中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共20条,第1-10条 帮助

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Single Amine or Guanidine Modification on Norvancomycin and Vancomycin to Overcome Multidrug-Resistance through Augmented Lipid II Binding and Increased Membrane Activity 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 22, 页码: 20639-20663
作者:  
Bian, Xiaolei;  Chen, Zhifu;  Li, Fang;  Xie, Yuanyuan;  Li, Yi
  |  收藏  |  浏览/下载:5/0  |  提交时间:2024/12/11
A Vancomycin-Templated DNA-Encoded Library for Combating Drug-Resistant Bacteria 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 5, 页码: 3778-3794
作者:  
Guan, Dongliang;  Liu, Jiaxiang;  Chen, Feifei;  Li, Jian;  Wang, Xiaowen
  |  收藏  |  浏览/下载:13/0  |  提交时间:2024/05/07
A facile and selective derivatization approach on kynurenine-NH2 in daptomycin, leading to the discovery of hexakynomycin to combat multidrug-resistant Gram-positive pathogens especially daptomycin-resistant bacteria 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 259, 页码: 14
作者:  
Guan, Dongliang;  Li, Jian;  Chen, Feifei;  Li, Jiaqi;  Bian, Xiaolei
  |  收藏  |  浏览/下载:17/0  |  提交时间:2023/10/17
Carbohydrate Strengthens the Immunotherapeutic Effect of Small-Molecule PD-L1 Inhibitors 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 66, 期号: 11, 页码: 7179-7204
作者:  
Dong, Qian;  Tong, Mengya;  Yu, Xiaolu;  Wang, Lei;  Ao, Jiwei
  |  收藏  |  浏览/下载:40/0  |  提交时间:2023/10/17
Single Modification at the N-Terminus of Norvancomycin to Combat Drug-Resistant Gram-Positive Bacteria 期刊论文  OAI收割
CHEMMEDCHEM, 2023, 卷号: 18, 期号: 9
作者:  
Guan, Dongliang;  Chen, Feifei;  Shi, Wei;  Lan, Lefu;  Huang, Wei
  |  收藏  |  浏览/下载:14/0  |  提交时间:2024/03/27
Potentiation of Vancomycin: Creating Cooperative Membrane Lysis through a "Derivatization-for-Sensitization" Approach 期刊论文  OAI收割
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2022, 卷号: 144, 期号: 23, 页码: 10622-10639
作者:  
Lei, E.;  Tao, Huanyu;  Jiao, Shang;  Yang, Anming;  Zhou, Yu
  |  收藏  |  浏览/下载:42/0  |  提交时间:2022/08/16
Impurity Identification and Scale-Up of a Novel Glycopeptide Antibiotic 期刊论文  OAI收割
ORGANIC PROCESS RESEARCH & DEVELOPMENT, 2021, 卷号: 25, 期号: 11, 页码: 2390-2402
作者:  
Jiao, Shang;  Guan, Dongliang;  Xu, Lili;  Liu, Bo;  Shi, Weiwei
  |  收藏  |  浏览/下载:36/0  |  提交时间:2022/01/18
Total and Semisyntheses of Polymyxin Analogues with 2-Thr or 10-Thr Modifications to Decipher the Structure-Activity Relationship and Improve the Antibacterial Activity 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 9, 页码: 5746-5765
作者:  
Li, Jian;  Guan, Dongliang;  Chen, Feifei;  Shi, Weiwei;  Lan, Lefu
  |  收藏  |  浏览/下载:21/0  |  提交时间:2021/08/17
Selective N-glycan editing on living cell surfaces to probe glycoconjugate function 期刊论文  OAI收割
NATURE CHEMICAL BIOLOGY, 2020, 页码: 15
作者:  
Tang, Feng;  Zhou, Mang;  Qin, Ken;  Shi, Wei;  Yashinov, Ansor
  |  收藏  |  浏览/下载:38/0  |  提交时间:2020/07/01
New linker structures applied in glycosite-specific antibody drug conjugates 期刊论文  OAI收割
ORGANIC CHEMISTRY FRONTIERS, 2019, 卷号: 6, 期号: 17, 页码: 3144-3149
作者:  
Faridoon;  Shi, Wei;  Qin, Ken;  Tang, Yubo;  Li, Mingjie
  |  收藏  |  浏览/下载:37/0  |  提交时间:2020/07/01