中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共131条,第1-10条 帮助

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Discovery, Optimization, and Evaluation of Novel Pyridin-2(1H)-one Analogues as Potent TRK Inhibitors for Cancer Treatment 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 2, 页码: 1168-1183
作者:  
Xu, Zichao;  Peng, Xia;  Zhang, Renjie;  Ji, Yinchun;  You, Mengke
  |  收藏  |  浏览/下载:10/0  |  提交时间:2024/02/27
Design, Synthesis, and Biological Evaluation of Potent and Selective PROTAC Degraders of Oncogenic KRASG12D 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 2, 页码: 1147-1167
作者:  
Zhou, Chuan;  Fan, Zisheng;  Gu, Yuejiao;  Ge, Zhiming;  Tao, Zhaofan
  |  收藏  |  浏览/下载:10/0  |  提交时间:2024/02/27
Targeting ST8SIA6-AS1 counteracts KRASG12C inhibitor resistance through abolishing the reciprocal activation of PLK1/c-Myc signaling 期刊论文  OAI收割
EXPERIMENTAL HEMATOLOGY & ONCOLOGY, 2023, 卷号: 12, 期号: 1, 页码: 22
作者:  
Wang, Yafang;  Yao, Mingyue;  Li, Cheng;  Yang, Kexin;  Qin, Xiaolong
  |  收藏  |  浏览/下载:7/0  |  提交时间:2024/01/26
Precise measurement method of carrier motion state in microgravity environment 期刊论文  OAI收割
MEASUREMENT, 2023, 卷号: 222, 页码: 17
作者:  
Liu, Mingyue;  Zhu, Huizhong;  Xu, Xinchao;  Ma, Youqing;  Zhang, Shuo
  |  收藏  |  浏览/下载:6/0  |  提交时间:2023/11/28
Structure-Activity Relationship Study of 1H-Pyrrole-3-carbonitrile Derivatives as STING Receptor Agonists 期刊论文  OAI收割
ACS MEDICINAL CHEMISTRY LETTERS, 2023, 页码: 9
作者:  
Shen, Chang;  Xu, Peijia;  Zhang, Changfa;  Su, Zhaoming;  Shan, Bin
  |  收藏  |  浏览/下载:24/0  |  提交时间:2023/10/17
Erosion Performance of TiAlSiN Coatings Prepared by High-Power Pulsed Magnetron Sputtering 期刊论文  OAI收割
METALS, 2023, 卷号: 13, 期号: 7, 页码: 1306
作者:  
Li, Hua;  Li, Liuhe;  Li, Duoduo;  Tang, Ling;  Luo, Yang
  |  收藏  |  浏览/下载:13/0  |  提交时间:2023/09/05
Goliath induces inflammation in obese mice by linking fatty acid β-oxidation to glycolysis 期刊论文  OAI收割
EMBO REPORTS, 2023, 卷号: 24, 期号: 4
作者:  
Hao, Shumeng;  Zhang, Sulin;  Ye, Jialin;  Chen, Lifan;  Wang, Yan
  |  收藏  |  浏览/下载:1/0  |  提交时间:2024/03/27
Discovery of a Potent, Cooperative, and Selective SOS1 PROTAC ZZ151 with In Vivo Antitumor Efficacy in KRAS-Mutant Cancers 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 66, 期号: 6, 页码: 4197-4214
作者:  
Zhou, Zehui;  Zhou, Guizhen;  Zhou, Chuan;  Fan, Zisheng;  Cui, Rongrong
  |  收藏  |  浏览/下载:2/0  |  提交时间:2024/03/27
Design, Synthesis, and Biological Evaluation of Bipyridazine Derivatives as Stimulator of Interferon Genes (STING) Receptor Agonists 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 66, 期号: 5, 页码: 3327-3347
作者:  
Shan, Bin;  Hou, Hui;  Zhang, Keke;  Li, Rui;  Shen, Chang
  |  收藏  |  浏览/下载:2/0  |  提交时间:2024/03/27
Design of a Coumarin-Based Fluorescent Probe for Efficient In Vivo Imaging of Amyloid-? Plaques 期刊论文  OAI收割
ACS CHEMICAL NEUROSCIENCE, 2023
作者:  
Cao, Yangyang;  Liu, Xiaohui;  Zhang, Jingjing;  Liu, Zhongmin;  Fu, Yan
  |  收藏  |  浏览/下载:2/0  |  提交时间:2024/03/27