中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
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上海药物研究所 [64]
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期刊论文 [254]
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Identification of Dihydrobenzofuran Neolignans as Novel PDE4 Inhibitors and Evaluation of Antiatopic Dermatitis Efficacy in DNCB-Induced Mice Model
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 6, 页码: 4855-4869
作者:
Gu, Chenming
;
Liu, Jiayuan
;
Qian, Fei
;
Yu, Wenchao
;
Huang, Doudou
  |  
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2024/05/07
Metabolic regulation of homologous recombination repair by MRE11 lactylation
期刊论文
OAI收割
CELL, 2024, 卷号: 187, 期号: 2, 页码: 40
作者:
Chen, Yuping
;
Wu, Jinhuan
;
Zhai, Linhui
;
Zhang, Tingting
;
Yin, Hui
  |  
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2024/04/09
The emergence of machine learning force fields in drug design
期刊论文
OAI收割
MEDICINAL RESEARCH REVIEWS, 2024, 页码: 36
作者:
Chen, Mingan
;
Jiang, Xinyu
;
Zhang, Lehan
;
Chen, Xiaoxu
;
Wen, Yiming
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2024/02/19
computational chemistry
drug design
force field
machine learning
molecular modeling
Reliability and Validity of Warwick-Edinburgh Mental Well-Being Scale among Chinese Civil Servants
期刊论文
OAI收割
INTERNATIONAL JOURNAL OF MENTAL HEALTH PROMOTION, 2024, 卷号: 26, 期号: 1, 页码: 61-67
作者:
Lei, Shulan
;
Wang, Shujuan
;
Zhu, Zhuohong
;
Lu, Min
;
Li, Xinying
  |  
收藏
  |  
浏览/下载:0/0
  |  
提交时间:2024/05/05
Reliability
validity
Warwick-Edinburgh Mental Well-Being Scale
Chinese civil servants
Preclinical and early clinical studies of a novel compound SYHA1813 that efficiently crosses the blood-brain barrier and exhibits potent activity against glioblastoma
期刊论文
OAI收割
ACTA PHARMACEUTICA SINICA B, 2023, 卷号: 13, 期号: 12, 页码: 4748-4764
作者:
Liu, Yingqiang
;
Zhan, Zhengsheng
;
Kang, Zhuang
;
Li, Mengyuan
;
Lv, Yongcong
  |  
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2024/01/26
Small molecule inhibitor
Tumor microenvironment
Immune-checkpoint
immune-deficient mouse models
including temozolomide (TMZ) insensitive tumors. Notably
Bioinspired soft robots for deep-sea exploration
期刊论文
OAI收割
NATURE COMMUNICATIONS, 2023, 卷号: 14, 期号: 1, 页码: 10
作者:
Li, Guorui
;
Wong, Tuck-Whye
;
Shih, Benjamin
;
Guo, Chunyu
;
Wang, Luwen
  |  
收藏
  |  
浏览/下载:33/0
  |  
提交时间:2024/01/03
SOTEM exploration and reservoir structure analysis of Yangbajain geothermal field, Xizang
期刊论文
OAI收割
CHINESE JOURNAL OF GEOPHYSICS-CHINESE EDITION, 2023, 卷号: 66, 期号: 11, 页码: 4805-4816
作者:
Chen WeiYing
;
Xue GuoQiang
;
Zhao Ping
;
Ren WangQi
;
He YiMing
  |  
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2024/01/02
Yangbajain geothermal field
SOTEM
Electrical structure
Migration pathway
Reservoir structure
Design, synthesis and biological evaluation of chalcone derivatives as potent and orally active hCYP3A4 inhibitors
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2023, 卷号: 95, 页码: 9
作者:
Lu, Shiwei
;
Zhang, Feng
;
Gong, Jiahao
;
Huang, Jian
;
Zhu, Guanghao
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2023/12/08
Cytochrome P450 3A4 (CYP3A4)
Inhibitors
Isoquinoline chalcones
Orally active
Design, synthesis and biological evaluation of salicylanilides as novel allosteric inhibitors of human pancreatic lipase
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2023, 卷号: 91, 页码: 11
作者:
Zhao, Yitian
;
Zhang, Min
;
Hou, Xudong
;
Han, Jiaxin
;
Qin, Xiaoya
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2023/10/17
Salicylanilide
hPL inhibitor
Structure -activity relationship
Anti -obesity
Three-dimensional electrical structure model of the Yangbajain geothermal field in Tibet: Evidence obtained from magnetotelluric data
期刊论文
OAI收割
SCIENCE CHINA-EARTH SCIENCES, 2023, 页码: 14
作者:
Xue, Guoqiang
;
Chen, Weiying
;
Zhao, Ping
;
Ren, Wangqi
;
He, Yiming
  |  
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2024/01/02
Geothermal field
Magnetotelluric
Partial melt body
3D electrical structure
Thermal reservoir geological model