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Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
南京地理与湖泊研究... [91]
上海药物研究所 [14]
西北高原生物研究所 [9]
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期刊论文 [121]
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Long-circulating enzyme-activated HSP90-targeted camptothecin derivatives
期刊论文
OAI收割
JOURNAL OF CONTROLLED RELEASE, 2025, 卷号: 383, 页码: 16
作者:
Ding, Mengyuan
;
Shen, Qianqian
;
Su, Yi
;
Lu, Yingxin
;
Jin, Jiyu
  |  
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2025/07/25
eHSP90
Camptothecin derivatives
Cathepsin B
Long-circulating
Unveiling p65 as the target of diphyllin in ameliorating metabolic dysfunction-associated steatotic liver disease via targeted protein degradation technology
期刊论文
OAI收割
FRONTIERS IN PHARMACOLOGY, 2025, 卷号: 16, 页码: 12
作者:
Zhu, Xuejing
;
Zhang, Lei
;
Cui, Wenqian
;
Wang, Liangjie
;
Xu, Fengjing
  |  
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2025/07/25
metabolic dysfunction-associated steatotic liver disease
diphyllin
p65
targeted protein degradation technology
NRF2
Comparative Study on Covalent and Noncovalent Endogenous Albumin-Binding β-Glucuronidase-Activated SN38 Prodrugs for Antitumor Efficacy
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 68, 期号: 8, 页码: 8361-8376
作者:
Lu, Yingxin
;
Jiang, Xing
;
Yang, Biyu
;
Ding, Mengyuan
;
Shen, Yanyan
  |  
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2025/05/27
New solid forms of tetrahydrocurcumin with improved solubility
期刊论文
OAI收割
CRYSTENGCOMM, 2024, 页码: 8
作者:
Tian, Fanyu
;
Xia, Mengyuan
;
Wang, Hao
;
Zhang, Bingrui
;
Ding, Zhenfeng
  |  
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2024/07/12
Enhancing physical and chemical stability of hygroscopic hydroxytyrosol by cocrystal formation
期刊论文
OAI收割
INTERNATIONAL JOURNAL OF PHARMACEUTICS, 2023, 卷号: 646, 页码: 8
作者:
Zhu, Bingqing
;
Xia, Mengyuan
;
Ding, Zhenfeng
;
Rong, Xiaoyi
;
Mei, Xuefeng
  |  
收藏
  |  
浏览/下载:39/0
  |  
提交时间:2023/12/11
Hydroxytyrosol
Cocrystal
Solidification
Hygroscopicity
Stability
Design, synthesis and biological evaluation of peptidomimetic benzothiazolyl ketones as 3CLpro inhibitors against SARS-CoV-2
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 257, 页码: 13
作者:
Yang, Hanxi
;
You, Mengyuan
;
Shu, Xiaoyang
;
Zhen, Jingyao
;
Zhu, Mengwei
  |  
收藏
  |  
浏览/下载:35/0
  |  
提交时间:2023/10/17
Peptidomimetics
Benzothiazolyl ketone
3CLpro inhibitor
Pharmacokinetic properties
SARS-CoV-2
Development of HSP90 inhibitors-SN38 conjugates for cancer treatment
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2023, 卷号: 137, 页码: 11
作者:
Cao, Yuting
;
Shen, Qianqian
;
Ding, Mengyuan
;
Chen, Yi
;
Lu, Wei
  |  
收藏
  |  
浏览/下载:84/0
  |  
提交时间:2023/10/17
HSP90
SN38 conjugate
Drug accumulation
Cancer treatment
Crystal Engineering to Solidify and Chemically Stabilize Oily dl-Butylphthalide
期刊论文
OAI收割
CRYSTAL GROWTH & DESIGN, 2023, 页码: 11
作者:
Xia, Mengyuan
;
Ding, Zhenfeng
;
Tian, Fanyu
;
Dai, Wenjuan
;
Zhang, Zaiyong
  |  
收藏
  |  
浏览/下载:39/0
  |  
提交时间:2023/10/17
Synthesis, and biological evaluation of EGFR/HER2-NAMPT conjugates for tumor treatment
期刊论文
OAI收割
MOLECULAR DIVERSITY, 2023, 页码: 20
作者:
Ding, Mengyuan
;
Shen, Qianqian
;
Lu, Wei
;
Zhu, Shulei
  |  
收藏
  |  
浏览/下载:110/0
  |  
提交时间:2023/10/17
EGFR
HER2
NAMPT
Resistance
Selectivity
Molecular docking
Design, synthesis and biological evaluation of covalent peptidomimetic 3CL protease inhibitors containing nitrile moiety
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2023, 卷号: 87, 页码: 12
作者:
Zhu, Mengwei
;
Fu, Tiantian
;
You, Mengyuan
;
Cao, Junyuan
;
Yang, Hanxi
  |  
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2023/10/17
COVID-19
SARS-CoV-2
3CL protease
Nirmatrelvir
Peptidomimetic inhibitors