中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共28条,第1-10条 帮助

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Berberine Derivative B68 Promotes Tumor Immune Clearance by Dual-Targeting BMI1 for Senescence Induction and CSN5 for PD-L1 Degradation 期刊论文  OAI收割
ADVANCED SCIENCE, 2024, 页码: 21
作者:  
Hu, Hongmei;  Wang, Qun;  Yu, Dianping;  Tao, Xiaoyu;  Guo, Mengmeng
  |  收藏  |  浏览/下载:6/0  |  提交时间:2025/02/28
Rh(III)-catalyzed late-stage C-H alkenylation and macrolactamization for the synthesis of cyclic peptides with unique Trp(C7)-alkene crosslinks 期刊论文  OAI收割
CHINESE CHEMICAL LETTERS, 2024, 卷号: 35, 期号: 8, 页码: 8
作者:  
Hu, Shulei;  Zhang, Yu;  Xie, Xiong;  Li, Luhan;  Chen, Kaixian
  |  收藏  |  浏览/下载:3/0  |  提交时间:2024/11/05
Discovery of Small-Molecule Degraders of the CDK9-Cyclin T1 Complex for Targeting Transcriptional Addiction in Prostate Cancer 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 65, 期号: 16, 页码: 11034-11057
作者:  
Li, Jiacheng;  Liu, Ting;  Song, Yuanli;  Wang, Mingyu;  Liu, Liping
  |  收藏  |  浏览/下载:17/0  |  提交时间:2024/03/21
L-5-hydroxytryptophan promotes antitumor immunity by inhibiting PD-L1 inducible expression 期刊论文  OAI收割
JOURNAL FOR IMMUNOTHERAPY OF CANCER, 2022, 卷号: 10, 期号: 6, 页码: 14
作者:  
Huang, Jing;  Wang, Xiaobo;  Li, Bing;  Shen, Shiyu;  Wang, Ruina
  |  收藏  |  浏览/下载:33/0  |  提交时间:2022/08/16
Inhibition of Autophagy by a Small Molecule through Covalent Modification of the LC3 Protein 期刊论文  OAI收割
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2021, 页码: 11
作者:  
Fan, Shijie;  Yue, Liyan;  Wan, Wei;  Zhang, Yuanyuan;  Zhang, Bidong
  |  收藏  |  浏览/下载:111/0  |  提交时间:2021/12/16
Expert consensus on thermal ablation therapy of pulmonary subsolid nodules (2021 Edition) 期刊论文  OAI收割
JOURNAL OF CANCER RESEARCH AND THERAPEUTICS, 2021, 卷号: 17
作者:  
Ye, Xin;  Fan, Weijun;  Wang, Zhongmin;  Wang, Junjie;  Wang, Hui
  |  收藏  |  浏览/下载:70/0  |  提交时间:2022/03/21
Dynamics of Post-Translational Modification Inspires Drug Design in the Kinase Family 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 20, 页码: 15111-15125
作者:  
Zhang, Huimin;  He, Jixiao;  Hu, Guang;  Zhu, Fei;  Jiang, Hao
  |  收藏  |  浏览/下载:70/0  |  提交时间:2022/01/04
Discovery of a subtype-selective, covalent inhibitor against palmitoylation pocket of TEAD3 期刊论文  OAI收割
ACTA PHARMACEUTICA SINICA B, 2021, 卷号: 11, 期号: 10, 页码: 3206-3219
作者:  
Lu, Tian;  Li, Yong;  Lu, Wenchao;  Spitters, Twgm;  Fang, Xueyu
  |  收藏  |  浏览/下载:52/0  |  提交时间:2021/12/01
The dynamic conformational landscape of the protein methyltransferase SETD8 期刊论文  OAI收割
ELIFE, 2019, 卷号: 8, 页码: 76
作者:  
Chen, Shi;  Wiewiora, Rafal P.;  Meng, Fanwang;  Babault, Nicolas;  Ma, Anqi
  |  收藏  |  浏览/下载:30/0  |  提交时间:2020/07/01
Rational design of 5-((1H-imidazol-1-yl)methyl)quinolin-8-ol derivatives as novel bromodomain-containing protein 4 inhibitors 期刊论文  OAI收割
European journal of medicinal chemistry, 2018, 卷号: 163, 页码: 281-294
作者:  
Xing, Jing;  Zhang, Rukang;  Jiang, Xiangrui;  Hu, Tianwen;  Wang, Xinjun
  |  收藏  |  浏览/下载:101/0  |  提交时间:2019/01/08