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Design, synthesis, and biological evaluation of thioamide-linked spiropyrrolidine derivatives as novel 3CL
pro
inhibitors against SARS-CoV-2
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2025, 卷号: 128, 页码: 11
作者:
Guma, Samuel Desta
;
Song, Kang
;
Sun, Haiguo
;
Yang, Lei
;
Zhou, Zhaoyin
  |  
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2025/08/20
SARS-CoV-2
3CL(pro) inhibitors
Thioamide derivatives
Spiropyrrolidine derivatives
Nirmatrelvir
HCoV-OC43
Antiviral
Metabolic stability
Design and synthesis of CDK9/EZH2 dual-target inhibitors to achieve synergistic antitumor effects
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 294, 页码: 14
作者:
Tian, Lina
  |  
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2025/08/20
CDK9
EZH2
Dual target inhibitor
DLBCL
The Flat Tail in the Burst Energy Distribution of FRB 20240114A
期刊论文
OAI收割
RESEARCH IN ASTRONOMY AND ASTROPHYSICS, 2025, 卷号: 25, 期号: 8
作者:
Huang YX(黄玉祥)
;
Zhang, Jun-Shuo
;
Xu, Heng
;
Hao LF(郝龙飞)
;
Li KJ(李柯伽)
  |  
收藏
  |  
浏览/下载:33/0
  |  
提交时间:2025/07/14
stars: general
stars: magnetars
radio continuum: stars
stars: neutron
Guiding precision medicine strategy for intravenous ginsenosides via pharmacokinetic-informed bioinformatic approaches: a study on XueShuanTong
期刊论文
OAI收割
PHYTOMEDICINE, 2025, 卷号: 143, 页码: 18
作者:
Jia, Wei-Wei
;
Tian, Nan-Nan
;
Song, Zi-Jing
;
Lan, Xiao-Fang
;
Yang, Xi-He
  |  
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2025/08/20
Precision medicine
Physiologically based pharmacokinetic model
Ginsenoside
Albumin-facilitated dissociation
Drug interaction
Drug transporter
Hepatic impairment
Bright Bursts with Submillisecond Structures of FRB 20230607A in a Highly Magnetized Environment
期刊论文
OAI收割
ASTROPHYSICAL JOURNAL, 2025, 卷号: 988, 期号: 1
作者:
Zhou, DeJiang
;
Han, J. L.
;
Zhang, Bing
;
Zhu, WeiWei
;
Wang, Wei-yang
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2025/07/28
Analysis of the shear failure between track slab and CA mortar layer caused by thermal effect for ballastless track
期刊论文
OAI收割
CASE STUDIES IN CONSTRUCTION MATERIALS, 2025, 卷号: 22, 页码: 16
作者:
Zhang, Tao
;
Zhang, Zheyuan
;
Tian, Hongming
;
Lu, Chen
;
Wang, Wei
  |  
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2025/06/27
Ballastless track
CA mortar
Constitutive model
Damage analysis
Study of ultra-high-energy gamma-ray source 1LHAASO J0056+6346u and its possible origins
期刊论文
OAI收割
SCIENCE CHINA-PHYSICS MECHANICS & ASTRONOMY, 2025, 卷号: 68, 期号: 7
作者:
Cao, Zhen
;
Aharonian, F.
;
Axikegu
;
Bai, Y. X.
;
Bao, Y. W.
  |  
收藏
  |  
浏览/下载:33/0
  |  
提交时间:2025/06/10
gamma rays
cosmic rays
supernova remnant
young massive cluster
pulsar
GATA1-mediated Notch signaling augment antitumor immunity of CD11b+CD27-natural killer cells maturation via BCL9/β-catenin signal
期刊论文
OAI收割
CELL REPORTS, 2025, 卷号: 44, 期号: 5, 页码: 23
作者:
Yang, Fan
;
Li, Anqi
;
Zhu, Yuanyuan
;
Zhou, Yan
;
Tian, Enming
  |  
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2025/08/20
Low perception of climate change by farmers and herders on Tibetan Plateau
期刊论文
OAI收割
GLOBAL ENVIRONMENTAL CHANGE-HUMAN AND POLICY DIMENSIONS, 2025, 卷号: 91, 页码: 102970
作者:
Yi, Jiawei
;
Tian, Yuan
;
Simpson, Nicholas P.
;
Du, Yunyan
;
Ma, Ting
  |  
收藏
  |  
浏览/下载:32/0
  |  
提交时间:2025/03/18
Climate change perception
Survey research
Farmers and herders
Tibetan Plateau
Safety evaluation system of salt cavern hydrogen storage based on matter-element extension method
期刊论文
OAI收割
JOURNAL OF ENERGY STORAGE, 2025, 卷号: 116, 页码: 17
作者:
Fu, Liupeng
;
Shi, Xilin
;
Fan, Jinyang
;
Yang, Chunhe
;
Zhu, Shijie
  |  
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2025/06/27
Salt cavern hydrogen storage (SCHS)
Two-butted-well horizontal (TWH) salt caverns
Novel safety evaluation system
Matter-element extension method