:2024/03/07
vegetation community complexity
human activities
climate change
vegetation map
DNA-encoded C-H functionality via photoredox-mediated hydrogen atom transformation catalysis
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2021, 卷号: 42, 页码: 4
作者:
Shan, Jinming
;
Ling, Xing
;
Liu, JiaXiang
;
Wang, Xuan
;
Lu, Xiaojie
  |  
收藏
  |  
浏览/下载:51/0
  |  
提交时间:2021/08/17
Photoredox
Hydrogen atom transfer
N-Boc saturated heterocycle
DNA Encoded Library (DEL)
Deformation of Antigorite and Its Geological Implications
期刊论文
OAI收割
JOURNAL OF GEOPHYSICAL RESEARCH-SOLID EARTH, 2021, 卷号: 126, 期号: 6, 页码: 24
作者:
Shao, Tongbin
;
Zhou, Yongsheng
;
Song, Maoshuang
;
Ma, Xi
;
Zhang, Lei
  |  
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2022/11/02
Diversified strategy for the synthesis of DNA-encoded oxindole libraries
期刊论文
OAI收割
CHEMICAL SCIENCE, 2021, 卷号: 12, 期号: 8, 页码: 2841-2847
作者:
Wang, Xuan
;
Liu, Jiaxiang
;
Yan, Ziqin
;
Liu, Xiaohong
;
Liu, Sixiu
  |  
收藏
  |  
浏览/下载:38/0
  |  
提交时间:2021/05/24