中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [21]
青海盐湖研究所 [11]
上海硅酸盐研究所 [6]
合肥物质科学研究院 [5]
采集方式
OAI收割 [43]
内容类型
期刊论文 [43]
发表日期
2023 [1]
2022 [7]
2021 [9]
2020 [5]
2019 [6]
2018 [7]
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学科主题
Materials ... [1]
Materials ... [1]
Metallurgy... [1]
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Structure-based identification of new orally bioavailable BRD9-PROTACs for treating acute myelocytic leukemia
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 262, 页码: 18
作者:
Zhang, Jingyu
;
Duan, Haiting
;
Gui, Renzhao
;
Wu, Mingfei
;
Shen, Liteng
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2023/12/19
Acute myeloid leukemia
Bromodomain-containing protein 9
Proteolysis-targeting chimera
Orally bioavailable
Docking
Structure-based rational design enables efficient discovery of a new selective and potent AKT PROTAC degrader
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 238, 页码: 15
作者:
Zhu, Cheng-Liang
;
Luo, Xiaomin
;
Tian, Tian
;
Rao, Zijian
;
Wang, Hanlin
  |  
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2022/08/16
AKT
Protein kinase B
PROTAC
Chemical degrader
Rational design
Structural Feature Analyzation Strategies toward Discovery of Orally Bioavailable PROTACs of Bruton's Tyrosine Kinase for the Treatment of Lymphoma
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 65, 期号: 13, 页码: 9096–9125
作者:
Zhang, Jingyu
;
Che, Jinxin
;
Luo, Xiaomin
;
Wu, Mingfei
;
Kan, Weijuan
  |  
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2024/03/21
Design, synthesis and biological evaluation of sulfonamides inhibitors of XPO1 displaying activity against multiple myeloma cells
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 235
作者:
Qu, Bingxue
;
Xu, Yongjin
;
Lu, Yang
;
Zhuang, Weihao
;
Jin, Xinxin
  |  
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2022/12/23
XPO1
Multiple myeloma
MM.1S
N-phenylsulfonamide
Oral administration
Microstructural and mechanical evolution of SiCf/SiC composites in wet oxygen atmosphere above 1000 degrees C
期刊论文
OAI收割
CERAMICS INTERNATIONAL, 2022, 卷号: 48, 期号: 6, 页码: 8473-8480
作者:
Guo, Feiyu
;
Chen, Xiaowu
;
Cheng, Guofeng
;
Wu, Huiyang
;
Zhou, Haijun
  |  
收藏
  |  
浏览/下载:32/0
  |  
提交时间:2022/06/15
Wet-oxygen
SiCf/SiC
Residual stress
Bending strength
Raman spectra
Identification of 2-Aminopyrimidine Derivatives as FLT3 Kinase Inhibitors with High Selectivity over c-KIT
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 65, 期号: 4, 页码: 3229-3248
作者:
Tong, Lexian
;
Wang, Peipei
;
Li, Xuemei
;
Dong, Xiaowu
;
Hu, Xiaobei
  |  
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2022/08/16
Discovery of seneciobipyrrolidine derivatives for the amelioration of glucose homeostasis disorders through 4E-BP1/Akt/AMPK signaling activation
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 228, 页码: 25
作者:
Che, Jinxin
;
Ma, Canliang
;
Lu, Jialiang
;
Chen, Binhui
;
Shi, Qiuqiu
  |  
收藏
  |  
浏览/下载:31/0
  |  
提交时间:2022/06/15
Seneciobipyrrolidine
Phenotypic screening
Glucose homeostasis
Proteomic analysis
L6 myotubes
4E-BP1
High efficacy of PD-1 inhibitor after initial failure of PD-L1 inhibitor in Relapsed/Refractory classical Hodgkin Lymphoma
期刊论文
OAI收割
BMC CANCER, 2022, 卷号: 22
作者:
Chen, Xi
;
Kong, Haiying
;
Luo, Linxiang
;
Han, Shuiyun
;
Lei, Tao
  |  
收藏
  |  
浏览/下载:55/0
  |  
提交时间:2022/02/14
Hodgkin lymphoma
PD-1 inhibitor
PD-L1 inhibitor
PD-L2
Molecular phenotype
Tumor microenvironment
Discover Novel Covalent Inhibitors Targeting FLT3 through Hybrid Virtual Screening Strategy
期刊论文
OAI收割
BIOLOGICAL & PHARMACEUTICAL BULLETIN, 2021, 卷号: 44, 期号: 12, 页码: 1872-1877
作者:
Hu, Shengquan
;
Liu, Jing
;
Chen, Sikang
;
Gao, Jian
;
Zhou, Yubo
  |  
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2022/06/15
acute myeloid leukemia
FMS-like tyrosine kinase 3
CovDock
hybrid virtual screening
autodock
Effects of interfacial residual stress on mechanical behavior of SiCf/SiC composites
期刊论文
OAI收割
JOURNAL OF ADVANCED CERAMICS, 2021, 页码: 11
作者:
Chen, Xiaowu
;
Cheng, Guofeng
;
Yang, Jinshan
;
Hu, Jianbao
;
Liao, Chunjin
  |  
收藏
  |  
浏览/下载:69/0
  |  
提交时间:2021/12/01
ceramic matrix composites
Raman spectroscopy
mechanical properties
residual stress