中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [6]
广州生物医药与健康研... [2]
采集方式
OAI收割 [8]
内容类型
期刊论文 [8]
发表日期
2022 [2]
2021 [1]
2020 [1]
2018 [1]
2015 [3]
学科主题
Chemistry [2]
Pharmacolo... [2]
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ASK120067 potently suppresses B-cell or T-cell malignancies in vitro and in vivo by inhibiting BTK and ITK
期刊论文
OAI收割
FRONTIERS IN PHARMACOLOGY, 2022, 卷号: 13, 页码: 9
作者:
Song, Peiran
;
Bai, Gang
;
Chan, Shingpan
;
Zhang, Tao
;
Tong, Linjiang
  |  
收藏
  |  
浏览/下载:39/0
  |  
提交时间:2023/04/10
Bruton's tyrosine kinase
interleukin-2-inducible T cell kinase
ASK120067
B-cell lymphoma
T-cell leukemia
Discovery of 3-Aminopyrazole Derivatives as New Potent and Orally Bioavailable AXL Inhibitors
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 65, 期号: 22, 页码: 15374-15390
作者:
Chan, Shingpan
;
Zhang, Yunong
;
Wang, Jie
;
Yu, Qiuchun
;
Peng, Xia
  |  
收藏
  |  
浏览/下载:35/0
  |  
提交时间:2023/04/10
Correction to: Discovery of a novel third-generation EGFR inhibitor and identification of a potential combination strategy to overcome resistance
期刊论文
OAI收割
Molecular Cancer, 2021, 卷号: 20, 期号: 1
作者:
Zhang,Tao
;
Qu,Rong
  |  
收藏
  |  
浏览/下载:68/0
  |  
提交时间:2021/11/04
Discovery of a novel third-generation EGFR inhibitor and identification of a potential combination strategy to overcome resistance
期刊论文
OAI收割
MOLECULAR CANCER, 2020, 卷号: 19, 期号: 1, 页码: 15
作者:
Zhang, Tao
;
Qu, Rong
;
Chan, Shingpan
;
Lai, Mengzhen
;
Tong, Linjiang
  |  
收藏
  |  
浏览/下载:89/0
  |  
提交时间:2020/07/01
Non-small cell lung cancer (NSCLC)
EGFR T790M
Small-molecule inhibitor
Drug resistance
Ack1
Discovery of JND3229 as a New EGFR(C797S) Mutant Inhibitor with In Vivo Monodrug Efficacy
期刊论文
OAI收割
ACS MEDICINAL CHEMISTRY LETTERS, 2018, 卷号: 9, 期号: 11, 页码: 1123-1127
作者:
Lu, Xiaoyun
;
Zhang, Tao
;
Zhu, Su-Jie
;
Xun, Qiuju
;
Tong, Lingjiang
  |  
收藏
  |  
浏览/下载:120/0
  |  
提交时间:2019/01/08
EGFR(C797s)
Clinical resistance
Fourth-generation nhibitors
Monodrug efficacy
2,4-Diarylamino-pyrimidines as kinase inhibitors co-targeting IGF1R and EGFR(L858R/T790M)
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2015, 卷号: 25, 期号: 19, 页码: 4277-4281
作者:
Chan, Shingpan
;
Han, Kun
;
Qu, Rong
;
Tong, Linjiang
;
Li, Yingjun
  |  
收藏
  |  
浏览/下载:51/0
  |  
提交时间:2019/01/08
EGFR
IGF1R
NSCLC
Dual inhibitor
2,4-Diarylamino-pyrimidines as kinase inhibitors co-targeting IGF1R and EGFR(L858R/T790M)
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2015, 卷号: 25, 期号: 19, 页码: 4277-4281
Chan, Shingpan
;
Han, Kun
;
Qu, Rong
;
Tong, Linjiang
;
Li, Yingjun
;
Zhang, Zhang
;
Cheng, Huimin
;
Lu, Xiaoyun
;
Patterson, Adam
;
Smaill, Jeff
;
Ren, Xiaomei
;
Ding, Jian
;
Xie, Hua
;
Ding, Ke
收藏
  |  
浏览/下载:253/0
  |  
提交时间:2016/12/16
2,4-Diarylamino-pyrimidines as kinase inhibitors co-targeting IGF1R and EGFR(L858R/T790M)
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2015, 卷号: 25, 期号: 19, 页码: 4277-4281
作者:
Smaill, Jeff
;
Lu, Xiaoyun
;
Cheng, Huimin
;
Zhang, Zhang
;
Li, Yingjun
  |  
收藏
  |  
浏览/下载:57/0
  |  
提交时间:2018/12/13