中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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BMAL1/PGC1a4-FNDC5/irisin axis impacts distinct outcomes of time-of-day resistance exercise
期刊论文
OAI收割
JOURNAL OF SPORT AND HEALTH SCIENCE, 2025, 卷号: 14, 页码: 23
作者:
Guo, Mingwei
;
Shen, Fei
;
Guo, Xiaozhen
;
Zhang, Jun
;
Ma, Ying
  |  
收藏
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浏览/下载:111/0
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提交时间:2025/04/01
Daily variance
Circadian
Muscle strength
Metabolic benefits
Resistance exercise
Pharmacokinetics, mass balance, and metabolism of [
14
C]PLB1004, a selective and irreversible EGFR-TKI in humans
期刊论文
OAI收割
CANCER CHEMOTHERAPY AND PHARMACOLOGY, 2025, 卷号: 95, 期号: 1, 页码: 14
作者:
Liu, Donghui
;
Li, Qian
;
Yan, Shu
;
Zhang, Xinyue
;
Li, Weiqiang
  |  
收藏
  |  
浏览/下载:38/0
  |  
提交时间:2025/04/01
PLB1004
[C-14]PLB1004
Radioactivity
Mass balance
EGFR-TKI
Pharmacokinetics, mass balance, and metabolism of [
14
C]FCN-437c, a selective and potent CDK4/6 inhibitor in humans
期刊论文
OAI收割
CANCER CHEMOTHERAPY AND PHARMACOLOGY, 2025, 卷号: 95, 期号: 1, 页码: 12
作者:
Gao, Lei
;
Ma, Sheng
;
Yan, Shu
;
Zhang, Hua
;
Tian, Ling
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2025/07/25
FCN-437c
CDK4/6 inhibitor
Mass balance
Radiopharmacokinetics
Drug metabolism
Discovery of pyrrolo[2,3-d]pyrimidine derivatives as novel FLT3/ IRAK4 inhibitors
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 296, 页码: 23
作者:
Yuan, Haibin
;
Gao, Yue
;
Wang, Peipei
;
Dong, Xiaowu
;
Li, Jia
  |  
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2025/08/20
AML
FLT3/IRAK4 inhibitor
Pyrrolo [2,3-d] pyrimidine
Acquired resistance
Adaptive resistance
Torque work of origin-destination flows: Quantifying urban place centrality from a physical perspective
期刊论文
OAI收割
COMPUTERS ENVIRONMENT AND URBAN SYSTEMS, 2025, 卷号: 121, 页码: 102311
作者:
Yan, Xiaorui
;
Pei, Tao
;
Song, Ci
;
Fang, Zidong
;
Liu, Xiaohan
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2025/07/18
Place centrality
Origin-destination flows
Torque work
Multiscale analysis
Intra-day dynamic
Urban science
Conformational restriction enables discovering a series of chroman derivatives as potent and selective NaV1.8 inhibitors with improved pharmacokinetic properties
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 293, 页码: 24
作者:
Li, Na
  |  
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2025/08/20
Voltage-gated sodium channel 1.8
Conformational restriction
Pharmacokinetic
Structure-activity relationship
Analgesic
Hepatic IκBζpromotes alcohol-associated liver disease and acute hepatitis by enhancing CXCL1-Mediated neutrophil infiltration
期刊论文
OAI收割
FREE RADICAL BIOLOGY AND MEDICINE, 2025, 卷号: 237, 页码: 558-569
作者:
Liu, Li
;
Qian, Shengying
;
Li, Wenjun
;
Dong, Siyue
;
Ya, Ru
  |  
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2025/08/20
Nfkbiz
ALD
Acute liver injury
GalNac
Inhibition of α-synuclein aggregation by MCC950 attenuates dopaminergic neuronal damage in MN9D cells
期刊论文
OAI收割
EUROPEAN JOURNAL OF PHARMACOLOGY, 2025, 卷号: 1001, 页码: 10
作者:
Gao, Huiwen
;
Liang, Yingneng
;
Wang, Mengfei
;
Li, Wen
;
Zheng, Wei
  |  
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2025/08/20
alpha-synuclein
MCC950
Parkinson's disease
Neuroprotection
Widespread consistent but rapid response of terrestrial ecosystem photosynthesis and respiratory to drought
期刊论文
OAI收割
JOURNAL OF HYDROLOGY, 2025, 卷号: 657, 页码: 133107
作者:
  |  
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2025/04/21
Gross primary productivity
Ecosystem respiration
Drought
Response time dynamics
Recent advances in traditional Chinese medicine metabolism: Sample pre-treatment, MS-oriented analytical strategies and typical applications
期刊论文
OAI收割
TRAC-TRENDS IN ANALYTICAL CHEMISTRY, 2025, 卷号: 189, 页码: 22
作者:
Hong, Li-li
;
Cui, Dian-xin
;
Wang, Hong-da
;
Jing, Qi
;
Li, Xue
  |  
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2025/06/23
Traditional Chinese medicine metabolism
Bio-samples pre-treatment
Mass spectrometry
Data acquisition
Data processing
Application