中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共33条,第1-10条 帮助

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Design, Synthesis, and Pharmacological Evaluation of Quinazoline and Quinoline Derivatives as Potent ENPP1 Inhibitors for Cancer Immunotherapy 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 页码: 18
作者:  
He, Jie;  Ma, Xiaoyu;  Sun, Jia;  Chen, Manman;  Xu, Lan
  |  收藏  |  浏览/下载:7/0  |  提交时间:2025/04/01
METI: deep profiling of tumor ecosystems by integrating cell morphology and spatial transcriptomics 期刊论文  OAI收割
NATURE COMMUNICATIONS, 2024, 卷号: 15
作者:  
Jiang, Jiahui;  Liu, Yunhe;  Qin, Jiangjiang;  Chen, Jianfeng;  Wu, Jingjing
  |  收藏  |  浏览/下载:8/0  |  提交时间:2024/11/20
Discovery of Pyrido[2,3-d]pyrimidin-7-one Derivatives as Highly Potent and Efficacious Ectonucleotide Pyrophosphatase/Phosphodiesterase 1 (ENPP1) Inhibitors for Cancer Treatment 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 5, 页码: 3986-4006
作者:  
Sun, Yaoliang;  Chen, Manman;  Han, Yuyan;  Li, Weiqiang;  Ma, Xiaoyu
  |  收藏  |  浏览/下载:21/0  |  提交时间:2024/05/07
Intact regulation of G1/S transition renders esophageal squamous cell carcinoma sensitive to PI3Kα inhibitors 期刊论文  OAI收割
SIGNAL TRANSDUCTION AND TARGETED THERAPY, 2023, 卷号: 8, 期号: 1, 页码: 153
作者:  
Zhang, Xu;  Wang, Yuxiang;  Zhang, Xi;  Shen, Yanyan;  Yang, Kang
  |  收藏  |  浏览/下载:20/0  |  提交时间:2024/03/27
SAF-248,a novel PI3Kδ-selective inhibitor,potently suppresses the growth of diffuse large B-cell lymphoma 期刊论文  OAI收割
ACTA PHARMACOLOGICA SINICA, 2022, 卷号: 43, 期号: 1, 页码: 209
作者:  
Zhang Xi;  Duan Yuting;  Wang Yi;  Zhao Xingdong;  Sun Yiming
  |  收藏  |  浏览/下载:17/0  |  提交时间:2023/05/22
PI3K alpha inhibitor impairs AKT phosphorylation and synergizes with novel angiogenesis inhibitor AL3810 in human hepatocellular carcinoma 期刊论文  OAI收割
SIGNAL TRANSDUCTION AND TARGETED THERAPY, 2021, 卷号: 6, 期号: 1, 页码: 3
作者:  
Xie, Qin;  Chi, Shuaishuai;  Fang, Yanfen;  Sun, Yiming;  Meng, Linghua
  |  收藏  |  浏览/下载:18/0  |  提交时间:2021/05/24
Evolution of DNA methylome from precancerous lesions to invasive lung adenocarcinomas 期刊论文  OAI收割
NATURE COMMUNICATIONS, 2021, 卷号: 12
作者:  
Hu, Xin;  Estecio, Marcos R.;  Chen, Runzhe;  Reuben, Alexandre;  Wang, Linghua
  |  收藏  |  浏览/下载:34/0  |  提交时间:2021/09/06
N-Cyclic sulfamoylaminoethyl substituted 1,2,5-oxadiazol-3-amines as new indoleamine 2, 3-dioxygenase 1 (IDO1) inhibitors. 期刊论文  OAI收割
CANCER IMMUNOLOGY RESEARCH, 2020, 卷号: 8, 期号: 3, 页码: 51-51
作者:  
Chen, Shulun;  Guo, Wei;  Sun, Pu;  Meng, Linghua;  Zhang, Ao
  |  收藏  |  浏览/下载:13/0  |  提交时间:2020/07/01
Design, synthesis and antitumor study of a series of N-Cyclic sulfamoylaminoethyl substituted 1,2,5-oxadiazol-3-amines as new indoleamine 2, 3-dioxygenase 1 (IDO1) inhibitors 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 179, 页码: 38-55
作者:  
Chen, Shulun;  Guo, Wei;  Liu, Xiaohua;  Sun, Pu;  Wang, Yi
  |  收藏  |  浏览/下载:24/0  |  提交时间:2020/07/01
Simultaneous inhibition of PI3K alpha and CDK4/6 synergistically suppresses KRAS-mutated non-small cell lung cancer 期刊论文  OAI收割
CANCER BIOLOGY & MEDICINE, 2019, 卷号: 16, 期号: 1, 页码: 66-+
作者:  
Wang, Yuxiang;  Li, Xian;  Liu, Xueling;  Chen, Yi;  Yang, Chunhao
  |  收藏  |  浏览/下载:26/0  |  提交时间:2020/07/01
PI3K alpha  CDK4/6  KRAS  NSCLC  CYH33