中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共33条,第1-10条 帮助

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One stone two birds: Introducing piperazine into a series of nucleoside derivatives as potent and selective PRMT5 inhibitors 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 281, 页码: 18
作者:  
Li, Huaxuan;  Yang, Hong;  Liu, Li;  Zheng, Jiahong;  Shi, Qiongyu
  |  收藏  |  浏览/下载:12/0  |  提交时间:2024/12/11
Discovery of CZL-046 with an (S)-3-Fluoropyrrolidin-2-one Scaffold as a p300 Bromodomain Inhibitor for the Treatment of Multiple Myeloma 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 20, 页码: 18606-18628
作者:  
Chen, Zonglong;  Yang, Hong;  Zhang, Yan;  Lyu, Xiaodong;  Shi, Qiongyu
  |  收藏  |  浏览/下载:8/0  |  提交时间:2024/11/05
Relationships of stomatal morphology to the environment across plant communities 期刊论文  OAI收割
NATURE COMMUNICATIONS, 2023, 卷号: 14, 期号: 1, 页码: 11
作者:  
Liu, Congcong;  Sack, Lawren;  Li, Ying;  Zhang, Jiahui;  Yu, Kailiang
  |  收藏  |  浏览/下载:13/0  |  提交时间:2024/01/02
Discovery of a New-Generation S-Adenosylmethionine-Noncompetitive Covalent Inhibitor Targeting the Lysine Methyltransferase Enhancer of Zeste Homologue 2 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 66, 期号: 11, 页码: 7629-7644
作者:  
Zhang, Yi;  Yang, Hong;  Li, Bingbing;  Li, Jiayi;  Li, Huaxuan
  |  收藏  |  浏览/下载:33/0  |  提交时间:2023/10/17
Structural Modification and Pharmacological Evaluation of Substituted Quinoline-5,8-diones as Potent NSD2 Inhibitors 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 页码: 18
作者:  
Tang, Hairong;  Yu, Aisong;  Xing, Li;  Chen, Xiaoyu;  Ding, Huaqian
  |  收藏  |  浏览/下载:29/0  |  提交时间:2023/04/10
Structure-activity relationship study of a series of nucleoside derivatives bearing sulfonamide scaffold as potent and selective PRMT5 inhibitors 期刊论文  OAI收割
BIOORGANIC CHEMISTRY, 2023, 卷号: 130, 页码: 20
作者:  
Chen, Yuting;  Shi, Qiongyu;  Yang, Hong;  Li, Jiayi;  Zhou, Kaixin
  |  收藏  |  浏览/下载:33/0  |  提交时间:2023/04/10
New Insights Into Multi-Component Atmospheric Wet Deposition Across China: A Multidimensional Analysis 期刊论文  OAI收割
EARTHS FUTURE, 2022, 卷号: 10, 期号: 11, 页码: 8
作者:  
Zhang, Qiongyu;  Zhu, Jianxing;  Wang, Qiufeng;  Xu, Li;  Li, Mingxu
  |  收藏  |  浏览/下载:28/0  |  提交时间:2022/12/30
New Insights Into Multi-Component Atmospheric Wet Deposition Across China: A Multidimensional Analysis 期刊论文  OAI收割
EARTHS FUTURE, 2022, 卷号: 10, 期号: 11, 页码: 8
作者:  
Zhang, Qiongyu;  Zhu, Jianxing;  Wang, Qiufeng;  Xu, Li;  Li, Mingxu
  |  收藏  |  浏览/下载:21/0  |  提交时间:2022/12/30
Discovery of a potent and selective proteolysis targeting chimera (PROTAC) degrader of NSD3 histone methyltransferase 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 239, 页码: 18
作者:  
Sun, Yaoliang;  Zhang, Ying;  Chen, Xiaoai;  Yu, Aisong;  Du, Wenhao
  |  收藏  |  浏览/下载:62/0  |  提交时间:2022/08/30
Discovery of novel benzimidazole derivatives as potent p300 bromodomain inhibitors with anti-proliferative activity in multiple cancer cells 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2022, 卷号: 66, 页码: 16
作者:  
Chen, Zonglong;  Li, Jiayi;  Yang, Hong;  He, Yulong;  Shi, Qiongyu
  |  收藏  |  浏览/下载:51/0  |  提交时间:2022/08/16