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上海药物研究所 [25]
武汉病毒研究所 [5]
金属研究所 [4]
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期刊论文 [38]
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2025 [5]
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Discovery of 3-(Fluoro-imidazolyl)pyridazine Derivatives as Potent STING Agonists with Antitumor Activity
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 68, 期号: 10, 页码: 9864-9885
作者:
Hou, Hui
;
Zhou, Jingyi
;
Sui, Qibang
;
Zhang, Changfa
;
Su, Zhaoming
  |  
收藏
  |  
浏览/下载:34/0
  |  
提交时间:2025/07/25
Residue-Selective Inhibitors Discovery via Covalent DNA-Encoded Chemical Libraries with Diverse Warheads
期刊论文
OAI收割
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2025, 卷号: 147, 期号: 18, 页码: 15469-15481
作者:
Wu, Xinyuan
;
Pan, Jiayi
;
Fan, Rufeng
;
Zhang, Yiwei
;
Wang, Chao
  |  
收藏
  |  
浏览/下载:41/0
  |  
提交时间:2025/06/23
Proteome-Wide Data Guides the Discovery of Lysine-Targeting Covalent Inhibitors Using DNA-Encoded Chemical Libraries
期刊论文
OAI收割
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2025, 页码: 14
作者:
Wu, Xinyuan
;
Li, Shunyao
;
Liang, Ting
;
Yu, Qing
;
Zhang, Yiwei
  |  
收藏
  |  
浏览/下载:47/0
  |  
提交时间:2025/06/23
Activity-based protein profiling data
Covalent DNA-encoded chemical library
Covalent ligand selection
Lysine-targeting covalent inhibitors
Microstructure evolution and interfacial healing mechanism of heterogeneous interfaces in Ni-Co based superalloys during hot compression bonding
期刊论文
OAI收割
MATERIALS CHARACTERIZATION, 2025, 卷号: 220, 页码: 13
作者:
Ren, Shaofei
;
Xiao, He
;
Wu, Shengqing
;
Zeng, Chenqi
;
Bai, Xiaolong
  |  
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2025/04/27
Hot compression bonding
Bonding interface
Continuous dynamic recrystallization
Necklace-like recrystallization
Interface healing
Design, synthesis, and structure-activity relationship studies of triazolo-pyrimidine derivatives as WRN inhibitors for the treatment of MSI tumors
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 282, 页码: 21
作者:
Sui, Qibang
;
Zhou, Yuanyang
;
Li, Manjia
;
Wang, Dan
  |  
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2024/12/25
Synthetic lethal
MSI tumors
WRN inhibitors
Triazolo-pyrimidine derivatives
Covalent DNA-Encoded Library Workflow Drives Discovery of SARS-CoV-2 Nonstructural Protein Inhibitors
期刊论文
OAI收割
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2024, 页码: 14
作者:
Wang, Xudong
;
Xiong, Liwei
;
Zhu, Ying
;
Liu, Sixiu
;
Zhao, Wenfeng
  |  
收藏
  |  
浏览/下载:78/0
  |  
提交时间:2024/12/25
Enhancing the Predictive Power of Machine Learning Models through a Chemical Space Complementary DEL Screening Strategy
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 页码: 12
作者:
Suo, Yanrui
;
Qian, Xu
;
Xiong, Zhaoping
;
Liu, Xiaohong
;
Wang, Chao
  |  
收藏
  |  
浏览/下载:154/0
  |  
提交时间:2024/11/26
Study on interfacial healing mechanism of a Ni-Co base dual-phase superalloy during hot-compression bonding
期刊论文
OAI收割
MATERIALS & DESIGN, 2024, 卷号: 241, 页码: 13
作者:
Ren, Shaofei
;
Bai, Xiaolong
;
Liu, Sheng
;
Sun, Mingyue
;
Xu, Bin
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收藏
  |  
浏览/下载:1/0
  |  
提交时间:2025/04/27
Hot -compression bonding
Bonding interface
Discontinuous dynamic recrystallization
Heterogeneous epitaxial recrystallization
Interface healing mechanism of fine-grained Ni-Co-based superalloy during hot-compression bonding
期刊论文
OAI收割
JOURNAL OF MATERIALS SCIENCE & TECHNOLOGY, 2024, 卷号: 173, 页码: 45-53
作者:
Ren, Shaofei
;
Bai, Xiaolong
;
Liu, Sheng
;
Sun, Mingyue
;
Xu, Bin
  |  
收藏
  |  
浏览/下载:52/0
  |  
提交时间:2024/01/08
Hot-compression bonding
Ni-Co-based superalloy
Discontinuous dynamic recrystallization
Heterogeneous epitaxial recrystallization
Targeting JMJD1C to selectively disrupt tumor T
reg
cell fitness enhances antitumor immunity
期刊论文
OAI收割
NATURE IMMUNOLOGY, 2024, 页码: 32
作者:
Long, Xuehui
;
Zhang, Sulin
;
Wang, Yuliang
;
Chen, Jingjing
;
Lu, Yanlai
  |  
收藏
  |  
浏览/下载:112/0
  |  
提交时间:2024/03/25