中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [20]
合肥物质科学研究院 [16]
金属研究所 [13]
地球环境研究所 [7]
深圳先进技术研究院 [6]
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期刊论文 [115]
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2024 [4]
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Discovery of the First BRD4 Second Bromodomain (BD2)-Selective Inhibitors
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 23, 页码: 21577-21616
作者:
Li, Junhua
;
Hu, Qingqing
;
Zhu, Run
;
Dong, Ruibo
;
Shen, Hui
  |  
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2025/01/10
Structural mechanism of human HCN1 hyperpolarization-activated channel inhibition by ivabradine
期刊论文
OAI收割
JOURNAL OF BIOLOGICAL CHEMISTRY, 2024, 卷号: 300, 期号: 11, 页码: 9
作者:
Che, Tong
;
Zhang, Wei
;
Cheng, Xinyu
;
Lv, Sijia
;
Zhang, Minqing
  |  
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2024/11/26
Discovery of Alkyl Conjugated Diene Diacids as Novel ACLY Inhibitors
期刊论文
OAI收割
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2024, 卷号: 44, 期号: 11, 页码: 3476-3489
作者:
Cheng, Tingting
;
Song, Gaolei
;
Cheng, Long
;
Wang, Fan
;
Sun, Xinyu
  |  
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2025/02/28
metabolic diseases
ATP-citrate lyase (ACLY)
lipogenesis
ACLY inhibitors
dienyldicarboxylic acid
Cryo-EM structure of human HCN3 channel and its regulation by cAMP
期刊论文
OAI收割
JOURNAL OF BIOLOGICAL CHEMISTRY, 2024, 卷号: 300, 期号: 6, 页码: 10
作者:
Yu, Bo
;
Lu, Qiuyuan
;
Li, Jian
;
Cheng, Xinyu
;
Hu, Han
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2024/12/11
D3CARP: a comprehensive platform with multiple-conformation based docking, ligand similarity search and deep learning approaches for target prediction and virtual screening
期刊论文
OAI收割
COMPUTERS IN BIOLOGY AND MEDICINE, 2023, 卷号: 164, 页码: 8
作者:
Shi, Yulong
  |  
收藏
  |  
浏览/下载:37/0
  |  
提交时间:2023/10/17
Target prediction
Virtual screening
Molecular docking
Ligand similarity search
Deep learning
Effect of cold rolling on microstructure, texture, and tensile properties of a Ni-Fe-based superalloy
期刊论文
OAI收割
JOURNAL OF ALLOYS AND COMPOUNDS, 2023, 卷号: 937, 页码: 14
作者:
Wang, Jiaqi
;
Cheng, Sihan
;
Wu, Yunsheng
;
Wang, Tingting
;
Qin, Xuezhi
  |  
收藏
  |  
浏览/下载:46/0
  |  
提交时间:2023/05/09
Ni-Fe-based superalloy
Cold rolling
Microstructure
Texture
Strength
Deformation twinning
Impact of aging on the sources, volatility, and viscosity of organic aerosols in Chinese outflows
期刊论文
OAI收割
ATMOSPHERIC CHEMISTRY AND PHYSICS, 2023, 卷号: 23, 期号: 1, 页码: 611-636
作者:
Feng, Tingting
;
Wang, Yingkun
;
Hu, Weiwei
;
Zhu, Ming
;
Song, Wei
  |  
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2024/08/21
Multi-decadal to centennial scales variability in the East Asian Summer Monsoon around the 5.5 kyr BP climate event
期刊论文
OAI收割
PALAEOGEOGRAPHY PALAEOCLIMATOLOGY PALAEOECOLOGY, 2022, 卷号: 607, 页码: 8
作者:
Wang, Fang
;
Cai, Binggui
;
Shen, Chuan-Chou
;
Cheng, Hai
;
Li, Miaofa
  |  
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2023/03/29
Asian summer monsoon
5
5 kyr B
P
event
Stalagmite
Oxygen isotope
Northeastern China
A potent PGK1 antagonist reveals PGK1 regulates the production of IL-1 beta and IL-6
期刊论文
OAI收割
ACTA PHARMACEUTICA SINICA B, 2022, 卷号: 12, 期号: 11, 页码: 4180-4192
作者:
Liao, Liping
;
Dang, Wenzhen
;
Lin, Tingting
;
Yu, Jinghua
;
Liu, Tonghai
  |  
收藏
  |  
浏览/下载:31/0
  |  
提交时间:2023/04/10
Glycolysis
Phosphoglycerate kinase 1
Macrophages
NRF2
Inflammation
Semiconductor-metal transition in lead iodide under pressure
期刊论文
OAI收割
APPLIED PHYSICS LETTERS, 2022, 卷号: 120
作者:
Cheng, Peng
;
Wang, Yunfeng
;
Ye, Tingting
;
Chu, Lingqiao
;
Yang, Jin
  |  
收藏
  |  
浏览/下载:31/0
  |  
提交时间:2022/12/23