中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共47条,第1-10条 帮助

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Design of Selective BRD4 Inhibitors for the Treatment of Autosomal Dominant Polycystic Kidney Disease 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 页码: 18
作者:  
Yang, Yueyue;  Liu, Hongli;  Yuan, Haoxing;  Lyu, Kaikai;  Zhong, Haiyang
  |  收藏  |  浏览/下载:16/0  |  提交时间:2025/04/01
Structure-Based Rational Design and Evaluation of BET-Aurora Kinase Dual-Inhibitors for Treatment of Cancers 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 页码: 21
作者:  
Lyu, Kaikai;  Ren, Ying;  Mou, Jie;  Yang, Yunfang;  Pan, Yaoyao
  |  收藏  |  浏览/下载:17/0  |  提交时间:2025/02/28
Design and development of a series of 4-(piperazin-1-yl)pyrimidines as irreversible menin inhibitors 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 280, 页码: 20
作者:  
Luo, Menglan;  Ye, Yunfei;  Tang, Lu;  Kan, Weijuan;  Chen, Lin
  |  收藏  |  浏览/下载:15/0  |  提交时间:2024/11/26
Remodeling tumor-associated macrophage for anti-cancer effects by rational design of irreversible inhibition of mitogen-activated protein kinase-activated protein kinase 2 期刊论文  OAI收割
MEDCOMM, 2024, 卷号: 5, 期号: 7, 页码: e634
作者:  
Wang, Danyi;  Sun, Deqiao;  Wang, Xiaoyan;  Peng, Xia;  Ji, Yinchun
  |  收藏  |  浏览/下载:1/0  |  提交时间:2025/06/04
Development of a series of quinazoline-2,5-diamine derivatives as potent hematopoietic progenitor kinase 1 (HPK1) inhibitors 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 248, 页码: 20
作者:  
Shi, Huanyu;  Tang, Haotian;  Li, Yan;  Chen, Danqi;  Liu, Tongchao
  |  收藏  |  浏览/下载:35/0  |  提交时间:2023/04/10
Design, synthesis and biological evaluation of 4-aminoquinoline derivatives as receptor-interacting protein kinase 2 (RIPK2) inhibitors 期刊论文  OAI收割
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, 2023, 卷号: 38, 期号: 1, 页码: 282-293
作者:  
Fan, Tiantian;  Ji, Yinchun;  Chen, Danqi;  Peng, Xia;  Ai, Jing
  |  收藏  |  浏览/下载:28/0  |  提交时间:2023/04/10
Design and development of a novel series of oral bivalent BET inhibitors with potent anticancer activities 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 239, 页码: 13
作者:  
Luo, Menglan;  Wu, Qian;  Yang, Yueyue;  Sun, Lin;  Huan, Xiajuan
  |  收藏  |  浏览/下载:60/0  |  提交时间:2022/08/30
Discovery of 4-cyclopropyl-3-(2-((1-cyclopropyl-1H-pyrazol-4-yl) amino) quinazolin-6-yl)-N-(3-(trifluoromethyl) phenyl) benzamides as potent discoidin domain receptor inhibitors for the treatment of idiopathic pulmonary fibrosis 期刊论文  OAI收割
ACTA PHARMACEUTICA SINICA B, 2022, 卷号: 12, 期号: 4, 页码: 1943-1962
作者:  
Wang, Qi;  Tang, Bixi;  Sun, Dandan;  Dong, Ying;  Ji, Yinchun
  |  收藏  |  浏览/下载:38/0  |  提交时间:2022/08/16
可持续发展目标视野下中国食物系统转型的战略思考 期刊论文  OAI收割
中国科学院院刊, 2022, 卷号: N/A, 页码: 12
作者:  
刘晓洁;  贺思琪;  陈伟强;  闫丹;  刘立涛
  |  收藏  |  浏览/下载:36/0  |  提交时间:2023/01/04
Structure-Based Discovery of Potent CARM1 Inhibitors for Solid Tumor and Cancer Immunology Therapy 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 22, 页码: 16650-16674
作者:  
Zhang, Zhuqing;  Guo, Zuhao;  Xu, Xiaowei;  Cao, Danyan;  Yang, Hong
  |  收藏  |  浏览/下载:46/0  |  提交时间:2022/06/15