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Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [18]
金属研究所 [1]
古脊椎动物与古人类研... [1]
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OAI收割 [20]
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期刊论文 [20]
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2024 [2]
2023 [3]
2022 [1]
2021 [2]
2020 [1]
2019 [3]
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Materials ... [1]
Metallurgy... [1]
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Single Amine or Guanidine Modification on Norvancomycin and Vancomycin to Overcome Multidrug-Resistance through Augmented Lipid II Binding and Increased Membrane Activity
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 22, 页码: 20639-20663
作者:
Bian, Xiaolei
;
Chen, Zhifu
;
Li, Fang
;
Xie, Yuanyuan
;
Li, Yi
  |  
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2024/12/11
A Vancomycin-Templated DNA-Encoded Library for Combating Drug-Resistant Bacteria
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 5, 页码: 3778-3794
作者:
Guan, Dongliang
;
Liu, Jiaxiang
;
Chen, Feifei
;
Li, Jian
;
Wang, Xiaowen
  |  
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2024/05/07
A facile and selective derivatization approach on kynurenine-NH2 in daptomycin, leading to the discovery of hexakynomycin to combat multidrug-resistant Gram-positive pathogens especially daptomycin-resistant bacteria
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 259, 页码: 14
作者:
Guan, Dongliang
;
Li, Jian
;
Chen, Feifei
;
Li, Jiaqi
;
Bian, Xiaolei
  |  
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2023/10/17
Lipopeptide
Daptomycin derivatives
Multidrug-resistant bacteria
Kynurenine
Hexakynomycin
Carbohydrate Strengthens the Immunotherapeutic Effect of Small-Molecule PD-L1 Inhibitors
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 66, 期号: 11, 页码: 7179-7204
作者:
Dong, Qian
;
Tong, Mengya
;
Yu, Xiaolu
;
Wang, Lei
;
Ao, Jiwei
  |  
收藏
  |  
浏览/下载:40/0
  |  
提交时间:2023/10/17
Single Modification at the N-Terminus of Norvancomycin to Combat Drug-Resistant Gram-Positive Bacteria
期刊论文
OAI收割
CHEMMEDCHEM, 2023, 卷号: 18, 期号: 9
作者:
Guan, Dongliang
;
Chen, Feifei
;
Shi, Wei
;
Lan, Lefu
;
Huang, Wei
  |  
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2024/03/27
norvancomycin
glycopeptide antibiotics
single modification
sulfonium
bacterial resistance
Potentiation of Vancomycin: Creating Cooperative Membrane Lysis through a "Derivatization-for-Sensitization" Approach
期刊论文
OAI收割
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2022, 卷号: 144, 期号: 23, 页码: 10622-10639
作者:
Lei, E.
;
Tao, Huanyu
;
Jiao, Shang
;
Yang, Anming
;
Zhou, Yu
  |  
收藏
  |  
浏览/下载:42/0
  |  
提交时间:2022/08/16
Impurity Identification and Scale-Up of a Novel Glycopeptide Antibiotic
期刊论文
OAI收割
ORGANIC PROCESS RESEARCH & DEVELOPMENT, 2021, 卷号: 25, 期号: 11, 页码: 2390-2402
作者:
Jiao, Shang
;
Guan, Dongliang
;
Xu, Lili
;
Liu, Bo
;
Shi, Weiwei
  |  
收藏
  |  
浏览/下载:36/0
  |  
提交时间:2022/01/18
glycopeptide antibiotics
impurity
analytical method
process optimization and development
Total and Semisyntheses of Polymyxin Analogues with 2-Thr or 10-Thr Modifications to Decipher the Structure-Activity Relationship and Improve the Antibacterial Activity
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 9, 页码: 5746-5765
作者:
Li, Jian
;
Guan, Dongliang
;
Chen, Feifei
;
Shi, Weiwei
;
Lan, Lefu
  |  
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2021/08/17
Selective N-glycan editing on living cell surfaces to probe glycoconjugate function
期刊论文
OAI收割
NATURE CHEMICAL BIOLOGY, 2020, 页码: 15
作者:
Tang, Feng
;
Zhou, Mang
;
Qin, Ken
;
Shi, Wei
;
Yashinov, Ansor
  |  
收藏
  |  
浏览/下载:38/0
  |  
提交时间:2020/07/01
New linker structures applied in glycosite-specific antibody drug conjugates
期刊论文
OAI收割
ORGANIC CHEMISTRY FRONTIERS, 2019, 卷号: 6, 期号: 17, 页码: 3144-3149
作者:
Faridoon
;
Shi, Wei
;
Qin, Ken
;
Tang, Yubo
;
Li, Mingjie
  |  
收藏
  |  
浏览/下载:37/0
  |  
提交时间:2020/07/01