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Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
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上海药物研究所 [150]
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期刊论文 [292]
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NMRExtractor: leveraging large language models to construct an experimental NMR database from open-source scientific publications
期刊论文
OAI收割
CHEMICAL SCIENCE, 2025, 卷号: 16, 期号: 25, 页码: 11548-11558
作者:
Wang, Qinggong
;
Zhang, Wei
;
Chen, Mingan
  |  
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2025/08/20
Methotrexate exerts antitumor immune activity and improves the clinical efficacy of immunotherapy in patients with solid tumors
期刊论文
OAI收割
SCIENCE TRANSLATIONAL MEDICINE, 2025, 卷号: 17, 期号: 801, 页码: 18
作者:
Yang, Ruirui
;
Wang, Bei
;
Su, Zhaoming
;
Song, Ying
;
Zhang, Yingying
  |  
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2025/08/20
Discovery and Identification of a Novel PORCN Inhibitor via Structure-Based Virtual Screening
期刊论文
OAI收割
ACS CHEMICAL BIOLOGY, 2025, 卷号: 20, 期号: 6, 页码: 1319-1332
作者:
Yang, Xinyu
;
Li, Yanbei
;
Zhou, Jingyi
;
Zhou, Yuanyang
;
Lin, Kexin
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收藏
  |  
浏览/下载:10/0
  |  
提交时间:2025/07/25
Palladium-Catalyzed Enantioselective Arylative Dearomatization of Naphthols and Phenols for Constructing Quinazoline-Containing Spirocycles
期刊论文
OAI收割
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2025, 页码: 9
作者:
Zhang, Chiyue
;
Xu, Gaoya
;
Zhao, Wenlu
;
Li, Xutong
;
Zheng, Mingyue
  |  
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2025/07/25
Antiproliferative activity
Catalytic asymmetric dearomatization
Palladium
Quinazoline-containing spirocycles
Three-dimensionality
Discovery of 3-(Fluoro-imidazolyl)pyridazine Derivatives as Potent STING Agonists with Antitumor Activity
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 68, 期号: 10, 页码: 9864-9885
作者:
Hou, Hui
;
Zhou, Jingyi
;
Sui, Qibang
;
Zhang, Changfa
;
Su, Zhaoming
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2025/07/25
Microbiota-shaped neutrophil senescence regulates sexual dimorphism in bladder cancer
期刊论文
OAI收割
NATURE IMMUNOLOGY, 2025, 卷号: 26, 期号: 5, 页码: 46
作者:
Zhu, Qingchen
;
Zhang, Guiheng
;
Cao, Ming
;
Huang, Huan
;
He, Dan
  |  
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2025/06/23
Bridging chemistry and artificial intelligence by a reaction description language
期刊论文
OAI收割
NATURE MACHINE INTELLIGENCE, 2025, 卷号: 7, 期号: 5, 页码: 16
作者:
Xiong, Jiacheng
;
Zhang, Wei
;
Wang, Yinquan
;
Huang, Jiatao
;
Shi, Yuqi
  |  
收藏
  |  
浏览/下载:9/0
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提交时间:2025/07/25
Residue-Selective Inhibitors Discovery via Covalent DNA-Encoded Chemical Libraries with Diverse Warheads
期刊论文
OAI收割
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2025, 卷号: 147, 期号: 18, 页码: 15469-15481
作者:
Wu, Xinyuan
;
Pan, Jiayi
;
Fan, Rufeng
;
Zhang, Yiwei
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收藏
  |  
浏览/下载:24/0
  |  
提交时间:2025/06/23
Proteome-Wide Data Guides the Discovery of Lysine-Targeting Covalent Inhibitors Using DNA-Encoded Chemical Libraries
期刊论文
OAI收割
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2025, 页码: 14
作者:
Wu, Xinyuan
;
Li, Shunyao
;
Liang, Ting
;
Yu, Qing
;
Zhang, Yiwei
  |  
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2025/06/23
Activity-based protein profiling data
Covalent DNA-encoded chemical library
Covalent ligand selection
Lysine-targeting covalent inhibitors
Recent advances in targeted degradation in the RAS pathway
期刊论文
OAI收割
FUTURE MEDICINAL CHEMISTRY, 2025, 卷号: 17, 期号: 6, 页码: 693-708
作者:
Ge, Zhiming
;
Fan, Zisheng
;
He, Wei
;
Zhou, Guizhen
;
Zhou, Yidi
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2025/04/24
RAS
cancer
mutation
degrader
PROTAC